JP2012502111A5 - - Google Patents

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Publication number
JP2012502111A5
JP2012502111A5 JP2011526999A JP2011526999A JP2012502111A5 JP 2012502111 A5 JP2012502111 A5 JP 2012502111A5 JP 2011526999 A JP2011526999 A JP 2011526999A JP 2011526999 A JP2011526999 A JP 2011526999A JP 2012502111 A5 JP2012502111 A5 JP 2012502111A5
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JP
Japan
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compound
alkyl
occurrence
haloalkyl
halogen
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JP2011526999A
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English (en)
Japanese (ja)
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JP2012502111A (ja
JP5567573B2 (ja
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Priority claimed from PCT/US2009/056675 external-priority patent/WO2010030891A2/en
Publication of JP2012502111A publication Critical patent/JP2012502111A/ja
Publication of JP2012502111A5 publication Critical patent/JP2012502111A5/ja
Application granted granted Critical
Publication of JP5567573B2 publication Critical patent/JP5567573B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2011526999A 2008-09-11 2009-09-11 アリールグアニジンｆ１ｆ０−ａｔｐアーゼ阻害剤およびそれと関連する方法 Expired - Fee Related JP5567573B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US9618408P 2008-09-11 2008-09-11
US61/096,184 2008-09-11
PCT/US2009/056675 WO2010030891A2 (en) 2008-09-11 2009-09-11 Aryl guanidine f1f0-atpase inhibitors and related methods

Publications (3)

Publication Number Publication Date
JP2012502111A JP2012502111A (ja) 2012-01-26
JP2012502111A5 true JP2012502111A5 (OSRAM) 2012-10-25
JP5567573B2 JP5567573B2 (ja) 2014-08-06

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ID=42005765

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011526999A Expired - Fee Related JP5567573B2 (ja) 2008-09-11 2009-09-11 アリールグアニジンｆ１ｆ０−ａｔｐアーゼ阻害剤およびそれと関連する方法

Country Status (5)

Country Link
US (1) US8497307B2 (OSRAM)
EP (1) EP2352724B1 (OSRAM)
JP (1) JP5567573B2 (OSRAM)
AU (1) AU2009291632B2 (OSRAM)
WO (1) WO2010030891A2 (OSRAM)

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ES2639439T3 (es) * 2010-12-08 2017-10-26 Lycera Corporation Inhibidores de F1F0-ATPasas de tipo pirazolilguanidina y sus usos terapéuticos de éstos
US9169199B2 (en) 2010-12-08 2015-10-27 Lycera Corporation Cycloalkyl guanidine F1F0-ATPase inhibitors and therapeutic uses thereof
WO2012078869A1 (en) 2010-12-08 2012-06-14 Lycera Corporation Pyridonyl guanidine f1f0-atpase inhibitors and therapeutic uses thereof
WO2013185045A1 (en) * 2012-06-08 2013-12-12 Lycera Corporation Indazole guanidine f1f0-atpase inhibitors and therapeutic uses thereof
US9580391B2 (en) 2012-06-08 2017-02-28 Lycera Corporation Saturated acyl guanidine for inhibition of F1F0-ATPase
EP2866893A4 (en) 2012-06-08 2015-12-23 Lycera Corp HETEROCYCLIC GUANIDINE F1FO ATPASE INHIBITORS
EP2874997A4 (en) 2012-07-19 2016-01-06 Univ Drexel NEW SIGMA RECEPTOR LIGANDS AND METHOD FOR REGULATING CELLULAR PROTEIN HOMEOSTASIS THEREWITH
CN103351360B (zh) * 2013-07-19 2015-03-25 浙江工业大学 一种含1,3,4-噻二唑基团的酰基硫脲类化合物、制备方法及其应用
CN103396349B (zh) * 2013-07-19 2014-12-17 浙江工业大学 一种含1-甲基环己基的酰基硫脲类化合物、制备方法及其应用
CA2931792A1 (en) 2013-12-10 2015-06-18 Lycera Corporation N-substituted pyrazolyl guanidine f1f0-atpase inhibitors and therapeutic uses thereof
EP3080089B1 (en) 2013-12-10 2019-05-08 Lycera Corporation Trifluoromethyl pyrazolyl guanidine f1fo-atpase inhibitors and therapeutic uses thereof
AU2014363958B2 (en) 2013-12-10 2018-11-08 Lycera Corporation Alkylpyrazolyl guanidine F1F0-ATPase inhibitors and therapeutic uses thereof
US11117870B2 (en) 2017-11-01 2021-09-14 Drexel University Compounds, compositions, and methods for treating diseases

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