JP2013510077A5 - - Google Patents
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- Publication number
- JP2013510077A5 JP2013510077A5 JP2012535688A JP2012535688A JP2013510077A5 JP 2013510077 A5 JP2013510077 A5 JP 2013510077A5 JP 2012535688 A JP2012535688 A JP 2012535688A JP 2012535688 A JP2012535688 A JP 2012535688A JP 2013510077 A5 JP2013510077 A5 JP 2013510077A5
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- JP
- Japan
- Prior art keywords
- alkyl
- alkoxy
- hydroxy
- halo
- amino
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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- 0 *c(cc1)cc(*)c1-c(cc1*)ccc1C1=CC=IN=C1 Chemical compound *c(cc1)cc(*)c1-c(cc1*)ccc1C1=CC=IN=C1 0.000 description 2
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25843209P | 2009-11-05 | 2009-11-05 | |
| US61/258,432 | 2009-11-05 | ||
| PCT/EP2010/006757 WO2011054530A1 (en) | 2009-11-05 | 2010-11-05 | Gpbp inhibition using q2 peptidomimetics |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013510077A JP2013510077A (ja) | 2013-03-21 |
| JP2013510077A5 true JP2013510077A5 (cg-RX-API-DMAC10.html) | 2013-12-26 |
| JP5883794B2 JP5883794B2 (ja) | 2016-03-15 |
Family
ID=43530495
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012535688A Expired - Fee Related JP5883794B2 (ja) | 2009-11-05 | 2010-11-05 | 擬似ｑ２ペプチドを用いるｇｐｂｐ抑制 |
Country Status (7)
| Country | Link |
|---|---|
| US (4) | US8586776B2 (cg-RX-API-DMAC10.html) |
| EP (1) | EP2496544B1 (cg-RX-API-DMAC10.html) |
| JP (1) | JP5883794B2 (cg-RX-API-DMAC10.html) |
| CN (1) | CN102781898B (cg-RX-API-DMAC10.html) |
| ES (1) | ES2523118T3 (cg-RX-API-DMAC10.html) |
| MX (1) | MX2012005281A (cg-RX-API-DMAC10.html) |
| WO (1) | WO2011054530A1 (cg-RX-API-DMAC10.html) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN105148269A (zh) * | 2011-02-21 | 2015-12-16 | 菲布他丁有限合伙公司 | 治疗和诊断疾病的方法 |
| JP2015524385A (ja) * | 2012-07-02 | 2015-08-24 | フィブロスタティン，エス．エル． | Ｇｐｂｐ−１阻害およびその治療的使用 |
| ES2489815B1 (es) * | 2013-02-21 | 2015-08-10 | Centro De Investigación Príncipe Felipe | Nuevos p-terfenilos hexakis-sustituidos con grupos bilaterales para el tratamiento de la infección por el virus de la inmunodeficiencia humana tipo 1 (VIH-1) y otras enfermedades |
| PT3013796T (pt) | 2013-06-27 | 2020-03-26 | Lg Chemical Ltd | Derivados biarílicos como agonistas de gpr120 |
| CN105723224A (zh) * | 2013-09-27 | 2016-06-29 | 菲布他丁有限合伙公司 | 古德帕斯丘抗原结合蛋白检测和抑制以及其在糖尿病中的应用 |
| MX385777B (es) * | 2014-12-24 | 2025-03-04 | Lg Chemical Ltd | Derivado de biarilo como agonista de gpr120. |
| WO2016107906A1 (en) | 2014-12-31 | 2016-07-07 | Fibrostatin, S.L. | Methods for inhibiting mesenchymal phenotype after epithelial-to-mesenchymal transition |
| WO2017134146A1 (en) * | 2016-02-02 | 2017-08-10 | Fibrostatin, S.L. | Gpbp inhibitors and uses and scaleable synthesis thereof |
| CN112479941B (zh) * | 2020-11-30 | 2023-01-13 | 沧州维智达美制药有限公司 | 一种2-取代-3-芳基卤苄衍生物的制备方法 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5723500A (en) * | 1995-09-22 | 1998-03-03 | Colgate-Palmolive Company | Antiplaque oral composition and method |
