JP2011518228A - 真菌感染症の治療法 - Google Patents

真菌感染症の治療法 Download PDF

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JP2011518228A
JP2011518228A JP2011506420A JP2011506420A JP2011518228A JP 2011518228 A JP2011518228 A JP 2011518228A JP 2011506420 A JP2011506420 A JP 2011506420A JP 2011506420 A JP2011506420 A JP 2011506420A JP 2011518228 A JP2011518228 A JP 2011518228A
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Japan
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alkyl
aryl
halogen
substituted
optionally
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JP2011506420A
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English (en)
Japanese (ja)
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JP2011518228A5 (enExample
Inventor
ルイス,キム
ラフラー,マイケル,デイビッド
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ノースイースタン・ユニバーシティ
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Publication of JP2011518228A publication Critical patent/JP2011518228A/ja
Publication of JP2011518228A5 publication Critical patent/JP2011518228A5/ja
Pending legal-status Critical Current

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4015Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2011506420A 2008-04-22 2009-04-22 真菌感染症の治療法 Pending JP2011518228A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4695308P 2008-04-22 2008-04-22
US61/046,953 2008-04-22
PCT/US2009/041403 WO2009132101A1 (en) 2008-04-22 2009-04-22 Methods of treating fungal infections

Publications (2)

Publication Number Publication Date
JP2011518228A true JP2011518228A (ja) 2011-06-23
JP2011518228A5 JP2011518228A5 (enExample) 2013-05-16

Family

ID=40790885

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011506420A Pending JP2011518228A (ja) 2008-04-22 2009-04-22 真菌感染症の治療法

Country Status (8)

Country Link
US (1) US20120252820A1 (enExample)
EP (1) EP2282730A1 (enExample)
JP (1) JP2011518228A (enExample)
CN (1) CN102083425A (enExample)
AU (1) AU2009239385A1 (enExample)
CA (1) CA2722404A1 (enExample)
MX (1) MX2010011678A (enExample)
WO (1) WO2009132101A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014130922A1 (en) * 2013-02-25 2014-08-28 Trustees Of Boston University Compositions and methods for treating fungal infections
CN103800437A (zh) * 2013-12-31 2014-05-21 芜湖乐锐思信息咨询有限公司 一种治疗虫霉病的中药
CN105641678A (zh) * 2014-12-03 2016-06-08 博瑞生物医药(苏州)股份有限公司 阿尼芬净胃肠外制剂及制备方法

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004024151A1 (en) * 2002-09-13 2004-03-25 New Pharma Research Sweden Ab Composition and potentiating method

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL6505398A (enExample) * 1965-04-28 1966-10-31
IL53440A0 (en) * 1977-11-22 1978-01-31 Teva Pharma 2-adamantyl hydrazines their preparation and pharmaceutical compositions containing them
US4923852A (en) * 1987-06-11 1990-05-08 Merck & Co., Inc. Aminoalkyl naphthalenediols as host resistance enhancers against viral infections
FR2631028B1 (fr) * 1988-05-09 1990-07-13 Cird Adamantyl-2 isothiazoline-4 ones-3, leur procede de preparation et leur utilisation comme agents bactericides et fongicides

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004024151A1 (en) * 2002-09-13 2004-03-25 New Pharma Research Sweden Ab Composition and potentiating method

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
JPN6013044755; Zentralblatt fuer Bakteriologie, Parasitenkunde, Infektionskrankheiten und Hygiene. 1. Abteilung, Me Vol.213,No.4,, 1970, p.462-469 *

Also Published As

Publication number Publication date
AU2009239385A1 (en) 2009-10-29
US20120252820A1 (en) 2012-10-04
WO2009132101A1 (en) 2009-10-29
MX2010011678A (es) 2011-01-21
CN102083425A (zh) 2011-06-01
CA2722404A1 (en) 2009-10-29
EP2282730A1 (en) 2011-02-16

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