JP2011529502A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2011529502A5 JP2011529502A5 JP2011521231A JP2011521231A JP2011529502A5 JP 2011529502 A5 JP2011529502 A5 JP 2011529502A5 JP 2011521231 A JP2011521231 A JP 2011521231A JP 2011521231 A JP2011521231 A JP 2011521231A JP 2011529502 A5 JP2011529502 A5 JP 2011529502A5
- Authority
- JP
- Japan
- Prior art keywords
- independently
- pharmaceutically acceptable
- acceptable salt
- compound
- halo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 150000003839 salts Chemical class 0.000 claims 28
- 239000011780 sodium chloride Substances 0.000 claims 25
- 150000001875 compounds Chemical class 0.000 claims 22
- 125000001475 halogen functional group Chemical group 0.000 claims 12
- 239000008194 pharmaceutical composition Substances 0.000 claims 11
- 229910052717 sulfur Inorganic materials 0.000 claims 11
- 229910052760 oxygen Inorganic materials 0.000 claims 10
- 125000000217 alkyl group Chemical group 0.000 claims 9
- 125000003545 alkoxy group Chemical group 0.000 claims 4
- 239000012458 free base Substances 0.000 claims 4
- 241000224016 Plasmodium Species 0.000 claims 2
- 125000003118 aryl group Chemical group 0.000 claims 2
- 125000000623 heterocyclic group Chemical group 0.000 claims 2
- 230000002401 inhibitory effect Effects 0.000 claims 2
- 241000894007 species Species 0.000 claims 2
- 125000002373 5 membered heterocyclic group Chemical group 0.000 claims 1
- 125000004070 6 membered heterocyclic group Chemical group 0.000 claims 1
- 125000002837 carbocyclic group Chemical group 0.000 claims 1
- 239000003937 drug carrier Substances 0.000 claims 1
- 201000004792 malaria Diseases 0.000 claims 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 1
- 0 *C(CC=NC(C(Nc(cc(C(F)(F)F)cc1NC(CCNC(N)=N)O)c1SCCN)=O)=C1)=C1C(Nc(cc(C(F)(F)F)cc1NC(CCNC(N)=N)=O)c1SCCN)=O Chemical compound *C(CC=NC(C(Nc(cc(C(F)(F)F)cc1NC(CCNC(N)=N)O)c1SCCN)=O)=C1)=C1C(Nc(cc(C(F)(F)F)cc1NC(CCNC(N)=N)=O)c1SCCN)=O 0.000 description 5
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8397208P | 2008-07-28 | 2008-07-28 | |
| US61/083,972 | 2008-07-28 | ||
| US16246709P | 2009-03-23 | 2009-03-23 | |
| US61/162,467 | 2009-03-23 | ||
| PCT/US2009/051909 WO2010014573A1 (en) | 2008-07-28 | 2009-07-28 | Anti-malarial compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2011529502A JP2011529502A (ja) | 2011-12-08 |
| JP2011529502A5 true JP2011529502A5 (US07846941-20101207-C00217.png) | 2012-08-30 |
Family
ID=41610687
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011521231A Pending JP2011529502A (ja) | 2008-07-28 | 2009-07-28 | 抗マラリア化合物 |
Country Status (12)
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20090092574A1 (en) | 2006-12-29 | 2009-04-09 | Scott Richard W | Ophthalmic And Otic Compositions Of Facially Amphiphilic Polymers And Oligomers And Uses Thereof |
| TWI478915B (zh) | 2008-10-27 | 2015-04-01 | Cellceutix Corp | 宿主防禦之合成模擬物及其用途 |
| MX2012007662A (es) * | 2010-01-07 | 2012-08-23 | Polymedix Inc | Compuestos anti-heparina. |
| KR20130048776A (ko) * | 2010-07-07 | 2013-05-10 | 유니버시티 오브 메디신 앤드 덴티스트리 오브 뉴 저지 | 면역조절방법 |
| TW201208677A (en) * | 2010-08-21 | 2012-03-01 | Polymedix Inc | Facially amphiphilic compounds, compositions, and uses thereof in treating cancer |
