JP2015505555A5 - - Google Patents
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- Publication number
- JP2015505555A5 JP2015505555A5 JP2014555310A JP2014555310A JP2015505555A5 JP 2015505555 A5 JP2015505555 A5 JP 2015505555A5 JP 2014555310 A JP2014555310 A JP 2014555310A JP 2014555310 A JP2014555310 A JP 2014555310A JP 2015505555 A5 JP2015505555 A5 JP 2015505555A5
- Authority
- JP
- Japan
- Prior art keywords
- inhibition
- cancer
- compound
- protein kinase
- autoimmune disorders
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 206010003816 Autoimmune disease Diseases 0.000 claims 1
- 101700030325 CHKB Proteins 0.000 claims 1
- 102000001253 Protein Kinases Human genes 0.000 claims 1
- 108060006633 Protein Kinases Proteins 0.000 claims 1
- 201000011510 cancer Diseases 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 230000000694 effects Effects 0.000 claims 1
- 230000002401 inhibitory effect Effects 0.000 claims 1
Claims (1)
- プロテインキナーゼまたはＣＨＫ１活性の阻害に対して反応性である状態が、癌および自己免疫障害から選択される、請求項２０〜２２のいずれか一項に記載の化合物または方法。
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB1201566.5A GB201201566D0 (en) | 2012-01-30 | 2012-01-30 | New chemical compounds |
| GB1201566.5 | 2012-01-30 | ||
| PCT/GB2013/050212 WO2013114113A1 (en) | 2012-01-30 | 2013-01-30 | 1h-pyrrolo[2,3-b] pyridine derivatives and their use as kinase inhibitors |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2015505555A JP2015505555A (ja) | 2015-02-23 |
| JP2015505555A5 true JP2015505555A5 (ja) | 2015-11-12 |
| JP6199316B2 JP6199316B2 (ja) | 2017-09-20 |
Family
ID=45876325
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014555310A Active JP6199316B2 (ja) | 2012-01-30 | 2013-01-30 | １Ｈ−ピロロ［２，３−ｂ］ピリジン誘導体およびキナーゼ阻害剤としてのその使用 |
Country Status (21)
| Country | Link |
|---|---|
| US (3) | US10000481B2 (ja) |
| EP (1) | EP2809670B1 (ja) |
| JP (1) | JP6199316B2 (ja) |
| CN (4) | CN104203948A (ja) |
| AU (1) | AU2013213954B2 (ja) |
| BR (1) | BR112014018795B1 (ja) |
| CA (1) | CA2862940C (ja) |
| DK (1) | DK2809670T3 (ja) |
| EA (1) | EA026657B1 (ja) |
| ES (1) | ES2637340T3 (ja) |
| GB (1) | GB201201566D0 (ja) |
| HK (1) | HK1200447A1 (ja) |
| HU (1) | HUE035332T2 (ja) |
| IL (1) | IL233595B (ja) |
| IN (1) | IN2014DN06104A (ja) |
| MX (1) | MX352927B (ja) |
| NZ (1) | NZ627361A (ja) |
| PL (1) | PL2809670T3 (ja) |
| PT (1) | PT2809670T (ja) |
| WO (1) | WO2013114113A1 (ja) |
| ZA (1) | ZA201405070B (ja) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201201566D0 (en) * | 2012-01-30 | 2012-03-14 | Vernalis R&D Ltd | New chemical compounds |
| MY168958A (en) * | 2012-04-23 | 2019-01-28 | Genentech Inc | Intermediates and processes for preparing compounds |
| CN105705499B (zh) * | 2013-08-22 | 2018-10-12 | 基因泰克公司 | 用于制备化合物的方法 |
| CN104829609B (zh) * | 2014-02-11 | 2016-08-03 | 北大方正集团有限公司 | 取代的吡啶并嘧啶化合物及其制备方法和应用 |
| MA41559A (fr) | 2015-09-08 | 2017-12-26 | Taiho Pharmaceutical Co Ltd | Composé de pyrimidine condensé ou un sel de celui-ci |
| US10032914B2 (en) * | 2015-10-20 | 2018-07-24 | Taiwan Semiconductor Manufacturing Co., Ltd. | Semiconductor device and manufacturing method thereof |
| IL261107B2 (en) | 2016-02-23 | 2023-11-01 | Taiho Pharmaceutical Co Ltd | A novel compressed pyrimidine compound or a salt thereof |
| TW202043198A (zh) | 2019-01-17 | 2020-12-01 | 美商Ｉｆｍ Ｄｕｅ有限公司 | 用於治療與sting活性相關之病況的化合物及組合物 |
| CN116261452A (zh) * | 2020-07-15 | 2023-06-13 | 艾福姆德尤股份有限公司 | 用于治疗与sting活性有关的疾病的化合物和组合物 |
