JP2012530141A5 - - Google Patents

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Publication number
JP2012530141A5
JP2012530141A5 JP2012516197A JP2012516197A JP2012530141A5 JP 2012530141 A5 JP2012530141 A5 JP 2012530141A5 JP 2012516197 A JP2012516197 A JP 2012516197A JP 2012516197 A JP2012516197 A JP 2012516197A JP 2012530141 A5 JP2012530141 A5 JP 2012530141A5
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JP
Japan
Prior art keywords
dosage form
apixaban
released
controlled release
weight
Prior art date
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JP2012516197A
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English (en)
Japanese (ja)
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JP2012530141A (ja
JP5775071B2 (ja
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Priority claimed from PCT/US2010/038660 external-priority patent/WO2010147978A1/en
Publication of JP2012530141A publication Critical patent/JP2012530141A/ja
Publication of JP2012530141A5 publication Critical patent/JP2012530141A5/ja
Application granted granted Critical
Publication of JP5775071B2 publication Critical patent/JP5775071B2/ja
Active legal-status Critical Current
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JP2012516197A 2009-06-16 2010-06-15 アピキサバンの製剤形 Active JP5775071B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18744209P 2009-06-16 2009-06-16
US61/187,442 2009-06-16
PCT/US2010/038660 WO2010147978A1 (en) 2009-06-16 2010-06-15 Dosage forms of apixaban

Publications (3)

Publication Number Publication Date
JP2012530141A JP2012530141A (ja) 2012-11-29
JP2012530141A5 true JP2012530141A5 (enExample) 2013-08-01
JP5775071B2 JP5775071B2 (ja) 2015-09-09

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ID=42677548

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012516197A Active JP5775071B2 (ja) 2009-06-16 2010-06-15 アピキサバンの製剤形

Country Status (24)

Country Link
US (4) US20120087978A1 (enExample)
EP (2) EP2442791B1 (enExample)
JP (1) JP5775071B2 (enExample)
KR (1) KR20120029428A (enExample)
CN (1) CN102802608A (enExample)
AU (1) AU2010260208B2 (enExample)
BR (1) BRPI1010739A2 (enExample)
CA (1) CA2765413A1 (enExample)
CY (1) CY1122685T1 (enExample)
DK (1) DK2442791T3 (enExample)
ES (1) ES2769357T3 (enExample)
HR (1) HRP20200297T1 (enExample)
HU (1) HUE048542T2 (enExample)
IL (1) IL216421A0 (enExample)
LT (1) LT2442791T (enExample)
MX (1) MX2011013080A (enExample)
PL (1) PL2442791T3 (enExample)
PT (1) PT2442791T (enExample)
RU (1) RU2012101214A (enExample)
SG (1) SG176785A1 (enExample)
SI (1) SI2442791T1 (enExample)
SM (1) SMT202000093T1 (enExample)
WO (1) WO2010147978A1 (enExample)
ZA (1) ZA201109334B (enExample)

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KR20190130411A (ko) 2018-05-14 2019-11-22 신일제약주식회사 아픽사반 약제학적 제제 및 그의 제조방법
CN112261935A (zh) * 2018-08-14 2021-01-22 江苏恒瑞医药股份有限公司 一种可注射的药物组合物及其制备方法
CN109010273B (zh) * 2018-10-08 2021-03-19 中国药科大学 一种阿哌沙班纳米混悬剂及其制备方法
KR102044676B1 (ko) * 2019-03-27 2019-11-14 주식회사 씨트리 생체적합성 고분자 기반 아픽사반 함유 미립구의 제조방법
KR102045721B1 (ko) * 2019-03-27 2019-11-18 주식회사 씨트리 아픽사반 함유 미립구 제조용 분산상의 조성물 및 이로부터 제조되는 생체적합성 고분자 기반 아픽사반 함유 미립구
CN110037990B (zh) * 2019-04-15 2023-03-28 海正药业(杭州)有限公司 一种阿哌沙班固体无定形分散体的制备工艺
WO2020219384A1 (en) * 2019-04-26 2020-10-29 Taho Pharmaceuticals Ltd. Apixaban transdermal delivery system and uses thereof
WO2020231791A1 (en) * 2019-05-10 2020-11-19 Fordoz Pharma Corp. Injectable polymer nanoparticle compositions of antithrombotic agents and methods thereof
JP7752487B2 (ja) * 2020-03-24 2025-10-10 日本ジェネリック株式会社 アピキサバン含有固体分散体
JP7520351B2 (ja) * 2020-08-14 2024-07-23 日医工株式会社 アピキサバン含有医薬組成物
BR112023004824A2 (pt) * 2020-09-18 2023-04-18 Bristol Myers Squibb Co Formas de dosagem para inibidores tyk2 compreendendo núcleos intumescíveis
CA3202161A1 (en) * 2020-12-13 2022-06-16 Matthaios VIDALIS Liquid apixaban formulation in small dose volume
PH12023553262A1 (en) * 2021-06-08 2024-03-25 Taho Pharmaceuticals Ltd Apixaban film product and uses thereof
CN115715770B (zh) * 2021-08-24 2024-01-26 新领医药技术(深圳)有限公司 阿哌沙班透皮贴剂及其制备方法
US12213972B2 (en) * 2022-07-27 2025-02-04 Slayback Pharma Llc Stable pharmaceutical compositions of apixaban
EP4642441A1 (en) * 2022-12-26 2025-11-05 Rexpharmatech Co., Ltd Sustained-release tablet comprising apixaban
WO2024220731A1 (en) * 2023-04-18 2024-10-24 Incyclix Bio, Llc. Advantageous human dosage regimens for administration of inx-315
WO2024261686A1 (en) * 2023-06-23 2024-12-26 Ronak Patel A gastroretentive composition comprising apixaban

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