CA2710293A1 - Dosage regimens and pharmaceutical compositions and packages for emergency contraception - Google Patents
Dosage regimens and pharmaceutical compositions and packages for emergency contraception Download PDFInfo
- Publication number
- CA2710293A1 CA2710293A1 CA2710293A CA2710293A CA2710293A1 CA 2710293 A1 CA2710293 A1 CA 2710293A1 CA 2710293 A CA2710293 A CA 2710293A CA 2710293 A CA2710293 A CA 2710293A CA 2710293 A1 CA2710293 A1 CA 2710293A1
- Authority
- CA
- Canada
- Prior art keywords
- dosage
- tanaproget
- hours
- nonsteroidal progestin
- nonsteroidal
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- 239000008194 pharmaceutical composition Substances 0.000 title claims abstract description 8
- 239000000583 progesterone congener Substances 0.000 claims abstract description 123
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- PYVFWTPEBMRKSR-UHFFFAOYSA-N tanaproget Chemical compound CN1C(C#N)=CC=C1C1=CC=C(NC(=S)OC2(C)C)C2=C1 PYVFWTPEBMRKSR-UHFFFAOYSA-N 0.000 claims description 94
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- 238000000227 grinding Methods 0.000 description 1
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- 239000002674 ointment Substances 0.000 description 1
- 239000003960 organic solvent Substances 0.000 description 1
- 239000003791 organic solvent mixture Substances 0.000 description 1
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- 230000000144 pharmacologic effect Effects 0.000 description 1
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- 239000010452 phosphate Substances 0.000 description 1
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- 150000004885 piperazines Chemical class 0.000 description 1
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- 229960001424 quinestrol Drugs 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/536—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US828707P | 2007-12-20 | 2007-12-20 | |
| US61/008,287 | 2007-12-20 | ||
| PCT/US2008/013933 WO2009082478A1 (en) | 2007-12-20 | 2008-12-19 | Dosage regimens and pharmaceutical compositions and packages for emergency contraception |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2710293A1 true CA2710293A1 (en) | 2009-07-02 |
Family
ID=40799234
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2710293A Abandoned CA2710293A1 (en) | 2007-12-20 | 2008-12-19 | Dosage regimens and pharmaceutical compositions and packages for emergency contraception |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20090170823A1 (enExample) |
| EP (1) | EP2234491A4 (enExample) |
| JP (2) | JP2011507853A (enExample) |
| AU (1) | AU2008341138A1 (enExample) |
| BR (1) | BRPI0819571A2 (enExample) |
| CA (1) | CA2710293A1 (enExample) |
| EA (1) | EA201070715A1 (enExample) |
| IL (1) | IL206465A0 (enExample) |
| WO (1) | WO2009082478A1 (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2007338843B2 (en) * | 2006-12-20 | 2013-05-09 | Teva Women's Health, Inc. | Orally disintegrating solid dosage forms comprising progestin and methods of making and use thereof |
| FR2937862B1 (fr) * | 2008-11-03 | 2010-11-19 | Mohammed Ridha Chakroun | Kit contraceptif |
| EP4079308A1 (en) * | 2008-12-23 | 2022-10-26 | Quest Diagnostics Investments Incorporated | Mass spectrometry assay for estrogenic compounds |
| AU2010237120B8 (en) * | 2009-04-14 | 2015-11-26 | Laboratoire Hra-Pharma | Method for on-demand contraception |
| KR20160013098A (ko) | 2013-05-21 | 2016-02-03 | 프리딕티브 테라퓨틱스, 엘엘씨 | 치료제 및 그 사용 방법 |
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| US4684534A (en) | 1985-02-19 | 1987-08-04 | Dynagram Corporation Of America | Quick-liquifying, chewable tablet |
| DK174724B1 (da) | 1986-07-15 | 2003-10-06 | Wyeth Corp | Anvendelse af et præparat omfattende et østrogen og et progestogen til fremstilling af en dosisform til tilvejebringelse af hormonerstatningsterapi og kontraception til kvinder i præmenopausen samt pakning til tilvejebringelse af præparatet |
