JP2011518819A5 - - Google Patents

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Publication number
JP2011518819A5
JP2011518819A5 JP2011505593A JP2011505593A JP2011518819A5 JP 2011518819 A5 JP2011518819 A5 JP 2011518819A5 JP 2011505593 A JP2011505593 A JP 2011505593A JP 2011505593 A JP2011505593 A JP 2011505593A JP 2011518819 A5 JP2011518819 A5 JP 2011518819A5
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JP
Japan
Prior art keywords
independently
nhr
alkyl
saturated aliphatic
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2011505593A
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English (en)
Japanese (ja)
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JP2011518819A (ja
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Publication date
Priority claimed from GBGB0807609.3A external-priority patent/GB0807609D0/en
Application filed filed Critical
Publication of JP2011518819A publication Critical patent/JP2011518819A/ja
Publication of JP2011518819A5 publication Critical patent/JP2011518819A5/ja
Withdrawn legal-status Critical Current

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JP2011505593A 2008-04-25 2009-04-27 アリール−キノリル化合物及びその使用 Withdrawn JP2011518819A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US4790208P 2008-04-25 2008-04-25
GBGB0807609.3A GB0807609D0 (en) 2008-04-25 2008-04-25 Therapeutic compounds and their use
US61/047,902 2008-04-25
GB0807609.3 2008-04-25
PCT/GB2009/001077 WO2009130487A1 (en) 2008-04-25 2009-04-27 Aryl-quinolyl compounds and their use

Publications (2)

Publication Number Publication Date
JP2011518819A JP2011518819A (ja) 2011-06-30
JP2011518819A5 true JP2011518819A5 (enExample) 2012-04-26

Family

ID=39522596

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011505593A Withdrawn JP2011518819A (ja) 2008-04-25 2009-04-27 アリール−キノリル化合物及びその使用

Country Status (10)

Country Link
US (1) US8383816B2 (enExample)
EP (1) EP2285805B1 (enExample)
JP (1) JP2011518819A (enExample)
CN (1) CN102066371A (enExample)
AU (1) AU2009239785A1 (enExample)
BR (1) BRPI0911525A2 (enExample)
CA (1) CA2721575A1 (enExample)
GB (1) GB0807609D0 (enExample)
WO (1) WO2009130487A1 (enExample)
ZA (1) ZA201007395B (enExample)

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AR070535A1 (es) * 2008-02-29 2010-04-14 Array Biopharma Inc Compuestos inhibidores de raf y metodos para usarlos
AU2009222144A1 (en) * 2008-02-29 2009-09-11 Array Biopharma Inc. Pyrazole [3, 4-b] pyridine Raf inhibitors
GB0807609D0 (en) 2008-04-25 2008-06-04 Cancer Rec Tech Ltd Therapeutic compounds and their use
CA2786834C (en) 2010-02-01 2018-10-16 Cancer Research Technology Limited 1-(5-tert-butyl-2-phenyl-2h-pyrazol-3-yl)-3-[2-fluoro-4-(1-methyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-7-yloxy)-phenyl]-urea and related compounds and their use in therapy
US8933228B2 (en) 2010-06-17 2015-01-13 Respivert, Ltd. Respiratory formulations and compounds for use therein
SG193301A1 (en) * 2011-03-09 2013-10-30 Merck Patent Gmbh Pyrido [2, 3 - b] pyrazine derivatives and their therapeutical uses
CA2916543C (en) * 2013-06-28 2023-03-14 Beigene, Ltd. Fused tricyclic urea compounds as raf kinase and/or raf kinase dimer inhibitors
GB201320732D0 (en) 2013-11-25 2014-01-08 Cancer Rec Tech Ltd Methods of chemical synthesis
GB201320729D0 (en) * 2013-11-25 2014-01-08 Cancer Rec Tech Ltd Therapeutic compounds and their use
EP3575305A1 (fr) 2018-05-31 2019-12-04 Biocidal Alternative Solutions Procédé de fabrication de composés comprenant un groupe fonctionnel oxazolopyridinones
JOP20180131B1 (ar) * 2018-12-24 2023-03-28 Univ Of Petra مركبات الكوينولون المستبدلة واستخدامها في علاج السرطان وطريقة تحضيرها
TWI812301B (zh) * 2021-06-24 2023-08-11 南韓商Lg化學股份有限公司 作為ron抑制劑之新穎尿素衍生物化合物

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GB0807609D0 (en) 2008-04-25 2008-06-04 Cancer Rec Tech Ltd Therapeutic compounds and their use
CA2786834C (en) 2010-02-01 2018-10-16 Cancer Research Technology Limited 1-(5-tert-butyl-2-phenyl-2h-pyrazol-3-yl)-3-[2-fluoro-4-(1-methyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-7-yloxy)-phenyl]-urea and related compounds and their use in therapy

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