JP2013509435A - 長時間作用型注入可能パリペリドンエステルに関連した投与レジメン - Google Patents

長時間作用型注入可能パリペリドンエステルに関連した投与レジメン Download PDF

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JP2013509435A
JP2013509435A JP2012537131A JP2012537131A JP2013509435A JP 2013509435 A JP2013509435 A JP 2013509435A JP 2012537131 A JP2012537131 A JP 2012537131A JP 2012537131 A JP2012537131 A JP 2012537131A JP 2013509435 A JP2013509435 A JP 2013509435A
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Japan
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dose
patient
paliperidone
paliperidone palmitate
palmitate
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JP2012537131A
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English (en)
Japanese (ja)
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JP2013509435A5 (ru
Inventor
ルウィンブリスコー，ピーター，エィチ．
ガスマン−メイヤー，クリスティアーナ
ゴパル，シハリ
アフ，デイヴィッド，ダブリュ．
レムリー，バート，エム．エム．
サンタニ，マヘシュ，エヌ．
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ヤンセン ファーマシューティカ エヌ．ベー．
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Application filed by ヤンセン ファーマシューティカ エヌ．ベー． filed Critical ヤンセン ファーマシューティカ エヌ．ベー．
Publication of JP2013509435A publication Critical patent/JP2013509435A/ja
Publication of JP2013509435A5 publication Critical patent/JP2013509435A5/ja
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2012537131A 2009-10-30 2010-10-29 長時間作用型注入可能パリペリドンエステルに関連した投与レジメン Pending JP2013509435A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25669609P 2009-10-30 2009-10-30
US61/256,696 2009-10-30
PCT/US2010/054807 WO2011053829A1 (en) 2009-10-30 2010-10-29 Dosing regimen associated with long-acting injectable paliperidone esters

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2015237117A Division JP2016102123A (ja) 2009-10-30 2015-12-04 長時間作用型注入可能パリペリドンエステルに関連した投与レジメン

Publications (2)

Publication Number Publication Date
JP2013509435A true JP2013509435A (ja) 2013-03-14
JP2013509435A5 JP2013509435A5 (ru) 2013-12-19

Family

ID=43302985

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2012537131A Pending JP2013509435A (ja) 2009-10-30 2010-10-29 長時間作用型注入可能パリペリドンエステルに関連した投与レジメン
JP2015237117A Pending JP2016102123A (ja) 2009-10-30 2015-12-04 長時間作用型注入可能パリペリドンエステルに関連した投与レジメン

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2015237117A Pending JP2016102123A (ja) 2009-10-30 2015-12-04 長時間作用型注入可能パリペリドンエステルに関連した投与レジメン

Country Status (12)

Country Link
US (2) US20110105536A1 (ru)
EP (1) EP2493473A1 (ru)
JP (2) JP2013509435A (ru)
KR (1) KR20120116401A (ru)
CN (1) CN102802631A (ru)
AU (2) AU2010313290A1 (ru)
BR (1) BR112012010195A2 (ru)
CA (1) CA2742393A1 (ru)
CL (1) CL2012001110A1 (ru)
MX (1) MX2012005083A (ru)
NZ (1) NZ599558A (ru)
WO (1) WO2011053829A1 (ru)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018510894A (ja) * 2015-04-07 2018-04-19 ヤンセン ファーマシューティカルズ，インコーポレーテッド 長時間作用型注射可能パリペリドンエステルの抜かした投与量のための投与レジメン

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA72189C2 (ru) 1997-11-17 2005-02-15 Янссен Фармацевтика Н.В. Водные суспензии субмикронной формы эфиров 9-гидроксирисперидона жирных кислот
JP5825786B2 (ja) 2007-12-19 2015-12-02 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプＪａｎｓｓｅｎ Ｐｈａｒｍａｃｅｕｔｉｃａ Ｎａａｍｌｏｚｅ Ｖｅｎｎｏｏｔｓｃｈａｐ 長時間作用型注入可能パリペリドンエステルに関連する投薬計画
US9271939B2 (en) 2010-03-15 2016-03-01 Inventia Healthcare Private Limited Stabilized prolonged release pharmaceutical composition comprising atypical antipsychotic
RU2627469C2 (ru) 2011-03-18 2017-08-08 Алкермес Фарма Айэленд Лимитед Фармацевтические композиции, содержащие водонерастворимое антипсихотическое средство и сложные эфиры сорбита
CN102993200B (zh) * 2011-09-10 2016-02-03 鲁翠涛 帕潘立酮氨基酸酯及其制备方法
US10004807B2 (en) 2012-03-19 2018-06-26 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising fatty acid esters
NZ630428A (en) * 2012-03-19 2017-02-24 Alkermes Pharma Ireland Ltd Pharmaceutical compositions comprising benzyl alcohol
AU2013235523B9 (en) 2012-03-19 2018-01-04 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising glycerol esters
NZ748572A (en) 2012-09-19 2020-07-31 Alkermes Pharma Ireland Ltd Pharmaceutical compositions having improved storage stability
AU2015231278B2 (en) 2014-03-20 2020-01-23 Alkermes Pharma Ireland Limited Aripiprazole formulations having increased injection speeds
ITUB20155193A1 (it) * 2015-11-03 2017-05-03 Italfarmaco Spa Sospensioni orali di Givinostat fisicamente e chimicamente stabili
AU2019230014A1 (en) 2018-03-05 2020-09-17 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy
WO2022049006A1 (en) * 2020-09-02 2022-03-10 Janssen Pharmaceutica Nv Pre-filled syringe with optimized stopper placement
KR20230116837A (ko) 2020-11-30 2023-08-04 얀센 파마슈티카 엔.브이. 서방형 팔리페리돈 주사용 제형과 관련된 투약 요법
HUE065573T2 (hu) 2020-11-30 2024-06-28 Janssen Pharmaceutica Nv Elnyújtott felszabadulású paliperidon injektálható készítményeihez kapcsolódó adagolási rendek
JP2023551009A (ja) 2020-11-30 2023-12-06 ヤンセン ファーマシューティカ エヌ．ベー． 持続放出パリペリドン注射可能製剤に関連する投与レジメン