| DK0650480T3 (da) * | 1992-07-01 | 2002-05-13 | Ortho Pharma Corp | 1-Arylsulfonyl-3-phenyl-1,4,5,6-tetrahydropyridaziner |
| DE4344463A1 (de) * | 1993-12-22 | 1995-06-29 | Schering Ag | Kombinationsprodukt zur Kontrazeption |
| US5633011A (en) * | 1994-08-04 | 1997-05-27 | Alza Corporation | Progesterone replacement therapy |
| ATE347894T1 (de) * | 1994-10-24 | 2007-01-15 | Schering Ag | Kompetitive progesteronantagonisten zur bedarfsorientierten weiblichen fertilitätskontrolle |
| ZA9510926B (en) * | 1994-12-23 | 1996-07-03 | Schering Ag | Compounds with progesterone-antagonistic and antiestrogenic action to be used together for female contraception |
| CA2253289A1 (en) * | 1996-05-16 | 1997-11-20 | Roderick L. Mackenzie | Emergency contraceptive kit |
| FR2772617B1 (fr) * | 1997-12-19 | 2001-03-09 | Besins Iscovesco Lab | Comprime de progesterone et son procede de preparation |
| US6368625B1 (en) | 1998-08-12 | 2002-04-09 | Cima Labs Inc. | Orally disintegrable tablet forming a viscous slurry |
| US6060078A (en) | 1998-09-28 | 2000-05-09 | Sae Han Pharm Co., Ltd. | Chewable tablet and process for preparation thereof |
| US6667050B1 (en) * | 1999-04-06 | 2003-12-23 | Galen (Chemicals) Limited | Chewable oral contraceptive |
| US6399593B1 (en) * | 1999-05-04 | 2002-06-04 | Wyeth | Cyclic regimens using cyclic urea and cyclic amide derivatives |
| US6355648B1 (en) * | 1999-05-04 | 2002-03-12 | American Home Products Corporation | Thio-oxindole derivatives |
| US6407101B1 (en) * | 1999-05-04 | 2002-06-18 | American Home Products Corporation | Cyanopyrroles |
| US6660726B2 (en) * | 2000-03-10 | 2003-12-09 | Endeavor Pharmaceuticals | Estrogenic compounds, pharmaceutical compositions thereof, and methods of using same |
| UA73119C2 (en) * | 2000-04-19 | 2005-06-15 | American Home Products Corpoir | Derivatives of cyclic thiocarbamates, pharmaceutical composition including noted derivatives of cyclic thiocarbamates and active ingredients of medicines as modulators of progesterone receptors |
| US6316029B1 (en) | 2000-05-18 | 2001-11-13 | Flak Pharma International, Ltd. | Rapidly disintegrating solid oral dosage form |
| HU227198B1 (en) * | 2001-11-27 | 2010-10-28 | Richter Gedeon Nyrt | Pharmaceutical composition for emergency contraception containing levonorgestrel |
| US20030158432A1 (en) | 2002-01-08 | 2003-08-21 | Leonard Thomas W. | Synthesis of a mixture of sulfated estrogens using a sulfur trioxide complex |
| PL372490A1 (en) * | 2002-03-11 | 2005-07-25 | Schering Aktiengesellschaft | 5-{2-hydroxy-3-[1-(3-trifluoromethylphenyl)-cyclopropyl]-propionylamino}-phtalide and related compounds with progesterone receptor modulating activity for use in fertility control and hormone replacement therapy |
| CN1662241A (zh) * | 2002-06-25 | 2005-08-31 | 惠氏公司 | 环硫代氨基甲酸酯衍生物在治疗与激素有关的病症中的用途 |
| BR0312054A (pt) * | 2002-06-25 | 2005-10-18 | Wyeth Corp | Uso de derivados de tio-oxindol na preparação de medicamentos úteis no tratamento de condições relacionadas com hormÈnio, e kit farmacêutico |
| AR040644A1 (es) * | 2002-06-25 | 2005-04-13 | Wyeth Corp | Un moduladores del receptor de progesterona benzoxazina-2-tiona, una composicion farmaceutica, uso del compuesto para preparar un dedicamento para tratar una enfermedad neoplasica-hormona-dependiente y el uso de un compuesto benzoxazina-2-tiona, benzoxazina-2-ilideno cianamida o benzoxazina-2-iliden |
| AR040783A1 (es) * | 2002-10-11 | 2005-04-20 | Ligand Pharm Inc | 5-(1',1'-cicloaquil/alquenil) metiliden-1,2 -dihidro-5-h-cromeno [3,4- f] quiinolinas como compuestos moduladores selectivos de receptores de progesterona |
| WO2004035883A2 (en) * | 2002-10-17 | 2004-04-29 | Nexen Nano Tech Co., Ltd | Fibrous nano-carbon and preparation method thereof |