| RU2200730C2 (ru) * | 1996-07-31 | 2003-03-20 | Шионоги Энд Ко., Лтд. | Пара-терфенильные соединения, способ их получения (варианты) и фармацевтическая композиция (варианты) |
| EP0944582B1 (de) * | 1996-12-11 | 2003-07-02 | Abbott GmbH & Co. KG | Ketobenzamide als calpain-inhibitoren |
| US6579969B1 (en) | 1999-02-24 | 2003-06-17 | Juan Saus | Goodpasture antigen binding protein |
| US6881547B1 (en) | 2001-01-31 | 2005-04-19 | Juan Saus | Methods and reagents for treating autoimmune disorders |
| CA2446380A1 (en) * | 2001-05-08 | 2002-11-14 | Yale University | Proteomimetic compounds and methods |
| WO2004070025A2 (en) | 2003-02-05 | 2004-08-19 | Juan Saus | Novel goodpasture antigen-binding protein isoforms and protein misfolded-mediated disorders |
| US20040248850A1 (en) * | 2003-02-11 | 2004-12-09 | Kemia, Inc. | Compounds for the treatment of HIV infection |
| US7279600B2 (en) * | 2003-05-02 | 2007-10-09 | Wyeth | Hydroxy-biphenyl-carbaldehyde oxime derivatives and their use as estrogenic agents |
| GB0416508D0 (en) * | 2004-07-23 | 2004-08-25 | Merck Sharp & Dohme | Therapeutic agents |
| GB0500784D0 (en) * | 2005-01-14 | 2005-02-23 | Novartis Ag | Organic compounds |
| JP4776279B2 (ja) * | 2005-06-09 | 2011-09-21 | 株式会社Ａｄｅｋａ | 新規化合物及び液晶組成物 |
| KR101309502B1 (ko) * | 2005-10-07 | 2013-09-24 | 미쓰비시 가가꾸 가부시키가이샤 | 탄화수소 화합물, 전하 수송 재료, 전하 수송 재료 조성물및 유기 전계 발광 소자 |
| WO2007086439A1 (ja) * | 2006-01-25 | 2007-08-02 | Hodogaya Chemical Co., Ltd. | ｐ－ターフェニル化合物混合物及び該化合物混合物を用いた電子写真用感光体 |
| WO2009008311A1 (ja) * | 2007-07-07 | 2009-01-15 | Idemitsu Kosan Co., Ltd. | クリセン誘導体及びそれを用いた有機エレクトロルミネッセンス素子 |
| CN101970420B (zh) * | 2007-10-04 | 2014-09-24 | 默克雪兰诺有限公司 | 噁二唑衍生物 |
| ATE543799T1 (de) * | 2007-10-19 | 2012-02-15 | Janssen Pharmaceutica Nv | Piperidinyl- und piperazinylmodulatoren von g- sekretase |
| AR069802A1 (es) * | 2007-12-20 | 2010-02-17 | Astrazeneca Ab | Compuestos de carbamoilo como inhibidores de dgat1 190 |
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2010
- 2010-11-05 WO PCT/EP2010/006757 patent/WO2011054530A1/en not_active Ceased
- 2010-11-05 JP JP2012535688A patent/JP5883794B2/ja not_active Expired - Fee Related
- 2010-11-05 EP EP10779469.5A patent/EP2496544B1/en active Active
- 2010-11-05 MX MX2012005281A patent/MX2012005281A/es active IP Right Grant
- 2010-11-05 ES ES10779469.5T patent/ES2523118T3/es active Active
- 2010-11-05 CN CN201080050226.2A patent/CN102781898B/zh active Active
- 2010-11-05 US US12/940,598 patent/US8586776B2/en not_active Expired - Fee Related
-
2013
- 2013-10-25 US US14/063,709 patent/US9199936B2/en not_active Expired - Fee Related
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2015
- 2015-11-18 US US14/944,721 patent/US20160083327A1/en not_active Abandoned
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2018
- 2018-02-08 US US15/892,317 patent/US10544083B2/en not_active Expired - Fee Related