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008074852A (ja) * 2006-09-22 2008-04-03 Janssen Pharmaceut Nv 肝機能が低下した精神医学上の患者をパリペリドンで治療
JP2009524685A (ja) * 2006-08-14 2009-07-02 テバ ファーマシューティカル インダストリーズ リミティド ９−ヒドロキシ−リスペリドン（パリペリドン）の結晶型
WO2009080651A1 (en) * 2007-12-19 2009-07-02 Janssen Pharmaceutica Nv Dosing regimen associated with long acting injectable paliperidone esters

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5254556A (en) 1988-11-07 1993-10-19 Janssen Pharmaceutica N.V. 3-piperidinyl-1,2-benzisoxazoles
TW487572B (en) 1996-05-20 2002-05-21 Janssen Pharmaceutica Nv Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters
UA72189C2 (ru) 1997-11-17 2005-02-15 Янссен Фармацевтика Н.В. Водные суспензии субмикронной формы эфиров 9-гидроксирисперидона жирных кислот
KR100338776B1 (ko) 2000-07-11 2002-05-31 윤종용 멀티 로우 어드레스 테스트 가능한 반도체 메모리 장치 및그 테스트 방법
EP1879890A1 (en) 2005-04-25 2008-01-23 Janssen Pharmaceutica N.V. Preparation of aseptic 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4h-pyridio[1,2-a]pyrimidin-4-one palmitate ester

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2009524685A (ja) * 2006-08-14 2009-07-02 テバ ファーマシューティカル インダストリーズ リミティド ９−ヒドロキシ−リスペリドン（パリペリドン）の結晶型
JP2008074852A (ja) * 2006-09-22 2008-04-03 Janssen Pharmaceut Nv 肝機能が低下した精神医学上の患者をパリペリドンで治療
WO2009080651A1 (en) * 2007-12-19 2009-07-02 Janssen Pharmaceutica Nv Dosing regimen associated with long acting injectable paliperidone esters

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018510894A (ja) * 2015-04-07 2018-04-19 ヤンセン ファーマシューティカルズ，インコーポレーテッド 長時間作用型注射可能パリペリドンエステルの抜かした投与量のための投与レジメン
JP2020090498A (ja) * 2015-04-07 2020-06-11 ヤンセン ファーマシューティカルズ，インコーポレーテッド 長時間作用型注射可能パリペリドンエステルの抜かした投与量のための投与レジメン
JP2021130680A (ja) * 2015-04-07 2021-09-09 ヤンセン ファーマシューティカルズ，インコーポレーテッド 長時間作用型注射可能パリペリドンエステルの抜かした投与量のための投与レジメン
JP7228503B2 (ja) 2015-04-07 2023-02-24 ヤンセン ファーマシューティカルズ，インコーポレーテッド 長時間作用型注射可能パリペリドンエステルの抜かした投与量のための投与レジメン
JP7422277B2 (ja) 2015-04-07 2024-01-26 ヤンセン ファーマシューティカ エヌ．ベー． 長時間作用型注射可能パリペリドンエステルの抜かした投与量のための投与レジメン

Also Published As

Publication number Publication date
CN102802631A (zh) 2012-11-28
AU2015243103A1 (en) 2015-11-05
US20110105536A1 (en) 2011-05-05
AU2010313290A1 (en) 2012-05-17
US20130331402A1 (en) 2013-12-12
WO2011053829A1 (en) 2011-05-05
NZ599558A (en) 2014-09-26
CA2742393A1 (en) 2011-05-05
CL2012001110A1 (es) 2012-10-19
KR20120116401A (ko) 2012-10-22
BR112012010195A2 (pt) 2016-04-26
JP2016102123A (ja) 2016-06-02
MX2012005083A (es) 2012-09-28
EP2493473A1 (en) 2012-09-05

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