JP2012012417A5 - - Google Patents

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Publication number
JP2012012417A5
JP2012012417A5 JP2011227135A JP2011227135A JP2012012417A5 JP 2012012417 A5 JP2012012417 A5 JP 2012012417A5 JP 2011227135 A JP2011227135 A JP 2011227135A JP 2011227135 A JP2011227135 A JP 2011227135A JP 2012012417 A5 JP2012012417 A5 JP 2012012417A5
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JP
Japan
Prior art keywords
compound
independently
occurrence
optionally substituted
nrco
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2011227135A
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English (en)
Japanese (ja)
Other versions
JP2012012417A (ja
Filing date
Publication date
Priority claimed from US11/098,751 external-priority patent/US7514448B2/en
Application filed filed Critical
Publication of JP2012012417A publication Critical patent/JP2012012417A/ja
Publication of JP2012012417A5 publication Critical patent/JP2012012417A5/ja
Pending legal-status Critical Current

Links

JP2011227135A 2004-06-30 2011-10-14 タンパク質キナーゼのインヒビターとして有用なアザインドール Pending JP2012012417A (ja)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US58438304P 2004-06-30 2004-06-30
US60/584,383 2004-06-30
US58472104P 2004-07-01 2004-07-01
US60/584,721 2004-07-01
US11/098,751 US7514448B2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases
US11/098,751 2005-04-04
PCT/US2005/011358 WO2005103050A2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases
USPCT/US05/11358 2005-04-04

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2007519460A Division JP5122280B2 (ja) 2004-06-30 2005-06-29 タンパク質キナーゼのインヒビターとして有用なアザインドール

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2013001760A Division JP2013064015A (ja) 2004-06-30 2013-01-09 タンパク質キナーゼのインヒビターとして有用なアザインドール

Publications (2)

Publication Number Publication Date
JP2012012417A JP2012012417A (ja) 2012-01-19
JP2012012417A5 true JP2012012417A5 (enExample) 2013-02-28

Family

ID=37801682

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2007519460A Expired - Fee Related JP5122280B2 (ja) 2004-06-30 2005-06-29 タンパク質キナーゼのインヒビターとして有用なアザインドール
JP2011227135A Pending JP2012012417A (ja) 2004-06-30 2011-10-14 タンパク質キナーゼのインヒビターとして有用なアザインドール

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2007519460A Expired - Fee Related JP5122280B2 (ja) 2004-06-30 2005-06-29 タンパク質キナーゼのインヒビターとして有用なアザインドール

Country Status (4)

Country Link
JP (2) JP5122280B2 (enExample)
IL (1) IL180303A0 (enExample)
MX (1) MX2007000092A (enExample)
NO (1) NO20070502L (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2007000092A (es) * 2004-06-30 2007-03-07 Vertex Pharma Azaindoles utiles como inhibidores de proteinas cinasas.
ES2401138T3 (es) * 2004-08-13 2013-04-17 Genentech, Inc. Inhibidores basados en tiazol de enzimas que usan ATP
DE102008038221A1 (de) * 2008-08-18 2010-02-25 Merck Patent Gmbh 7-Azaindolderivate
DE102009058280A1 (de) * 2009-12-14 2011-06-16 Merck Patent Gmbh Thiazolderivate
CA2794808C (en) * 2010-04-16 2019-08-20 Ac Immune S.A. Compounds for the treatment of diseases associated with amyloid or amyloid-like proteins
EP2585468A1 (en) * 2010-06-23 2013-05-01 Vertex Pharmaceuticals Incorporated Pyrrolo- pyrazine derivatives useful as inhibitors of atr kinase
DE102011105469A1 (de) * 2011-06-24 2012-12-27 Merck Patent Gmbh 7-Azaindolderivate
UY34832A (es) * 2012-05-31 2013-12-31 Phenex Pharmaceuticals Ag TIAZOLES SUSTITUIDOS POR CARBOXAMIDA O SULFONAMIDA Y DERIVADOS RELACIONADOS COMO MODULADORES PARA EL RECEPTOR NUCLEAR HUÉRFANO RORy (lambda)
BR112016017981B1 (pt) * 2014-02-04 2023-01-17 Taiho Pharmaceutical Co., Ltd. Compostos derivados de azaindola, inibidor de jak3, composição farmacêutica e agente compreendendo ditos compostos, e uso dos mesmos para tratar uma doença que envolve jak3
KR20230104782A (ko) * 2020-10-05 2023-07-10 인라이븐 테라퓨틱스, 인크. Bcr-abl 티로신 키나제 억제용 7-아자인돌 화합물
WO2023110843A1 (en) * 2021-12-15 2023-06-22 Almirall, S.A. Heterobicyclic derivatives as itk inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6265403B1 (en) * 1999-01-20 2001-07-24 Merck & Co., Inc. Angiogenesis inhibitors
JP2003525291A (ja) * 2000-03-01 2003-08-26 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ２，４−二置換チアゾリル誘導体
SE0202463D0 (sv) * 2002-08-14 2002-08-14 Astrazeneca Ab Novel compounds
TW200604168A (en) * 2004-04-02 2006-02-01 Vertex Pharma Azaindoles useful as inhibitors of rock and other protein kinases
MX2007000092A (es) * 2004-06-30 2007-03-07 Vertex Pharma Azaindoles utiles como inhibidores de proteinas cinasas.

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