JP2014523851A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2014523851A5 JP2014523851A5 JP2013546480A JP2013546480A JP2014523851A5 JP 2014523851 A5 JP2014523851 A5 JP 2014523851A5 JP 2013546480 A JP2013546480 A JP 2013546480A JP 2013546480 A JP2013546480 A JP 2013546480A JP 2014523851 A5 JP2014523851 A5 JP 2014523851A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- substituted
- optionally substituted
- ring
- alkyl group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2013546480A JP5976011B2 (ja) | 2011-04-05 | 2012-04-05 | スルホンアミド誘導体およびその用途 |
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2011084100 | 2011-04-05 | ||
| JP2011084100 | 2011-04-05 | ||
| JP2013546480A JP5976011B2 (ja) | 2011-04-05 | 2012-04-05 | スルホンアミド誘導体およびその用途 |
| PCT/JP2012/059949 WO2012137982A2 (en) | 2011-04-05 | 2012-04-05 | Sulfonamide derivative and use thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2014523851A JP2014523851A (ja) | 2014-09-18 |
| JP2014523851A5 true JP2014523851A5 (https=) | 2015-05-21 |
| JP5976011B2 JP5976011B2 (ja) | 2016-08-23 |
Family
ID=46028103
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013546480A Active JP5976011B2 (ja) | 2011-04-05 | 2012-04-05 | スルホンアミド誘導体およびその用途 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US9527807B2 (https=) |
| EP (1) | EP2694472B1 (https=) |
| JP (1) | JP5976011B2 (https=) |
| WO (1) | WO2012137982A2 (https=) |
Families Citing this family (53)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6134654B2 (ja) | 2012-02-08 | 2017-05-24 | 武田薬品工業株式会社 | 複素環化合物およびその用途 |
| JO3225B1 (ar) * | 2012-11-27 | 2018-03-08 | Lilly Co Eli | 6-((s)-1-{1-[5-(2-هيدروكسي-إيثوكسي)-بيريدين-2-يل]-1h-بيرازول-3-يل}إيثيل)-3h-1 ، 3-بنزو ثيازول-2- أون باعتباره مضاد مستقبل ampa يعتمد على tarp- جاما 8 |
| EP3122727B1 (en) | 2014-03-24 | 2018-01-31 | Bayer CropScience Aktiengesellschaft | Process for preparing 3,5-bis(haloalkyl)pyrazole derivatives from alpha , alpha-dihaloamines and ketimines |
| EP3015458A1 (en) * | 2014-11-03 | 2016-05-04 | Bayer CropScience AG | Process for preparing 3,5-bis(haloalkyl)pyrazole derivatives from a,a-dihaloamines and ketimines |
| LT3984994T (lt) | 2016-02-04 | 2024-10-10 | Takeda Pharmaceutical Company Limited | Pakeistas piperidino junginys kaip 2 tipo oreksino agonistas narkolepsijai gydyti |
| EP3436021A4 (en) | 2016-03-29 | 2019-11-06 | RespireRx Pharmaceuticals Inc. | COMPOSITIONS AND METHODS FOR TREATING ATTENTION DEFICIT DISORDER |
| AR108838A1 (es) | 2016-06-21 | 2018-10-03 | Bristol Myers Squibb Co | Ácidos de carbamoiloximetil triazol ciclohexilo como antagonistas de lpa |
| US11059780B2 (en) | 2017-03-08 | 2021-07-13 | Takeda Pharmaceutical Company Limited | Substituted pyrrolidine compound and use thereof |
