JP2011507853A - 緊急避妊のための投与量レジメンならびに薬学的組成物およびパッケージ - Google Patents
緊急避妊のための投与量レジメンならびに薬学的組成物およびパッケージ Download PDFInfo
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- JP2011507853A JP2011507853A JP2010539503A JP2010539503A JP2011507853A JP 2011507853 A JP2011507853 A JP 2011507853A JP 2010539503 A JP2010539503 A JP 2010539503A JP 2010539503 A JP2010539503 A JP 2010539503A JP 2011507853 A JP2011507853 A JP 2011507853A
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- tanaproget
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- progestin
- estrogen
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/536—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
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|---|---|---|---|
| US828707P | 2007-12-20 | 2007-12-20 | |
| PCT/US2008/013933 WO2009082478A1 (en) | 2007-12-20 | 2008-12-19 | Dosage regimens and pharmaceutical compositions and packages for emergency contraception |
Related Child Applications (1)
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| JP2014118432A Division JP2014193918A (ja) | 2007-12-20 | 2014-06-09 | 緊急避妊のための投与量レジメンならびに薬学的組成物およびパッケージ |
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| JP2011507853A true JP2011507853A (ja) | 2011-03-10 |
| JP2011507853A5 JP2011507853A5 (enExample) | 2013-02-14 |
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| JP2014118432A Withdrawn JP2014193918A (ja) | 2007-12-20 | 2014-06-09 | 緊急避妊のための投与量レジメンならびに薬学的組成物およびパッケージ |
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Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20090170823A1 (enExample) |
| EP (1) | EP2234491A4 (enExample) |
| JP (2) | JP2011507853A (enExample) |
| AU (1) | AU2008341138A1 (enExample) |
| BR (1) | BRPI0819571A2 (enExample) |
| CA (1) | CA2710293A1 (enExample) |
| EA (1) | EA201070715A1 (enExample) |
| IL (1) | IL206465A0 (enExample) |
| WO (1) | WO2009082478A1 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012523446A (ja) * | 2009-04-14 | 2012-10-04 | ラボラトワール・アシュエールア−ファルマ | オンデマンド避妊方法 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| RU2465907C2 (ru) * | 2006-12-20 | 2012-11-10 | Тева Вимен'С Хелс, Инк. | Распадающиеся в полости рта твердые дозированные формы, содержащие прогестин, и способы получения и применение указанных дозированных форм |
| FR2937862B1 (fr) * | 2008-11-03 | 2010-11-19 | Mohammed Ridha Chakroun | Kit contraceptif |
| EP4733407A3 (en) * | 2008-12-23 | 2026-08-19 | Quest Diagnostics Investments LLC | Mass spectrometry assay for estrogenic compounds |
| AU2014268779A1 (en) | 2013-05-21 | 2016-01-21 | Predictive Therapeutics, LLC | Therapeutic and method of use |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2000511890A (ja) * | 1996-05-16 | 2000-09-12 | ガイネティックス・インコーポレイテッド | 緊急避妊キット |
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| US4684534A (en) | 1985-02-19 | 1987-08-04 | Dynagram Corporation Of America | Quick-liquifying, chewable tablet |
| DK174724B1 (da) | 1986-07-15 | 2003-10-06 | Wyeth Corp | Anvendelse af et præparat omfattende et østrogen og et progestogen til fremstilling af en dosisform til tilvejebringelse af hormonerstatningsterapi og kontraception til kvinder i præmenopausen samt pakning til tilvejebringelse af præparatet |
| JPH07508987A (ja) * | 1992-07-01 | 1995-10-05 | オーソ・フアーマシユーチカル・コーポレーシヨン | １−アリールスルホニル，アリールカルボニルおよび１−アリールホスホニル−３−フェニル−１，４，５，６−テトラヒドロピリダジン |
| DE4344463A1 (de) * | 1993-12-22 | 1995-06-29 | Schering Ag | Kombinationsprodukt zur Kontrazeption |
| US5633011A (en) * | 1994-08-04 | 1997-05-27 | Alza Corporation | Progesterone replacement therapy |
| NZ295365A (en) * | 1994-10-24 | 1999-07-29 | Schering Ag | Competitive progesterone antagonists for regulating female fertility as required |
| ZA9510926B (en) * | 1994-12-23 | 1996-07-03 | Schering Ag | Compounds with progesterone-antagonistic and antiestrogenic action to be used together for female contraception |
| FR2772617B1 (fr) * | 1997-12-19 | 2001-03-09 | Besins Iscovesco Lab | Comprime de progesterone et son procede de preparation |
| US6368625B1 (en) | 1998-08-12 | 2002-04-09 | Cima Labs Inc. | Orally disintegrable tablet forming a viscous slurry |
| US6060078A (en) * | 1998-09-28 | 2000-05-09 | Sae Han Pharm Co., Ltd. | Chewable tablet and process for preparation thereof |
| US6667050B1 (en) * | 1999-04-06 | 2003-12-23 | Galen (Chemicals) Limited | Chewable oral contraceptive |
| US6399593B1 (en) * | 1999-05-04 | 2002-06-04 | Wyeth | Cyclic regimens using cyclic urea and cyclic amide derivatives |
