JP2013526507A5 - - Google Patents
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- JP2013526507A5 JP2013526507A5 JP2013509548A JP2013509548A JP2013526507A5 JP 2013526507 A5 JP2013526507 A5 JP 2013526507A5 JP 2013509548 A JP2013509548 A JP 2013509548A JP 2013509548 A JP2013509548 A JP 2013509548A JP 2013526507 A5 JP2013526507 A5 JP 2013526507A5
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- treatment
- pain
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- disorders
- inflammatory diseases
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10162629 | 2010-05-12 | ||
| EP10162629.9 | 2010-05-12 | ||
| PCT/EP2011/057545 WO2011141474A1 (en) | 2010-05-12 | 2011-05-10 | Novel ccr2 receptor antagonists, method for producing the same, and use thereof as medicaments |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015120556A Division JP5796266B1 (ja) | 2010-05-12 | 2015-06-15 | 新規ｃｃｒ２受容体アンタゴニスト、その製造方法及び薬物としてのその使用 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013526507A JP2013526507A (ja) | 2013-06-24 |
| JP2013526507A5 true JP2013526507A5 (https=) | 2014-11-06 |
Family
ID=42782240
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013509548A Withdrawn JP2013526507A (ja) | 2010-05-12 | 2011-05-10 | 新規ｃｃｒ２受容体アンタゴニスト、その製造方法及び薬物としてのその使用 |
| JP2015120556A Active JP5796266B1 (ja) | 2010-05-12 | 2015-06-15 | 新規ｃｃｒ２受容体アンタゴニスト、その製造方法及び薬物としてのその使用 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015120556A Active JP5796266B1 (ja) | 2010-05-12 | 2015-06-15 | 新規ｃｃｒ２受容体アンタゴニスト、その製造方法及び薬物としてのその使用 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US8877745B2 (https=) |
| EP (1) | EP2569298B1 (https=) |
| JP (2) | JP2013526507A (https=) |
| WO (1) | WO2011141474A1 (https=) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2687931C (en) | 2007-05-31 | 2016-05-24 | Boehringer Ingelheim International Gmbh | Ccr2 receptor antagonists and uses thereof |
| HUE025547T2 (en) | 2008-12-19 | 2016-02-29 | Boehringer Ingelheim Int | Cyclic pyrimidine-4-carboxamides as CCR2 receptor antagonists for the treatment of inflammation, asthma and COPD |
| ES2674275T3 (es) | 2009-12-17 | 2018-06-28 | Centrexion Therapeutics Corporation | Antagonistas del receptor CCR2 y usos de los mismos |
| WO2011141477A1 (en) | 2010-05-12 | 2011-11-17 | Boehringer Ingelheim International Gmbh | New ccr2 receptor antagonists, method for producing the same, and use thereof as medicaments |
| EP2569298B1 (en) | 2010-05-12 | 2015-11-25 | Boehringer Ingelheim International GmbH | Novel ccr2 receptor antagonists, method for producing the same, and use thereof as medicaments |
| WO2011144501A1 (en) | 2010-05-17 | 2011-11-24 | Boehringer Ingelheim International Gmbh | Ccr2 antagonists and uses thereof |
| EP2576542B1 (en) | 2010-05-25 | 2015-04-22 | Boehringer Ingelheim International GmbH | Cyclic amide derivatives of pyridazine-3-carboxylic acids and their use in the treatment of pulmonary, pain, immune related and cardiovascular diseases |
| EP2576538B1 (en) | 2010-06-01 | 2015-10-28 | Boehringer Ingelheim International GmbH | New CCR2 antagonists |
| EP2731941B1 (en) | 2011-07-15 | 2019-05-08 | Boehringer Ingelheim International GmbH | Novel and selective ccr2 antagonists |
| WO2013030665A1 (en) * | 2011-09-02 | 2013-03-07 | Purdue Pharma L.P. | Pyrimidines as sodium channel blockers |
| EP3071559B1 (en) * | 2013-11-18 | 2018-01-10 | Elanco Tiergesundheit AG | (hetero)arylamides for controlling endoparasites |
| US10738026B2 (en) | 2014-02-12 | 2020-08-11 | Purdue Pharma L.P. | Isoquinoline derivatives and use thereof |
| ES2746839T3 (es) * | 2014-12-18 | 2020-03-09 | Pfizer | Derivados de pirimidina y triazina y su uso como inhibidores de AXL |
| ES2904252T3 (es) * | 2015-05-21 | 2022-04-04 | Chemocentryx Inc | Moduladores de CCR2 |