| JP7012703B2 (ja) | 2017-03-08 | 2022-02-14 | 武田薬品工業株式会社 | 置換ピロリジン化合物およびその用途 |
| WO2019027003A1 (ja) * | 2017-08-03 | 2019-02-07 | 武田薬品工業株式会社 | 複素環化合物およびその用途 |
| US10428023B2 (en) | 2017-08-03 | 2019-10-01 | Takeda Pharmaceutical Company Limited | Heterocyclic compound and use thereof |
| EP3693360B1 (en) | 2017-10-06 | 2023-12-13 | Takeda Pharmaceutical Company Limited | Heterocyclic compounds |
| ES2970624T3 (es) | 2017-10-06 | 2024-05-29 | Takeda Pharmaceuticals Co | Compuesto heterocíclico |
| EP4011875A1 (en) | 2017-12-19 | 2022-06-15 | Bristol-Myers Squibb Company | Triazole n-linked carbamoyl cyclohexyl acids as lpa antagonists |
| US11447475B2 (en) | 2017-12-19 | 2022-09-20 | Bristol-Myers Squibb Company | Isoxazole N-linked carbamoyl cyclohexyl acids as LPA antagonists |
| US11180488B2 (en) | 2017-12-19 | 2021-11-23 | Bristol-Myers Squibb Company | Isoxazole o-linked carbamoyl cyclohexyl acids as LPA antagonists |
| EA202091505A1 (ru) | 2017-12-19 | 2020-09-22 | Бристол-Маерс Сквибб Компани | Триазолазолы циклогексильной кислоты в качестве антагонистов lpa |
| KR102756639B1 (ko) | 2017-12-19 | 2025-01-16 | 브리스톨-마이어스 스큅 컴퍼니 | Lpa 길항제로서의 시클로헥실 산 이속사졸 아졸 |
| KR102777148B1 (ko) | 2017-12-19 | 2025-03-05 | 브리스톨-마이어스 스큅 컴퍼니 | Lpa 길항제로서의 시클로헥실 산 트리아졸 아진 |
| EP3728209B1 (en) | 2017-12-19 | 2025-12-24 | Bristol-Myers Squibb Company | Cyclohexyl acid isoxazole azines as lpa antagonists |
| EA039459B1 (ru) * | 2017-12-25 | 2022-01-28 | Такеда Фармасьютикал Компани Лимитед | Гетероциклическое соединение и его применение в качестве средства для лечения заболеваний, связанных с рецептором орексина 2 типа |
| KR20200132858A (ko) * | 2018-03-20 | 2020-11-25 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 간질 치료제 |
| WO2020004537A1 (ja) | 2018-06-29 | 2020-01-02 | 武田薬品工業株式会社 | 複素環化合物およびその用途 |
| JP7339250B2 (ja) | 2018-06-29 | 2023-09-05 | 武田薬品工業株式会社 | 複素環化合物およびその用途 |
| US20220041572A1 (en) | 2018-09-18 | 2022-02-10 | Bristol-Myers Squibb Company | Cycloheptyl acids as lpa antagonists |
| ES2946657T3 (es) | 2018-09-18 | 2023-07-24 | Bristol Myers Squibb Co | Acidos ciclopentílicos como antagonistas de LPA |
| EP3896060B1 (en) | 2018-12-12 | 2023-08-16 | Takeda Pharmaceutical Company Limited | Heterocyclic compound |
| US12071434B2 (en) | 2018-12-12 | 2024-08-27 | Takeda Pharmaceutical Company Limited | Heterocyclic compound |
| JP7253640B2 (ja) * | 2019-01-31 | 2023-04-06 | 武田薬品工業株式会社 | 複素環化合物およびその用途 |
| US11098029B2 (en) | 2019-02-13 | 2021-08-24 | Merck Sharp & Dohme Corp. | 5-alkyl pyrrolidine orexin receptor agonists |
| WO2020167701A1 (en) | 2019-02-13 | 2020-08-20 | Merck Sharp & Dohme Corp. | Pyrrolidine orexin receptor agonists |
