JP2014503534A5 - - Google Patents

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Publication number
JP2014503534A5
JP2014503534A5 JP2013544730A JP2013544730A JP2014503534A5 JP 2014503534 A5 JP2014503534 A5 JP 2014503534A5 JP 2013544730 A JP2013544730 A JP 2013544730A JP 2013544730 A JP2013544730 A JP 2013544730A JP 2014503534 A5 JP2014503534 A5 JP 2014503534A5
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JP
Japan
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alkyl
alkylene
halo
phenyl
och
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JP2013544730A
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English (en)
Japanese (ja)
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JP2014503534A (ja
JP5944921B2 (ja
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Priority claimed from PCT/US2011/064829 external-priority patent/WO2012082853A1/en
Publication of JP2014503534A publication Critical patent/JP2014503534A/ja
Publication of JP2014503534A5 publication Critical patent/JP2014503534A5/ja
Application granted granted Critical
Publication of JP5944921B2 publication Critical patent/JP5944921B2/ja
Expired - Fee Related legal-status Critical Current
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JP2013544730A 2010-12-15 2011-12-14 ネプリライシン阻害剤 Expired - Fee Related JP5944921B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US42318010P 2010-12-15 2010-12-15
US61/423,180 2010-12-15
PCT/US2011/064829 WO2012082853A1 (en) 2010-12-15 2011-12-14 Neprilysin inhibitors

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2015186389A Division JP2016028089A (ja) 2010-12-15 2015-09-24 ネプリライシン阻害剤

Publications (3)

Publication Number Publication Date
JP2014503534A JP2014503534A (ja) 2014-02-13
JP2014503534A5 true JP2014503534A5 (https=) 2014-11-20
JP5944921B2 JP5944921B2 (ja) 2016-07-05

Family

ID=45478501

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JP2013544730A Expired - Fee Related JP5944921B2 (ja) 2010-12-15 2011-12-14 ネプリライシン阻害剤
JP2015186389A Withdrawn JP2016028089A (ja) 2010-12-15 2015-09-24 ネプリライシン阻害剤

Family Applications After (1)

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JP2015186389A Withdrawn JP2016028089A (ja) 2010-12-15 2015-09-24 ネプリライシン阻害剤

Country Status (28)

Country Link
US (9) US8586536B2 (https=)
EP (1) EP2651896B1 (https=)
JP (2) JP5944921B2 (https=)
KR (1) KR101892500B1 (https=)
CN (2) CN103261164B (https=)
AU (1) AU2011343899B2 (https=)
BR (1) BR112013016595B1 (https=)
CA (1) CA2817368C (https=)
CO (1) CO6741228A2 (https=)
DK (1) DK2651896T3 (https=)
ES (1) ES2550324T3 (https=)
HR (1) HRP20151115T1 (https=)
HU (1) HUE028051T2 (https=)
IL (1) IL226327A (https=)
ME (1) ME02295B (https=)
MX (1) MX2013006805A (https=)
MY (1) MY170935A (https=)
NZ (1) NZ610983A (https=)
PH (1) PH12013501240A1 (https=)
PL (1) PL2651896T3 (https=)
PT (1) PT2651896E (https=)
RS (1) RS54348B1 (https=)
RU (1) RU2622288C2 (https=)
SG (2) SG190432A1 (https=)
SI (1) SI2651896T1 (https=)
SM (1) SMT201500271B (https=)
WO (1) WO2012082853A1 (https=)
ZA (1) ZA201304205B (https=)

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KR101854874B1 (ko) 2011-02-17 2018-05-04 세라밴스 바이오파마 알앤디 아이피, 엘엘씨 네프릴리신 억제제로서 치환된 아미노부티릭 유도체
JP5959066B2 (ja) 2011-02-17 2016-08-02 セラヴァンス バイオファーマ アール＆ディー アイピー， エルエルシー ネプリライシン阻害剤としての置換アミノ酪酸誘導体
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ES2653215T3 (es) 2011-05-31 2018-02-06 Theravance Biopharma R&D Ip, Llc Inhibidores de neprilisina
JP5959075B2 (ja) 2011-05-31 2016-08-02 セラヴァンス バイオファーマ アール＆ディー アイピー， エルエルシー ネプリライシン阻害剤
TWI560172B (en) 2011-11-02 2016-12-01 Theravance Biopharma R&D Ip Llc Neprilysin inhibitors
ES2609810T3 (es) 2012-05-31 2017-04-24 Theravance Biopharma R&D Ip, Llc Inhibidores de neprilisina donadores de óxido nítrico
CN104470521B (zh) 2012-06-08 2017-04-12 施万生物制药研发Ip有限责任公司 脑啡肽酶抑制剂
MX356260B (es) 2012-06-08 2018-05-21 Theravance Biopharma R&D Ip Llc Inhibidores de la neprilisina.
MX366149B (es) 2012-08-08 2019-06-28 Theravance Biopharma R&D Ip Llc Inhibidores de neprilisina.

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