JP2011521940A5 - - Google Patents

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Publication number
JP2011521940A5
JP2011521940A5 JP2011511102A JP2011511102A JP2011521940A5 JP 2011521940 A5 JP2011521940 A5 JP 2011521940A5 JP 2011511102 A JP2011511102 A JP 2011511102A JP 2011511102 A JP2011511102 A JP 2011511102A JP 2011521940 A5 JP2011521940 A5 JP 2011521940A5
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JP
Japan
Prior art keywords
composition
group
cas
exendin
obesity
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Withdrawn
Application number
JP2011511102A
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English (en)
Japanese (ja)
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JP2011521940A (ja
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Priority claimed from PCT/IB2009/005659 external-priority patent/WO2009144555A1/en
Publication of JP2011521940A publication Critical patent/JP2011521940A/ja
Publication of JP2011521940A5 publication Critical patent/JP2011521940A5/ja
Withdrawn legal-status Critical Current

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JP2011511102A 2008-05-28 2009-05-18 ピラゾロスピロケトンアセチルCoAカルボキシラーゼ阻害剤 Withdrawn JP2011521940A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US5665208P 2008-05-28 2008-05-28
US61/056,652 2008-05-28
US5868908P 2008-06-04 2008-06-04
US61/058,689 2008-06-04
US17111209P 2009-04-21 2009-04-21
US61/171,112 2009-04-21
PCT/IB2009/005659 WO2009144555A1 (en) 2008-05-28 2009-05-18 Pyrazolospiroketone acetyl-coa carboxylase inhibitors

Publications (2)

Publication Number Publication Date
JP2011521940A JP2011521940A (ja) 2011-07-28
JP2011521940A5 true JP2011521940A5 (enExample) 2012-07-05

Family

ID=40974463

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011511102A Withdrawn JP2011521940A (ja) 2008-05-28 2009-05-18 ピラゾロスピロケトンアセチルCoAカルボキシラーゼ阻害剤

Country Status (5)

Country Link
US (1) US20110009443A1 (enExample)
EP (1) EP2297164A1 (enExample)
JP (1) JP2011521940A (enExample)
CA (1) CA2724603A1 (enExample)
WO (1) WO2009144555A1 (enExample)

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EP3194367B1 (en) * 2014-09-17 2021-08-18 Boehringer Ingelheim International GmbH Tetrahydroisoquinoline derivatives and pharmaceutical compositions useful for the treatment of obesity and diabetes
WO2016092413A1 (en) 2014-12-10 2016-06-16 Pfizer Inc. Indole and indazole compounds that activate ampk
EP3237401B1 (en) 2014-12-22 2019-03-06 Pfizer Inc Antagonists of prostaglandin ep3 receptor
MA42035A (fr) 2015-05-05 2018-03-14 Pfizer 2-thiopyrimidinones
US10308615B2 (en) 2015-05-29 2019-06-04 Pfizer Inc. Heterocyclic compounds as inhibitors of Vanin-1 enzyme
ES2832893T3 (es) 2015-06-17 2021-06-11 Pfizer Compuestos tricíclicos y su uso como inhibidores de la fosfodiesterasa
WO2016203335A1 (en) 2015-06-18 2016-12-22 Pfizer Inc. Novel pyrido[2,3-b]pyrazinones as bet-family bromodomain inhibitors
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RS61719B1 (sr) 2015-08-27 2021-05-31 Pfizer Biciklična fuzionisana hetaroaril ili aril jedinjenja kao modulatori irak4
WO2017037567A1 (en) 2015-09-03 2017-03-09 Pfizer Inc. Regulators of frataxin
WO2017051276A1 (en) 2015-09-24 2017-03-30 Pfizer Inc. N-[2-(2-amino-6,6-disubstituted-4, 4a, 5, 6-tetrahydropyrano [3,4-d][1,3] thiazin-8a (8h)-yl) -1, 3-thiazol-4-yl] amides
EP3353174A1 (en) 2015-09-24 2018-08-01 Pfizer Inc N-[2-(3-amino-2,5-dimethyl-1,1-dioxido-5,6-dihydro-2h-1,2,4-thiadiazin-5-yl)-1,3-thiazol-4-yl]amides useful as bace inhibitors
JP2018531924A (ja) 2015-09-24 2018-11-01 ファイザー・インク テトラヒドロピラノ[3,4−d][1,3]オキサジン誘導体、およびbace阻害剤としてのその使用
JP6503515B2 (ja) 2015-12-29 2019-04-17 ファイザー・インク ケトヘキソキナーゼ阻害薬としての置換3−アザビシクロ[3.1.0]ヘキサン
JP2019519478A (ja) 2016-04-19 2019-07-11 ユレカ・ソシエテ・ア・レスポンサビリテ・リミテUreka Sarl ペプチド−オリゴ尿素フォルダマー化合物及びそれらの使用方法
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JP2025509281A (ja) 2022-03-09 2025-04-11 ガシャーブラム・バイオ・インコーポレイテッド ヘテロ環式glp-1アゴニスト
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EP2097420B1 (en) * 2006-11-29 2012-04-04 Pfizer Products Inc. Spiroketone inhibitors of acetyl-coa carboxylase

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