MX2007000092A - Azaindoles utiles como inhibidores de proteinas cinasas. - Google Patents

Azaindoles utiles como inhibidores de proteinas cinasas.

Info

Publication number
MX2007000092A
MX2007000092A MX2007000092A MX2007000092A MX2007000092A MX 2007000092 A MX2007000092 A MX 2007000092A MX 2007000092 A MX2007000092 A MX 2007000092A MX 2007000092 A MX2007000092 A MX 2007000092A MX 2007000092 A MX2007000092 A MX 2007000092A
Authority
MX
Mexico
Prior art keywords
compound according
optionally substituted
nitrogen
sulfur
oxygen
Prior art date
Application number
MX2007000092A
Other languages
English (en)
Spanish (es)
Inventor
Guy Brenchley
Michael Mortimore
Francoise Pierad
Juan Miguel Jimenez
Ronald Kengtel
Francesca Mazzei
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US2005/011358 external-priority patent/WO2005103050A2/en
Application filed by Vertex Pharma filed Critical Vertex Pharma
Priority claimed from PCT/US2005/023429 external-priority patent/WO2006004984A1/en
Publication of MX2007000092A publication Critical patent/MX2007000092A/es

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Enzymes And Modification Thereof (AREA)
MX2007000092A 2004-06-30 2005-06-29 Azaindoles utiles como inhibidores de proteinas cinasas. MX2007000092A (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US58438304P 2004-06-30 2004-06-30
US58472104P 2004-07-01 2004-07-01
PCT/US2005/011358 WO2005103050A2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases
US11/098,751 US7514448B2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases
PCT/US2005/023429 WO2006004984A1 (en) 2004-06-30 2005-06-29 Azaindoles useful as inhibitors of protein kinases

Publications (1)

Publication Number Publication Date
MX2007000092A true MX2007000092A (es) 2007-03-07

Family

ID=37801682

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2007000092A MX2007000092A (es) 2004-06-30 2005-06-29 Azaindoles utiles como inhibidores de proteinas cinasas.

Country Status (4)

Country Link
JP (2) JP5122280B2 (enExample)
IL (1) IL180303A0 (enExample)
MX (1) MX2007000092A (enExample)
NO (1) NO20070502L (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2007000092A (es) * 2004-06-30 2007-03-07 Vertex Pharma Azaindoles utiles como inhibidores de proteinas cinasas.
AU2005272815A1 (en) * 2004-08-13 2006-02-23 Genentech, Inc. Thiazole based inhibitors of ATP-utilizing enzymes
DE102008038221A1 (de) * 2008-08-18 2010-02-25 Merck Patent Gmbh 7-Azaindolderivate
DE102009058280A1 (de) * 2009-12-14 2011-06-16 Merck Patent Gmbh Thiazolderivate
DK2558446T5 (da) 2010-04-16 2019-12-09 Ac Immune Sa Nye forbindelser til behandling af sygdomme associerede med amyloid- eller amyloidlignende proteiner
MX2013000103A (es) * 2010-06-23 2013-06-13 Vertex Pharma Derivados de pirrolo-pirazina utiles como inhibidores de cinasa art.
DE102011105469A1 (de) * 2011-06-24 2012-12-27 Merck Patent Gmbh 7-Azaindolderivate
JP6225178B2 (ja) * 2012-05-31 2017-11-01 フェネックス ファーマシューティカルス アーゲー オーファン核内受容体RORγの調整剤としてのカルボキサミドまたはスルホンアミド置換されたチアゾールおよび関連する誘導体
AU2015215582B2 (en) * 2014-02-04 2016-10-13 Taiho Pharmaceutical Co., Ltd. Azaindole derivative
IL301740A (en) * 2020-10-05 2023-05-01 Enliven Therapeutics Inc 7-azaindole compounds for inhibition of bcr-abl tyrosine kinases
WO2023110843A1 (en) * 2021-12-15 2023-06-22 Almirall, S.A. Heterobicyclic derivatives as itk inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6265403B1 (en) * 1999-01-20 2001-07-24 Merck & Co., Inc. Angiogenesis inhibitors
US7105550B2 (en) * 2000-03-01 2006-09-12 Christopher Love 2,4-disubstituted thiazolyl derivatives
SE0202463D0 (sv) * 2002-08-14 2002-08-14 Astrazeneca Ab Novel compounds
AU2005236002A1 (en) * 2004-04-02 2005-11-03 Vertex Pharmaceuticals Incorporated Azaindoles useful as inhibitors of rock and other protein kinases
MX2007000092A (es) * 2004-06-30 2007-03-07 Vertex Pharma Azaindoles utiles como inhibidores de proteinas cinasas.

Also Published As

Publication number Publication date
IL180303A0 (en) 2007-06-03
JP5122280B2 (ja) 2013-01-16
JP2008513352A (ja) 2008-05-01
JP2012012417A (ja) 2012-01-19
NO20070502L (no) 2007-01-26

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