JP2013523621A5 - - Google Patents

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Publication number
JP2013523621A5
JP2013523621A5 JP2013500538A JP2013500538A JP2013523621A5 JP 2013523621 A5 JP2013523621 A5 JP 2013523621A5 JP 2013500538 A JP2013500538 A JP 2013500538A JP 2013500538 A JP2013500538 A JP 2013500538A JP 2013523621 A5 JP2013523621 A5 JP 2013523621A5
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JP
Japan
Prior art keywords
compound
formula
iii
precursor compound
precursor
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JP2013500538A
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English (en)
Japanese (ja)
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JP5830519B2 (ja
JP2013523621A (ja
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Publication date
Priority claimed from PCT/EP2010/053998 external-priority patent/WO2010109007A2/en
Priority claimed from GBGB1015203.1A external-priority patent/GB201015203D0/en
Application filed filed Critical
Priority claimed from PCT/EP2011/054744 external-priority patent/WO2011117421A1/en
Publication of JP2013523621A publication Critical patent/JP2013523621A/ja
Publication of JP2013523621A5 publication Critical patent/JP2013523621A5/ja
Application granted granted Critical
Publication of JP5830519B2 publication Critical patent/JP5830519B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2013500538A 2010-03-26 2011-03-28 Pbrリガンドとしての三環式インドール誘導体 Active JP5830519B2 (ja)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
EPPCT/EP2010/053998 2010-03-26
PCT/EP2010/053998 WO2010109007A2 (en) 2009-03-27 2010-03-26 Indole derivatives
IN1824/DEL/2010 2010-08-02
IN1824DE2010 2010-08-02
GBGB1015203.1A GB201015203D0 (en) 2010-03-26 2010-09-13 Active enantiomer
GB1015203.1 2010-09-13
US12/880,218 2010-09-13
US12/880,218 US8501153B2 (en) 2009-03-27 2010-09-13 Active enantiomer
PCT/EP2011/054744 WO2011117421A1 (en) 2010-03-26 2011-03-28 Tricyclic indole derivatives as pbr ligands

Publications (3)

Publication Number Publication Date
JP2013523621A JP2013523621A (ja) 2013-06-17
JP2013523621A5 true JP2013523621A5 (https=) 2014-04-10
JP5830519B2 JP5830519B2 (ja) 2015-12-09

Family

ID=44259848

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013500538A Active JP5830519B2 (ja) 2010-03-26 2011-03-28 Pbrリガンドとしての三環式インドール誘導体

Country Status (15)

Country Link
EP (1) EP2552891B1 (https=)
JP (1) JP5830519B2 (https=)
KR (1) KR101886879B1 (https=)
CN (1) CN102834379B (https=)
AU (1) AU2011231508B2 (https=)
BR (1) BR112012021579A2 (https=)
CA (1) CA2792394C (https=)
ES (1) ES2688574T3 (https=)
IL (1) IL221510A (https=)
MX (1) MX2012010954A (https=)
NZ (1) NZ602025A (https=)
RU (1) RU2551423C2 (https=)
SG (1) SG183837A1 (https=)
WO (1) WO2011117421A1 (https=)
ZA (1) ZA201208067B (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2946159B2 (ja) 1993-04-01 1999-09-06 高浜工業株式会社 瓦焼成用のスペ−サ装着装置
GB201016038D0 (en) * 2010-09-24 2010-11-10 Ge Healthcare Ltd In vivo imaging method
GB201016411D0 (en) * 2010-09-30 2010-11-10 Ge Healthcare Ltd In vivo imaging method for cancer
KR20150088802A (ko) 2012-11-30 2015-08-03 지이 헬쓰케어 리미티드 트리시클릭 인돌 유도체의 결정화 방법
GB201312768D0 (en) * 2013-07-17 2013-08-28 Ge Healthcare Ltd Work-up procedure
GB201316764D0 (en) * 2013-09-20 2013-11-06 Ge Healthcare Ltd Novel compounds
KR102668112B1 (ko) 2014-12-04 2024-05-23 지이 헬쓰케어 리미티드 방사성 약제로부터의 아세트알데히드의 제거 방법
CN106748802B (zh) * 2016-12-26 2018-11-13 南京理工大学 一种制备含氟仲胺的方法
CN114085221B (zh) * 2021-11-29 2022-12-09 暨南大学 含氮杂环化合物、标记的含氮杂环化合物及其制备方法和应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2599740B1 (fr) * 1986-06-05 1988-08-12 Rhone Poulenc Sante Derives de benzo(b)thiophene de benzo(b)furannecarboxamides, leurs procedes de preparation et les medicaments les contenant
FR2788776B1 (fr) * 1999-01-26 2001-02-23 Synthelabo Derives de 4-oxo-3, 5-dihydro-4h-pyridazino [4,5-b] indole-1 -carboxamide, leur preparation et leur application en therapeutique
US7160909B2 (en) 2001-08-09 2007-01-09 Eli Lilly And Company Cyclopenta[b]indole derivatives as sPLA2 inhibitors
GB0523506D0 (en) * 2005-11-18 2005-12-28 Hammersmith Imanet Ltd Novel in vivo imaging compounds
CN101528226B (zh) * 2006-08-24 2012-01-11 澳大利亚核科学技术组织 靶向外周苯二氮卓受体的氟化配体
GB0905328D0 (en) * 2009-03-27 2009-05-13 Ge Healthcare Ltd Indole derivatives

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