| MX383744B (es) | 2015-07-02 | 2025-03-14 | Centrexion Therapeutics Corp | Citrato de (4-((3r,4r)-3-metoxitetrahidro-piran-4-ilamino)piperidin-1-il) (5-metil-6-(((2r, 6s)-6-(p-tolil)tetrahidro-2h-piran-2-il) metilamino) pirimidin-4-il) metanona. |
| CN105560234A (zh) * | 2016-02-18 | 2016-05-11 | 郑海英 | 一种治疗口腔颌面炎症的药物组合物 |
| CN118267479A (zh) | 2017-09-25 | 2024-07-02 | 凯莫森特里克斯股份有限公司 | 使用趋化因子受体2(ccr2)拮抗剂和pd-1/pd-l1抑制剂的联合治疗 |
| US20190269664A1 (en) | 2018-01-08 | 2019-09-05 | Chemocentryx, Inc. | Methods of treating solid tumors with ccr2 antagonists |
| IL275898B2 (en) | 2018-01-08 | 2025-05-01 | Chemocentryx Inc | Methods for treating solid tumors with CCR2 antagonists |
| CN110872302B (zh) * | 2018-08-31 | 2022-09-27 | 沈阳中化农药化工研发有限公司 | 含嘧啶的螺环类化合物及其用途 |
| WO2024015761A2 (en) * | 2022-07-11 | 2024-01-18 | Rutgers, The State University Of New Jersey | Gαlpha12 inhibitors and methods using same |
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| CA2705405A1 (en) | 2007-11-22 | 2009-05-28 | Boehringer Ingelheim International Gmbh | New compounds |
| EP2062889A1 (de) | 2007-11-22 | 2009-05-27 | Boehringer Ingelheim Pharma GmbH & Co. KG | Verbindungen |
| EP2297137A1 (en) | 2008-06-18 | 2011-03-23 | F. Hoffmann-La Roche AG | Novel heteroaryl carboxamide derivatives |
| JP5693452B2 (ja) | 2008-08-04 | 2015-04-01 | シーエイチディーアイ ファウンデーション，インコーポレーテッド | 特定のキヌレニン−３−モノオキシゲナーゼインヒビター、医薬組成物およびそれらの使用方法 |
| GB0815369D0 (en) | 2008-08-22 | 2008-10-01 | Summit Corp Plc | Compounds for treatment of duchenne muscular dystrophy |
| AU2009289378A1 (en) | 2008-09-02 | 2010-03-11 | Boehringer Ingelheim International Gmbh | Novel benzamides, production thereof, and use thereof as medicaments |
| HUE025547T2 (en) * | 2008-12-19 | 2016-02-29 | Boehringer Ingelheim Int | Cyclic pyrimidine-4-carboxamides as CCR2 receptor antagonists for the treatment of inflammation, asthma and COPD |
| CA2750635A1 (en) | 2009-02-23 | 2010-08-26 | Merck Canada Inc. | Heterocyclic derivatives as inhibitors of stearoyl-coenzyme a delta-9 desaturase |
| US20130143905A1 (en) | 2009-12-17 | 2013-06-06 | Boehringer Ingelheim International Gmbh | Novel antagonists for ccr2 and uses thereof |
| ES2674275T3 (es) | 2009-12-17 | 2018-06-28 | Centrexion Therapeutics Corporation | Antagonistas del receptor CCR2 y usos de los mismos |
| EP2569298B1 (en) | 2010-05-12 | 2015-11-25 | Boehringer Ingelheim International GmbH | Novel ccr2 receptor antagonists, method for producing the same, and use thereof as medicaments |
| WO2011141477A1 (en) | 2010-05-12 | 2011-11-17 | Boehringer Ingelheim International Gmbh | New ccr2 receptor antagonists, method for producing the same, and use thereof as medicaments |
| WO2011144501A1 (en) | 2010-05-17 | 2011-11-24 | Boehringer Ingelheim International Gmbh | Ccr2 antagonists and uses thereof |
| EP2576542B1 (en) | 2010-05-25 | 2015-04-22 | Boehringer Ingelheim International GmbH | Cyclic amide derivatives of pyridazine-3-carboxylic acids and their use in the treatment of pulmonary, pain, immune related and cardiovascular diseases |
| EP2576538B1 (en) | 2010-06-01 | 2015-10-28 | Boehringer Ingelheim International GmbH | New CCR2 antagonists |
| JP5786257B2 (ja) | 2011-06-16 | 2015-09-30 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 新規の選択的ｃｃｒ２拮抗薬 |
| EP2731941B1 (en) | 2011-07-15 | 2019-05-08 | Boehringer Ingelheim International GmbH | Novel and selective ccr2 antagonists |
-
2011
- 2011-05-10 EP EP11719249.2A patent/EP2569298B1/en active Active
- 2011-05-10 WO PCT/EP2011/057545 patent/WO2011141474A1/en not_active Ceased
- 2011-05-10 JP JP2013509548A patent/JP2013526507A/ja not_active Withdrawn
- 2011-05-10 US US13/696,859 patent/US8877745B2/en active Active
-
2015
- 2015-06-15 JP JP2015120556A patent/JP5796266B1/ja active Active
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