| RU2453533C1 (ru) * | 2011-02-08 | 2012-06-20 | Государственное образовательное учреждение высшего профессионального образования "Ярославский государственный университет им. П.Г. Демидова" | Способ получения 1,3- и 1,4-бис(2-амино-4-(трифторметил)фенокси)бензола |
| WO2012158672A2 (en) | 2011-05-16 | 2012-11-22 | Polymedix, Inc. | Compounds for use in treatment of mucositis |
| AU2012352621A1 (en) | 2011-12-13 | 2014-07-24 | Cellceutix Corporation | Cyclic compounds and methods of making and using the same |
| SG10201608528YA (en) * | 2011-12-21 | 2016-12-29 | Novira Therapeutics Inc | Hepatitis b antiviral agents |
| US20150094294A1 (en) * | 2012-02-29 | 2015-04-02 | Cellceutix Corporation | Compounds and methods for treating malaria |
| WO2015029807A1 (en) * | 2013-08-30 | 2015-03-05 | Semiconductor Energy Laboratory Co., Ltd. | Organic compound, light-emitting element, light-emitting device, electronic device, and lighting device |
| ES2894657T3 (es) * | 2017-07-04 | 2022-02-15 | Sanofi Sa | Compuestos de etinilo, su preparación y su uso terapéutico para el tratamiento de la malaria |
| WO2021248008A1 (en) | 2020-06-05 | 2021-12-09 | Innovation Pharmaceuticals Inc. | Arylamide compounds for treatment and prevention of viral infections |
Family Cites Families (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB951797A (en) | 1960-12-20 | 1964-03-11 | Monsanto Chemicals | Heterocyclic compounds |
| US3450772A (en) | 1964-12-04 | 1969-06-17 | Mobil Oil Corp | Polyphenyl ethers |
| SU425905A1 (ru) * | 1972-07-27 | 1974-04-30 | Ю. А. Москвичев, Г. С. Миронов, М. И. Фарберов, | СПОСОБ ПОЛУЧЕНИЯ п,п'-БИС- |
| SU1121264A1 (ru) * | 1983-04-29 | 1984-10-30 | Московский ордена Ленина и ордена Трудового Красного Знамени химико-технологический институт им.Д.И.Менделеева | Способ получени 3,6-бис(диметиламино)тиоксантен-10,10-диоксида |
| US5310726A (en) * | 1990-03-19 | 1994-05-10 | Merck & Co., Inc. | Lipopeptide compounds |
| US5066409A (en) | 1990-09-12 | 1991-11-19 | The Dow Chemical Company | Novel aryl ether sulfones |
| CA2126979A1 (en) * | 1991-12-31 | 1993-07-22 | Eliezer Rapaport | Antiparasitic oligonucleotides active against drug resistant malaria |
| US5798340A (en) * | 1993-09-17 | 1998-08-25 | Gilead Sciences, Inc. | Nucleotide analogs |
| RU2067572C1 (ru) * | 1994-02-04 | 1996-10-10 | Ярославский государственный технический университет | Многоядерные бисазиды |
| US5641737A (en) | 1995-12-18 | 1997-06-24 | The United States Of America As Represented By The Secretary Of The Air Force | Powdered sulfones as high temperature lubricants |
| ATE239003T1 (de) * | 1998-08-20 | 2003-05-15 | Univ North Carolina | Dibenzothiophene derivate und ihre verwendung |
| US6229012B1 (en) | 1998-10-01 | 2001-05-08 | Xerox Corporation | Triazine compositions |
| US6645531B1 (en) * | 2000-01-06 | 2003-11-11 | Marantech Holding Llc | Multivalent electron active compositions and methods of making and using same |
| JP2001261674A (ja) * | 2000-03-22 | 2001-09-26 | Mitsui Chemicals Inc | ベンゾチオフェン誘導体およびそれを有効成分として含有する核内レセプター作動薬 |
| US6660410B2 (en) | 2000-03-27 | 2003-12-09 | Idemitsu Kosan Co., Ltd. | Organic electroluminescence element |
| US6420342B1 (en) * | 2000-05-08 | 2002-07-16 | N.V. Nutricia | Nutritional preparation comprising ribose and medical use thereof |
| WO2002039987A2 (en) | 2000-11-14 | 2002-05-23 | Neurosearch A/S | Use of malaria parasite anion channel blockers for treating malaria |