| EP1620075B1 (en) * | 2003-05-07 | 2020-06-24 | Samyang Biopharmaceuticals Corporation | Highly plastic granules for making fast melting tablets |
| AR047398A1 (es) * | 2003-11-24 | 2006-01-18 | Wyeth Corp | Acoplamiento cruzado carbono- carbono catalizado por metales de transicion sobre soportes solidos |
| EP1691746B1 (en) * | 2003-12-08 | 2015-05-27 | Gel-Del Technologies, Inc. | Mucoadhesive drug delivery devices and methods of making and using thereof |
| CN1672685A (zh) * | 2004-03-26 | 2005-09-28 | 董可娟 | 一种新的避孕药物 |
| US7399870B2 (en) * | 2004-03-30 | 2008-07-15 | Wyeth | Synthesis of pyrrole-2-carbonitriles |
| CA2561313C (en) * | 2004-04-08 | 2012-12-04 | Wyeth | Methods for minimizing thioamide impurities |
| WO2005100291A2 (en) * | 2004-04-08 | 2005-10-27 | Wyeth | Method for preparing 3-cyclopentyloxy-4-methoxybenzaldehyde |
| DE602005010840D1 (de) * | 2004-04-08 | 2008-12-18 | Wyeth Corp | Thioamidderivate als progesteronrezeptormodulatoren |
| CN1953967B (zh) | 2004-04-27 | 2013-03-13 | 惠氏公司 | 孕酮受体调节剂的纯化 |
| AU2005238520B2 (en) * | 2004-04-27 | 2011-09-08 | Wyeth | Cyanopyrrole containing cyclic carbamate and thiocarbamate biaryls and methods for preparing the same |
| WO2005105817A2 (en) | 2004-04-27 | 2005-11-10 | Wyeth | Coupling process for generating reactive boron containing derivatives of n-substituted pyrrole-2 carbonitriles to produce biaryls |
| PE20060378A1 (es) * | 2004-07-07 | 2006-06-02 | Wyeth Corp | Regimenes y kits de progestina ciclica |
| GT200500183A (es) * | 2004-08-09 | 2006-04-10 | Moduladores del receptor de progesterona que comprenden derivados de pirrol-oxindol y sus usos | |
| MX2007001812A (es) * | 2004-08-13 | 2007-03-26 | Wyeth Corp | Derivados de tanaproget, metabolitos, y usos de los mismos. |
| CN101027321A (zh) | 2004-08-20 | 2007-08-29 | 惠氏公司 | 孕酮受体结构 |
| JP4197684B2 (ja) * | 2005-03-23 | 2008-12-17 | 株式会社東芝 | 携帯無線機 |
| PL1877059T3 (pl) * | 2005-04-28 | 2010-07-30 | Wyeth Llc | Mikroniozowany tanaproget i zawierające go kompozycje |
| ES2327783T3 (es) * | 2005-04-28 | 2009-11-03 | Wyeth | Composiciones que contienen tanaproget micronizado. |
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| MX2007013469A (es) | 2005-04-28 | 2008-01-22 | Wyeth Corp | Forma ii polimorfa de tanaproget. |
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| DE102005050729A1 (de) * | 2005-10-19 | 2007-04-26 | Schering Ag | Verfahren zur präventiven bedarfsweisen hormonalen Kontrazeption |
| US20070093548A1 (en) * | 2005-10-25 | 2007-04-26 | Wyeth | Use of progesterone receptor modulators |
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| AU2007338843B2 (en) * | 2006-12-20 | 2013-05-09 | Teva Women's Health, Inc. | Orally disintegrating solid dosage forms comprising progestin and methods of making and use thereof |
-
2008
- 2008-12-19 EA EA201070715A patent/EA201070715A1/ru unknown
- 2008-12-19 US US12/339,329 patent/US20090170823A1/en not_active Abandoned
- 2008-12-19 EP EP08865187A patent/EP2234491A4/en not_active Withdrawn
- 2008-12-19 WO PCT/US2008/013933 patent/WO2009082478A1/en not_active Ceased
- 2008-12-19 BR BRPI0819571A patent/BRPI0819571A2/pt not_active IP Right Cessation
- 2008-12-19 JP JP2010539503A patent/JP2011507853A/ja active Pending
- 2008-12-19 CA CA2710293A patent/CA2710293A1/en not_active Abandoned
- 2008-12-19 AU AU2008341138A patent/AU2008341138A1/en not_active Abandoned
-
2010
- 2010-06-17 IL IL206465A patent/IL206465A0/en unknown
-
2014
- 2014-06-09 JP JP2014118432A patent/JP2014193918A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| WO2009082478A1 (en) | 2009-07-02 |
| US20090170823A1 (en) | 2009-07-02 |
| JP2011507853A (ja) | 2011-03-10 |
| EP2234491A4 (en) | 2010-12-22 |
| JP2014193918A (ja) | 2014-10-09 |
| IL206465A0 (en) | 2010-12-30 |
| AU2008341138A1 (en) | 2009-07-02 |
| BRPI0819571A2 (pt) | 2019-09-24 |
| EP2234491A1 (en) | 2010-10-06 |
| EA201070715A1 (ru) | 2011-02-28 |
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