| CN114599648A (zh) | 2019-06-18 | 2022-06-07 | 百时美施贵宝公司 | 作为lpa拮抗剂的三唑羧酸 |
| EP3986553B1 (en) | 2019-06-18 | 2026-03-25 | Bristol-Myers Squibb Company | Cyclobutyl carboxylic acids as lpa antagonists |
| KR20220024549A (ko) | 2019-06-18 | 2022-03-03 | 브리스톨-마이어스 스큅 컴퍼니 | Lpa 길항제로서의 이속사졸 카르복실산 |
| US12312332B2 (en) | 2019-08-08 | 2025-05-27 | Merck Sharp & Dohme Llc | Heteroaryl pyrrolidine and piperidine orexin receptor agonists |
| EP4065585B1 (en) | 2019-11-25 | 2025-08-20 | Alkermes, Inc. | Substituted macrocyclic compounds and related methods of treatment |
| US12448377B2 (en) | 2019-11-27 | 2025-10-21 | Takeda Pharmaceutical Company Limited | Heterocyclic compound |
| BR112023002957A2 (pt) | 2020-08-18 | 2023-04-04 | Merck Sharp & Dohme Llc | Composto, composição farmacêutica, e, métodos para tratar narcolepsia e para tratar hipersonia em um sujeito mamífero |
| US11760747B2 (en) * | 2020-12-21 | 2023-09-19 | Alkermes, Inc. | Substituted piperidino compounds and related methods of treatment |
| US12006330B2 (en) | 2020-12-21 | 2024-06-11 | Alkermes, Inc. | Substituted macrocyclic compounds and related methods of treatment |
| IL315808A (en) | 2022-03-28 | 2024-11-01 | Bayer Ag | Process for preparing cis-4-aminotetrahydrofuran-2-carboxylic esters |
| WO2023199091A1 (en) | 2022-04-12 | 2023-10-19 | Takeda Pharmaceutical Company Limited | Heterocyclic compound |
| WO2023249871A1 (en) * | 2022-06-21 | 2023-12-28 | Alkermes, Inc. | Substituted pyrrolidinyl and piperidinyl compounds and related methods of treatment |
| JP2025521507A (ja) * | 2022-06-21 | 2025-07-10 | アルカームス インコーポレーテッド | 置換縮合二環式化合物および関連する治療方法 |
| CA3260225A1 (en) * | 2022-06-21 | 2023-12-28 | Alkermes, Inc. | Fused, Substituted Bicyclic Compounds and Associated Treatment Methods |
| TW202409023A (zh) | 2022-07-14 | 2024-03-01 | 美商富曼西公司 | 除草苯并𠯤 |
| CN115433102B (zh) * | 2022-10-16 | 2024-02-27 | 大连双硼医药化工有限公司 | 一种反式-(1r,2r)-2-氨基环己烷羧酸乙酯盐酸盐的制备方法 |
| TW202428580A (zh) | 2022-10-31 | 2024-07-16 | 日商武田藥品工業股份有限公司 | 雜環化合物 |
| AR131202A1 (es) | 2022-11-30 | 2025-02-26 | Takeda Pharmaceuticals Co | Compuesto heterocíclico y uso del mismo |
| PE20252742A1 (es) | 2023-03-16 | 2025-12-05 | Takeda Pharmaceuticals Co | Compuestos heterociclicos macrociclicos y sus usos |
| WO2025111184A1 (en) | 2023-11-21 | 2025-05-30 | Fmc Corporation | Substituted tetrahydroquinoline and tetrahydroquinoxaline herbicides |
| WO2025229494A1 (en) | 2024-04-29 | 2025-11-06 | Takeda Pharmaceutical Company Limited | Heterocyclic compound |
| WO2025229495A1 (en) | 2024-04-29 | 2025-11-06 | Takeda Pharmaceutical Company Limited | Heterocyclic compound |
Family Cites Families (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2765322A (en) | 1953-03-03 | 1956-10-02 | Rohm & Haas | Preparation of bis(4-glycidyloxyphenyl)-sulfone |
