JP2013523621A5 - - Google Patents
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- Publication number
- JP2013523621A5 JP2013523621A5 JP2013500538A JP2013500538A JP2013523621A5 JP 2013523621 A5 JP2013523621 A5 JP 2013523621A5 JP 2013500538 A JP2013500538 A JP 2013500538A JP 2013500538 A JP2013500538 A JP 2013500538A JP 2013523621 A5 JP2013523621 A5 JP 2013523621A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- iii
- precursor compound
- precursor
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EPPCT/EP2010/053998 | 2010-03-26 | ||
| PCT/EP2010/053998 WO2010109007A2 (en) | 2009-03-27 | 2010-03-26 | Indole derivatives |
| IN1824/DEL/2010 | 2010-08-02 | ||
| IN1824DE2010 | 2010-08-02 | ||
| GBGB1015203.1A GB201015203D0 (en) | 2010-03-26 | 2010-09-13 | Active enantiomer |
| GB1015203.1 | 2010-09-13 | ||
| US12/880,218 | 2010-09-13 | ||
| US12/880,218 US8501153B2 (en) | 2009-03-27 | 2010-09-13 | Active enantiomer |
| PCT/EP2011/054744 WO2011117421A1 (en) | 2010-03-26 | 2011-03-28 | Tricyclic indole derivatives as pbr ligands |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013523621A JP2013523621A (ja) | 2013-06-17 |
| JP2013523621A5 true JP2013523621A5 (https=) | 2014-04-10 |
| JP5830519B2 JP5830519B2 (ja) | 2015-12-09 |
Family
ID=44259848
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013500538A Active JP5830519B2 (ja) | 2010-03-26 | 2011-03-28 | Pbrリガンドとしての三環式インドール誘導体 |
Country Status (15)
| Country | Link |
|---|---|
| EP (1) | EP2552891B1 (https=) |
| JP (1) | JP5830519B2 (https=) |
| KR (1) | KR101886879B1 (https=) |
| CN (1) | CN102834379B (https=) |
| AU (1) | AU2011231508B2 (https=) |
| BR (1) | BR112012021579A2 (https=) |
| CA (1) | CA2792394C (https=) |
| ES (1) | ES2688574T3 (https=) |
| IL (1) | IL221510A (https=) |
| MX (1) | MX2012010954A (https=) |
| NZ (1) | NZ602025A (https=) |
| RU (1) | RU2551423C2 (https=) |
| SG (1) | SG183837A1 (https=) |
| WO (1) | WO2011117421A1 (https=) |
| ZA (1) | ZA201208067B (https=) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2946159B2 (ja) | 1993-04-01 | 1999-09-06 | 高浜工業株式会社 | 瓦焼成用のスペ−サ装着装置 |
| GB201016038D0 (en) * | 2010-09-24 | 2010-11-10 | Ge Healthcare Ltd | In vivo imaging method |
| GB201016411D0 (en) * | 2010-09-30 | 2010-11-10 | Ge Healthcare Ltd | In vivo imaging method for cancer |
| KR20150088802A (ko) | 2012-11-30 | 2015-08-03 | 지이 헬쓰케어 리미티드 | 트리시클릭 인돌 유도체의 결정화 방법 |
| GB201312768D0 (en) * | 2013-07-17 | 2013-08-28 | Ge Healthcare Ltd | Work-up procedure |
| GB201316764D0 (en) * | 2013-09-20 | 2013-11-06 | Ge Healthcare Ltd | Novel compounds |
| KR102668112B1 (ko) | 2014-12-04 | 2024-05-23 | 지이 헬쓰케어 리미티드 | 방사성 약제로부터의 아세트알데히드의 제거 방법 |
| CN106748802B (zh) * | 2016-12-26 | 2018-11-13 | 南京理工大学 | 一种制备含氟仲胺的方法 |
| CN114085221B (zh) * | 2021-11-29 | 2022-12-09 | 暨南大学 | 含氮杂环化合物、标记的含氮杂环化合物及其制备方法和应用 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2599740B1 (fr) * | 1986-06-05 | 1988-08-12 | Rhone Poulenc Sante | Derives de benzo(b)thiophene de benzo(b)furannecarboxamides, leurs procedes de preparation et les medicaments les contenant |
| FR2788776B1 (fr) * | 1999-01-26 | 2001-02-23 | Synthelabo | Derives de 4-oxo-3, 5-dihydro-4h-pyridazino [4,5-b] indole-1 -carboxamide, leur preparation et leur application en therapeutique |
| US7160909B2 (en) | 2001-08-09 | 2007-01-09 | Eli Lilly And Company | Cyclopenta[b]indole derivatives as sPLA2 inhibitors |
| GB0523506D0 (en) * | 2005-11-18 | 2005-12-28 | Hammersmith Imanet Ltd | Novel in vivo imaging compounds |
| CN101528226B (zh) * | 2006-08-24 | 2012-01-11 | 澳大利亚核科学技术组织 | 靶向外周苯二氮卓受体的氟化配体 |
| GB0905328D0 (en) * | 2009-03-27 | 2009-05-13 | Ge Healthcare Ltd | Indole derivatives |
-
2011
- 2011-03-28 EP EP11710228.5A patent/EP2552891B1/en active Active
- 2011-03-28 MX MX2012010954A patent/MX2012010954A/es active IP Right Grant
- 2011-03-28 KR KR1020127025137A patent/KR101886879B1/ko active Active
- 2011-03-28 ES ES11710228.5T patent/ES2688574T3/es active Active
- 2011-03-28 BR BR112012021579-5A patent/BR112012021579A2/pt not_active IP Right Cessation
- 2011-03-28 JP JP2013500538A patent/JP5830519B2/ja active Active
- 2011-03-28 CN CN201180016200.0A patent/CN102834379B/zh active Active
- 2011-03-28 WO PCT/EP2011/054744 patent/WO2011117421A1/en not_active Ceased
- 2011-03-28 RU RU2012141697/04A patent/RU2551423C2/ru active
- 2011-03-28 AU AU2011231508A patent/AU2011231508B2/en active Active
- 2011-03-28 CA CA2792394A patent/CA2792394C/en active Active
- 2011-03-28 SG SG2012064382A patent/SG183837A1/en unknown
- 2011-03-28 NZ NZ602025A patent/NZ602025A/en unknown
-
2012
- 2012-08-16 IL IL221510A patent/IL221510A/en not_active IP Right Cessation
- 2012-10-25 ZA ZA2012/08067A patent/ZA201208067B/en unknown
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