| US6355648B1 (en) * | 1999-05-04 | 2002-03-12 | American Home Products Corporation | Thio-oxindole derivatives |
| US6407101B1 (en) * | 1999-05-04 | 2002-06-18 | American Home Products Corporation | Cyanopyrroles |
| US6660726B2 (en) * | 2000-03-10 | 2003-12-09 | Endeavor Pharmaceuticals | Estrogenic compounds, pharmaceutical compositions thereof, and methods of using same |
| UA73119C2 (en) * | 2000-04-19 | 2005-06-15 | American Home Products Corpoir | Derivatives of cyclic thiocarbamates, pharmaceutical composition including noted derivatives of cyclic thiocarbamates and active ingredients of medicines as modulators of progesterone receptors |
| US6316029B1 (en) * | 2000-05-18 | 2001-11-13 | Flak Pharma International, Ltd. | Rapidly disintegrating solid oral dosage form |
| HU227198B1 (en) * | 2001-11-27 | 2010-10-28 | Richter Gedeon Nyrt | Pharmaceutical composition for emergency contraception containing levonorgestrel |
| US20030158432A1 (en) | 2002-01-08 | 2003-08-21 | Leonard Thomas W. | Synthesis of a mixture of sulfated estrogens using a sulfur trioxide complex |
| DK1482925T3 (da) * | 2002-03-11 | 2007-05-14 | Bayer Schering Pharma Ag | 5- (2-hydroxy-3 -'1 - (3-trifluormethylphenyl) cyclopropylpropionylamino) phtalid og relaterede forbindelser med progesteronreceptormoducerende aktivitet til anvendelse i fertilitetskontrol og hormonerstatningsterapi |
| EP1531824A4 (en) * | 2002-06-25 | 2005-09-21 | Wyeth Corp | CYCLOTHIOCARBAMATE DERIVATIVES AS PR-MODULATORS AND THEIR USE IN THE TREATMENT OF SKIN DISEASES |
| JP2005535623A (ja) * | 2002-06-25 | 2005-11-24 | ワイス | ホルモン関連症状の治療における、チオ−オキシインドール誘導体の使用 |
| AU2003247608A1 (en) | 2002-06-25 | 2004-01-06 | Wyeth | Use of cyclothiocarbamate derivatives in treatment of hormone-related conditions |
| AR040783A1 (es) * | 2002-10-11 | 2005-04-20 | Ligand Pharm Inc | 5-(1',1'-cicloaquil/alquenil) metiliden-1,2 -dihidro-5-h-cromeno [3,4- f] quiinolinas como compuestos moduladores selectivos de receptores de progesterona |
| WO2004035883A2 (en) * | 2002-10-17 | 2004-04-29 | Nexen Nano Tech Co., Ltd | Fibrous nano-carbon and preparation method thereof |
| JP4739217B2 (ja) * | 2003-05-07 | 2011-08-03 | サムヤン コーポレイション | 速く溶ける錠剤を製造するための高可塑性顆粒 |
| AR047398A1 (es) * | 2003-11-24 | 2006-01-18 | Wyeth Corp | Acoplamiento cruzado carbono- carbono catalizado por metales de transicion sobre soportes solidos |
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| CN1672685A (zh) * | 2004-03-26 | 2005-09-28 | 董可娟 | 一种新的避孕药物 |
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| JP4950027B2 (ja) * | 2004-04-08 | 2012-06-13 | ワイス・エルエルシー | チオアミド不純物を最小限に抑えるための方法 |
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| JP5108506B2 (ja) | 2004-04-27 | 2012-12-26 | ワイス・エルエルシー | シアノピロール含有環式カルバメートおよびチオカルバメートビアリール、およびこれらの製造方法 |
| BRPI0510260A (pt) * | 2004-04-27 | 2007-10-23 | Wyeth Corp | método para purificar um composto, e, kit farmacêutico |
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2008
- 2008-12-19 US US12/339,329 patent/US20090170823A1/en not_active Abandoned
- 2008-12-19 BR BRPI0819571A patent/BRPI0819571A2/pt not_active IP Right Cessation
- 2008-12-19 EP EP08865187A patent/EP2234491A4/en not_active Withdrawn
- 2008-12-19 EA EA201070715A patent/EA201070715A1/ru unknown
- 2008-12-19 JP JP2010539503A patent/JP2011507853A/ja active Pending
- 2008-12-19 CA CA2710293A patent/CA2710293A1/en not_active Abandoned
- 2008-12-19 WO PCT/US2008/013933 patent/WO2009082478A1/en not_active Ceased
- 2008-12-19 AU AU2008341138A patent/AU2008341138A1/en not_active Abandoned
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2010
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2014
- 2014-06-09 JP JP2014118432A patent/JP2014193918A/ja not_active Withdrawn
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| JP2000511890A (ja) * | 1996-05-16 | 2000-09-12 | ガイネティックス・インコーポレイテッド | 緊急避妊キット |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012523446A (ja) * | 2009-04-14 | 2012-10-04 | ラボラトワール・アシュエールア−ファルマ | オンデマンド避妊方法 |
| JP2016188232A (ja) * | 2009-04-14 | 2016-11-04 | ラボラトワール・アシュエールア−ファルマＬａｂｏｒａｔｏｉｒｅ Ｈｒａ−Ｐｈａｒｍａ | オンデマンド避妊方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2009082478A1 (en) | 2009-07-02 |
| IL206465A0 (en) | 2010-12-30 |
| EA201070715A1 (ru) | 2011-02-28 |
| CA2710293A1 (en) | 2009-07-02 |
| US20090170823A1 (en) | 2009-07-02 |
| JP2014193918A (ja) | 2014-10-09 |
| BRPI0819571A2 (pt) | 2019-09-24 |
| EP2234491A1 (en) | 2010-10-06 |
| EP2234491A4 (en) | 2010-12-22 |
| AU2008341138A1 (en) | 2009-07-02 |
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