| US5315013A (en) | 1988-01-07 | 1994-05-24 | E. I. Du Pont De Nemours And Company | Substituted pyrazole angiotensin II antagonists |
| KR100338855B1 (ko) | 1996-07-31 | 2002-12-28 | 시오노기세이야쿠가부시키가이샤 | 신규 파라테르페닐 화합물 |
| DE19803396A1 (de) | 1998-01-29 | 1999-08-05 | Bayer Ag | Substituierte Phenyluracile |
| US6902847B1 (en) | 1998-05-20 | 2005-06-07 | Osaka Gas Company Limited | Non-aqueous secondary cell and method for controlling the same |
| ES2230864T3 (es) * | 1998-07-24 | 2005-05-01 | Teijin Limited | Derivados del acido antranilico. |
| BR0012068A (pt) | 1999-06-30 | 2002-05-14 | Daiichi Seiyaku Co | Compostos inibidores de vla-4 |
| TWI262917B (en) | 2002-02-01 | 2006-10-01 | Dainippon Sumitomo Pharma Co | 2-Furancarboxylic hydrazides and pharmaceutical compositions containing the same |
| JP2003238538A (ja) | 2002-02-12 | 2003-08-27 | Nippon Nohyaku Co Ltd | 新規4−置換フェニル−5−ハロピリミジン誘導体及びこれを有効成分とする除草剤 |
| JP2005060385A (ja) | 2003-07-31 | 2005-03-10 | Dainippon Pharmaceut Co Ltd | 2−フランカルボン酸ヒドラジド化合物からなる医薬 |
| GB0417709D0 (en) | 2004-08-09 | 2004-09-08 | Glaxo Group Ltd | Compounds |
| WO2006015827A1 (en) | 2004-08-09 | 2006-02-16 | Glaxo Group Limited | Compounds which potentiate glutamate receptor and uses thereof in medicine |
| KR20070050070A (ko) | 2004-08-09 | 2007-05-14 | 글락소 그룹 리미티드 | 글루타메이트 수용체를 강화시키는 화합물 및 의약에서의그의 용도 |
| EP1849465A4 (en) | 2005-02-18 | 2008-12-24 | Takeda Pharmaceutical | AGENS TO CONTROL THE FUNCTION OF THE GPR34 RECEPTOR |
| UA92007C2 (ru) | 2005-05-04 | 2010-09-27 | Н.В. Органон | Производные 4-фенил-5-оксо-1,4,5,6,7,8-гексагидрохинолина для лечения бесплодности |
| DE602006003661D1 (de) | 2005-06-06 | 2008-12-24 | Lilly Co Eli | Ampa-rezeptoren-verstärker |
| AU2006265639A1 (en) | 2005-07-01 | 2007-01-11 | Jenrin Discovery | MAO-B inhibitors useful for treating obesity |
| JP5014334B2 (ja) * | 2005-10-06 | 2012-08-29 | イーライ リリー アンド カンパニー | Ampa受容体増強剤 |
| JP2010517926A (ja) | 2006-02-08 | 2010-05-27 | グラクソ グループ リミテッド | グルタミン酸受容体を増強する、統合失調症の治療に有用な4−フェニル−3−(2−プロピルスルホニルアミノ)テトラヒドロフラン誘導体 |
| GB0602560D0 (en) | 2006-02-08 | 2006-03-22 | Glaxo Group Ltd | Compounds |
| US8097652B2 (en) | 2006-12-11 | 2012-01-17 | Eli Lilly And Company | AMPA receptor potentiators |
| WO2008113795A1 (en) | 2007-03-20 | 2008-09-25 | Glaxo Group Limited | Compounds which potentiate ampa receptor and uses thereof in medicine |
| EP2142505A1 (en) | 2007-04-03 | 2010-01-13 | Pfizer, Inc. | Sulfonamides and pharmaceutical compositions thereof |
| AR069781A1 (es) | 2007-12-19 | 2010-02-17 | Glaxo Group Ltd | Compuestos de n-(2,3-dihidro-inden-2-il) propanosulfonamida, composicion farmaceutica que los comprenden y su uso para el tratamiento de la ezquizofrenia. |