| MXPA03004920A (es) * | 2001-02-14 | 2003-09-05 | Warner Lambert Co | Pirimidinas inhibidoras de metaloproteinasas de matriz. |
| DE10109204A1 (de) | 2001-02-26 | 2002-09-19 | 4Sc Ag | Verbindungen zur Behandlung von Protozoen-Erkrankungen |
| CN100366703C (zh) | 2002-03-22 | 2008-02-06 | 出光兴产株式会社 | 用于有机电致发光器件的材料以及使用该材料的有机电致发光器件 |
| US20040157804A1 (en) * | 2002-10-16 | 2004-08-12 | Gilead Sciences, Inc. | Pre-organized tricyclic integrase inhibitor compounds |
| JP2006521355A (ja) | 2003-03-17 | 2006-09-21 | ザ・トラステイーズ・オブ・ザ・ユニバーシテイ・オブ・ペンシルベニア・センター・フオー・テクノロジー・トランスフアー | 表面的に両親媒性のポリマー及びオリゴマーならびにそれらの使用 |
| US7169857B2 (en) | 2003-10-03 | 2007-01-30 | Virginia Commonwealth University | Homogenous compositions of fluoropolymers and crystalline solids or cross-linking agents and methods of making the same |
| JP5112601B2 (ja) * | 2003-10-07 | 2013-01-09 | 三井化学株式会社 | 複素環化合物および該化合物を含有する有機電界発光素子 |
| WO2006021833A2 (en) * | 2003-11-25 | 2006-03-02 | University Of Cincinnati | Bisbenzamidines for the treatment of pneumonia |
| CN1922133A (zh) | 2004-01-23 | 2007-02-28 | 宾夕法尼亚州大学理事会 | 表面两亲性聚芳基和聚芳基炔基聚合物和低聚物及其用途 |
| US7504769B2 (en) * | 2004-12-16 | 2009-03-17 | E. I. Du Pont De Nemours + Company | Aromatic chalcogen compounds and their use |
| EP2433627A1 (en) * | 2005-02-25 | 2012-03-28 | The Trustees Of The University Of Pennsylvania | Facially amphiphilic polymers and oligomers, compositions thereof, and use thereof in methods of treating cancer |
| RU2296756C2 (ru) * | 2005-05-17 | 2007-04-10 | Федеральное унитарное государственное предприятие "Государственный научно-исследовательский институт биологического приборостроения" (ГосНИИ БП) | Комплексообразующие дибензосодержащие пятичленные циклические соединения, содержащие два симметричных бета-дикарбонильных заместителя с фторированными радикалами |
| US20070224446A1 (en) * | 2006-03-24 | 2007-09-27 | Idemitsu Kosan Co., Ltd. | Material for organic electroluminescence device and organic electroluminescence device using the same |
| JP2008137978A (ja) | 2006-12-05 | 2008-06-19 | Canon Inc | カルバゾール誘導体及びこれを用いた有機発光素子 |
| US20090092574A1 (en) | 2006-12-29 | 2009-04-09 | Scott Richard W | Ophthalmic And Otic Compositions Of Facially Amphiphilic Polymers And Oligomers And Uses Thereof |
-
2009
- 2009-07-28 MX MX2011000971A patent/MX2011000971A/es not_active Application Discontinuation
- 2009-07-28 CA CA2732572A patent/CA2732572A1/en not_active Abandoned
- 2009-07-28 RU RU2011107295/04A patent/RU2530899C2/ru not_active IP Right Cessation
- 2009-07-28 BR BRPI0916649-1A patent/BRPI0916649A2/pt not_active IP Right Cessation
- 2009-07-28 CN CN2009801378005A patent/CN102164892A/zh active Pending
- 2009-07-28 KR KR1020117004117A patent/KR20110063435A/ko not_active Application Discontinuation
- 2009-07-28 EP EP09803456A patent/EP2321275A4/en not_active Withdrawn
- 2009-07-28 JP JP2011521231A patent/JP2011529502A/ja active Pending
- 2009-07-28 WO PCT/US2009/051909 patent/WO2010014573A1/en active Application Filing
- 2009-07-28 AU AU2009276744A patent/AU2009276744A1/en not_active Abandoned
- 2009-07-28 US US12/510,593 patent/US8796275B2/en active Active
-
2011
- 2011-01-27 IL IL210935A patent/IL210935A0/en unknown
-
2014
- 2014-08-05 US US14/452,116 patent/US20150072997A1/en not_active Abandoned