| EP4182310A1 (en) | 2020-07-15 | 2023-05-24 | IFM Due, Inc. | Compounds and compositions for treating conditions associated with sting activity |
| TW202216685A (zh) * | 2020-07-15 | 2022-05-01 | 美商Ｉｆｍ Ｄｕｅ有限公司 | 用於治療與sting活性相關的病狀之化合物及組合物 |
| WO2023137034A1 (en) * | 2022-01-12 | 2023-07-20 | Ifm Due, Inc. | Compounds and compositions for treating conditions associated with sting activity |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US1012976A (en) * | 1909-03-25 | 1911-12-26 | Adolf Bordt | Adding-machine. |
| WO2003028724A1 (en) | 2001-10-04 | 2003-04-10 | Smithkline Beecham Corporation | Chk1 kinase inhibitors |
| US7531553B2 (en) * | 2003-03-21 | 2009-05-12 | Amgen Inc. | Heterocyclic compounds and methods of use |
| KR101223914B1 (ko) * | 2003-11-21 | 2013-01-18 | 어레이 바이오파마 인크. | Ａｋｔ 단백질 키나제 억제제 |
| EP2242755B1 (en) * | 2008-01-08 | 2012-09-12 | Array Biopharma, Inc. | Pyrrolopyridines as kinase inhibitors |
| CN101970424B (zh) * | 2008-01-22 | 2013-06-12 | 弗奈利斯（R&D）有限公司 | 具有检测点激酶1抑制活性的吲哚基吡啶酮衍生物 |
| AR071717A1 (es) * | 2008-05-13 | 2010-07-07 | Array Biopharma Inc | Pirrolo[2,3-b]piridinas inhibidoras de quinasas chk1 y chk2,composiciones farmaceuticas que las contienen,proceso para prepararlas y uso de las mismas en el tratamiento y prevencion del cancer. |
| KR20110015699A (ko) | 2008-06-11 | 2011-02-16 | 제넨테크, 인크. | 디아자카르바졸 및 사용 방법 |
| ES2433230T3 (es) * | 2009-08-06 | 2013-12-10 | Merck Patent Gmbh | Compuestos bicíclicos novedosos de urea |
| EP2571361A4 (en) * | 2010-05-19 | 2013-11-13 | Univ North Carolina | PYRAZOLOPYRIMIDINE COMPOUNDS FOR CANCER TREATMENT |
| GB201201566D0 (en) * | 2012-01-30 | 2012-03-14 | Vernalis R&D Ltd | New chemical compounds |
-
2012
- 2012-01-30 GB GBGB1201566.5A patent/GB201201566D0/en not_active Ceased
-
2013
- 2013-01-30 JP JP2014555310A patent/JP6199316B2/ja active Active
- 2013-01-30 BR BR112014018795-9A patent/BR112014018795B1/pt active IP Right Grant
- 2013-01-30 HU HUE13703121A patent/HUE035332T2/en unknown
- 2013-01-30 DK DK13703121.7T patent/DK2809670T3/en active
- 2013-01-30 EP EP13703121.7A patent/EP2809670B1/en active Active
- 2013-01-30 EA EA201491376A patent/EA026657B1/ru not_active IP Right Cessation
- 2013-01-30 CN CN201380014717.5A patent/CN104203948A/zh active Pending
- 2013-01-30 PT PT137031217T patent/PT2809670T/pt unknown
- 2013-01-30 CN CN201610920724.7A patent/CN107011341A/zh active Pending
- 2013-01-30 CA CA2862940A patent/CA2862940C/en active Active
- 2013-01-30 PL PL13703121T patent/PL2809670T3/pl unknown
- 2013-01-30 CN CN201610920720.9A patent/CN106866658B/zh active Active
- 2013-01-30 US US14/375,353 patent/US10000481B2/en active Active
- 2013-01-30 CN CN202010405942.3A patent/CN111484493A/zh active Pending
- 2013-01-30 NZ NZ627361A patent/NZ627361A/en unknown
- 2013-01-30 IN IN6104DEN2014 patent/IN2014DN06104A/en unknown
- 2013-01-30 MX MX2014009112A patent/MX352927B/es active IP Right Grant
- 2013-01-30 ES ES13703121.7T patent/ES2637340T3/es active Active
- 2013-01-30 WO PCT/GB2013/050212 patent/WO2013114113A1/en active Application Filing
- 2013-01-30 AU AU2013213954A patent/AU2013213954B2/en active Active
-
2014
- 2014-07-10 IL IL233595A patent/IL233595B/en active IP Right Grant
- 2014-07-11 ZA ZA2014/05070A patent/ZA201405070B/en unknown
-
2015
- 2015-01-23 HK HK15100794.1A patent/HK1200447A1/xx unknown
-
2018
- 2018-06-15 US US16/009,439 patent/US10889582B2/en active Active
-
2020
- 2020-11-30 US US17/107,176 patent/US20210206762A1/en not_active Abandoned
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