| GB0801265D0 (en) | 2008-01-23 | 2008-02-27 | Glaxo Group Ltd | Compounds |
| GB0801220D0 (en) | 2008-01-23 | 2008-02-27 | Glaxo Group Ltd | Compounds |
| WO2009119088A1 (ja) | 2008-03-25 | 2009-10-01 | 武田薬品工業株式会社 | 複素環化合物 |
| TW201012803A (en) * | 2008-06-06 | 2010-04-01 | Organon Nv | Heterocyclic derivatives |
| CA2739559A1 (en) | 2008-10-08 | 2010-04-15 | Pfizer Inc. | Tetrahydrofuranyl sulfonamides and pharmaceutical compositions thereof |
| EP2417101B1 (en) * | 2009-04-09 | 2013-10-23 | Merck Sharp & Dohme B.V. | Indane derivatives |
| AP3066A (en) * | 2009-06-26 | 2014-12-31 | Pfizer | Heterocyclic sulfonamides, uses and pharmaceuticalcompositions thereof |
| RU2012106426A (ru) | 2009-07-23 | 2013-08-27 | Новартис Аг | 1н-хиназолин-2,4-дионы, предназначенные для лечения нейронного восковидного липофусциноза |
| LT2603513T (lt) | 2010-08-10 | 2020-05-25 | Takeda Pharmaceutical Company Limited | Heterociklinis junginys ir jo panaudojimas kaip ampa receptoriaus teigiamo alosterinio moduliatoriaus |
-
2012
- 2012-04-05 EP EP12719088.2A patent/EP2694472B1/en active Active
- 2012-04-05 JP JP2013546480A patent/JP5976011B2/ja active Active
- 2012-04-05 US US14/009,456 patent/US9527807B2/en active Active
- 2012-04-05 WO PCT/JP2012/059949 patent/WO2012137982A2/en not_active Ceased
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2014523851A5 (https=) | ||
| JP2013528204A5 (https=) | ||
| DK1700856T3 (en) | thiazole | |
| JP2018524390A5 (https=) | ||
| JP2015500861A5 (https=) | ||
| JP2017502940A5 (https=) | ||
| AU2018236691A1 (en) | N-acyl-n'-(pyridin-2-yl) ureas and analogs exhibiting anti-cancer and anti-proliferative activities | |
| CN109963854A (zh) | 杂芳基并[4,3-c]嘧啶-5-胺类衍生物、其制备方法及其在医药上的应用 | |
| JP2014526435A5 (https=) | ||
| JP2016515560A5 (https=) | ||
| HRP20201171T1 (hr) | Derivati izoindolin-1-ona kao modulatori aktivnosti pozitivnog alosternog modulatora kolinergijskog muskarinskog m1 receptora za liječenje alzheimerove bolesti | |
| JP2014530900A5 (https=) | ||
| RU2019132212A (ru) | Селективные ингибиторы hdac6 | |
| JP2014511891A5 (https=) | ||
| JP2014507455A5 (https=) | ||
| JP2014534981A5 (https=) | ||
| AR092045A1 (es) | Combinaciones farmaceuticas | |
| JP2014518544A5 (https=) | ||
| JP2016514117A5 (https=) | ||
| RU2015101102A (ru) | Гетероароматическое метильное производное циклического амина | |
| RU2017120217A (ru) | 2-амино-5,5-дифтор-6-(фторметил)-6-фенил-3,4,5,6-тетрагидпропиридины в качестве ингибиторов bace1 | |
| JP2016523260A5 (https=) | ||
| RU2014115290A (ru) | Производные 1-фенил 2-пиридинилалкиловых спиртов в качестве ингибиторов | |
| JP2019510794A5 (https=) | ||
| JP2017509676A5 (https=) |