JP2013528597A5 - - Google Patents

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Publication number
JP2013528597A5
JP2013528597A5 JP2013509549A JP2013509549A JP2013528597A5 JP 2013528597 A5 JP2013528597 A5 JP 2013528597A5 JP 2013509549 A JP2013509549 A JP 2013509549A JP 2013509549 A JP2013509549 A JP 2013509549A JP 2013528597 A5 JP2013528597 A5 JP 2013528597A5
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Japan
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treatment
pain
hereinafter
disorders
inflammatory diseases
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JP2013509549A
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Japanese (ja)
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JP5646736B2 (ja
JP2013528597A (ja
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Priority claimed from PCT/EP2011/057550 external-priority patent/WO2011141477A1/en
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Publication of JP2013528597A5 publication Critical patent/JP2013528597A5/ja
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JP2013509549A 2010-05-12 2011-05-10 新規ｃｃｒ２受容体アンタゴニスト、これらの製造方法、及び薬物としてのこれらの使用 Active JP5646736B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP10162627.3 2010-05-12
EP10162627 2010-05-12
PCT/EP2011/057550 WO2011141477A1 (en) 2010-05-12 2011-05-10 New ccr2 receptor antagonists, method for producing the same, and use thereof as medicaments

Publications (3)

Publication Number Publication Date
JP2013528597A JP2013528597A (ja) 2013-07-11
JP2013528597A5 true JP2013528597A5 (https=) 2014-11-06
JP5646736B2 JP5646736B2 (ja) 2014-12-24

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JP2013509549A Active JP5646736B2 (ja) 2010-05-12 2011-05-10 新規ｃｃｒ２受容体アンタゴニスト、これらの製造方法、及び薬物としてのこれらの使用

Country Status (4)

Country Link
US (1) US8946218B2 (https=)
EP (1) EP2569295B1 (https=)
JP (1) JP5646736B2 (https=)
WO (1) WO2011141477A1 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2687931C (en) 2007-05-31 2016-05-24 Boehringer Ingelheim International Gmbh Ccr2 receptor antagonists and uses thereof
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EP2569298B1 (en) 2010-05-12 2015-11-25 Boehringer Ingelheim International GmbH Novel ccr2 receptor antagonists, method for producing the same, and use thereof as medicaments
WO2011141477A1 (en) 2010-05-12 2011-11-17 Boehringer Ingelheim International Gmbh New ccr2 receptor antagonists, method for producing the same, and use thereof as medicaments
WO2011144501A1 (en) 2010-05-17 2011-11-24 Boehringer Ingelheim International Gmbh Ccr2 antagonists and uses thereof
EP2576542B1 (en) 2010-05-25 2015-04-22 Boehringer Ingelheim International GmbH Cyclic amide derivatives of pyridazine-3-carboxylic acids and their use in the treatment of pulmonary, pain, immune related and cardiovascular diseases
EP2576538B1 (en) 2010-06-01 2015-10-28 Boehringer Ingelheim International GmbH New CCR2 antagonists
EP2731941B1 (en) * 2011-07-15 2019-05-08 Boehringer Ingelheim International GmbH Novel and selective ccr2 antagonists
MX383744B (es) 2015-07-02 2025-03-14 Centrexion Therapeutics Corp Citrato de (4-((3r,4r)-3-metoxitetrahidro-piran-4-ilamino)piperidin-1-il) (5-metil-6-(((2r, 6s)-6-(p-tolil)tetrahidro-2h-piran-2-il) metilamino) pirimidin-4-il) metanona.
IL302553A (en) * 2020-11-05 2023-07-01 Icahn School Med Mount Sinai Cxcr1/cxcr2 inhibitors for use in treating myelofibrosis

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EP2731941B1 (en) 2011-07-15 2019-05-08 Boehringer Ingelheim International GmbH Novel and selective ccr2 antagonists

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