JP2011506294A5 - - Google Patents
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- Publication number
- JP2011506294A5 JP2011506294A5 JP2010536469A JP2010536469A JP2011506294A5 JP 2011506294 A5 JP2011506294 A5 JP 2011506294A5 JP 2010536469 A JP2010536469 A JP 2010536469A JP 2010536469 A JP2010536469 A JP 2010536469A JP 2011506294 A5 JP2011506294 A5 JP 2011506294A5
- Authority
- JP
- Japan
- Prior art keywords
- carboxylate
- methyl
- piperazine
- morpholin
- ylmethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0702696 | 2007-12-05 | ||
| US2298308P | 2008-01-23 | 2008-01-23 | |
| PCT/EP2008/066877 WO2009071658A1 (en) | 2007-12-05 | 2008-12-05 | Piperazines as anti-obesity agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2011506294A JP2011506294A (ja) | 2011-03-03 |
| JP2011506294A5 true JP2011506294A5 (enExample) | 2013-02-07 |
Family
ID=40409928
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010536469A Pending JP2011506294A (ja) | 2007-12-05 | 2008-12-05 | 抗肥満薬としてのピペラジン |
Country Status (17)
| Country | Link |
|---|---|
| US (3) | US20110059969A1 (enExample) |
| EP (1) | EP2229362A1 (enExample) |
| JP (1) | JP2011506294A (enExample) |
| KR (1) | KR20100093104A (enExample) |
| CN (1) | CN102026975A (enExample) |
| AU (1) | AU2008333173A1 (enExample) |
| BR (1) | BRPI0819989A2 (enExample) |
| CA (1) | CA2707555A1 (enExample) |
| CO (1) | CO6280487A2 (enExample) |
| CR (1) | CR11479A (enExample) |
| DO (1) | DOP2010000167A (enExample) |
| EA (1) | EA201000926A1 (enExample) |
| EC (1) | ECSP10010234A (enExample) |
| IL (1) | IL205874A0 (enExample) |
| MX (1) | MX2010006259A (enExample) |
| WO (1) | WO2009071658A1 (enExample) |
| ZA (1) | ZA201003976B (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2715527A1 (en) * | 2007-12-05 | 2009-06-11 | Michael Higginbottom | New compounds iv |
| CA2707248A1 (en) * | 2007-12-05 | 2009-06-11 | Astrazeneca Ab | New compounds ii |
| KR101810975B1 (ko) * | 2010-07-08 | 2017-12-20 | 에스케이바이오팜 주식회사 | 카바모일옥시 아릴알칸노일 아릴피페라진계 화합물을 포함하는 약학적 조성물 |
| EP2683716A1 (en) | 2011-03-11 | 2014-01-15 | Glaxo Group Limited | Pyrido[3,4-b]pyrazine derivatives as syk inhibitors |
| US11807622B2 (en) | 2019-01-30 | 2023-11-07 | Insilico Medicine Ip Limited | TLR 9 inhibitors |
| US10689360B1 (en) * | 2019-01-30 | 2020-06-23 | Insilico Medicine Ip Limited | TLR inhibitors |
| CN113149891B (zh) * | 2020-01-07 | 2024-02-02 | 南京药石科技股份有限公司 | 一种2-氨基-2-（1-甲基-4-哌啶基）乙醇的制备方法 |
| CN117777048B (zh) * | 2023-09-25 | 2024-09-20 | 上海科利生物医药有限公司 | 一种手性2-羟甲基吗啉-4-羧酸叔丁酯的制备方法 |
Family Cites Families (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3420193A1 (de) * | 1984-05-30 | 1985-12-05 | Boehringer Ingelheim KG, 6507 Ingelheim | Neue substituierte pyrrolidinone, verfahren zu ihrer herstellung und arzneimittel |
| KR20000016402A (ko) | 1996-06-06 | 2000-03-25 | 피터 기딩스 | 렙틴(ob단백질)의 프레그먼트 |
| US6057337A (en) * | 1998-02-02 | 2000-05-02 | Shiseido Co., Ltd. | 1,2-DI-substituted piperidine derivative, hair growth promoter and external composition for skin using the same |
| JP2001131149A (ja) | 1999-11-08 | 2001-05-15 | Sumitomo Pharmaceut Co Ltd | 選択的セロトニン再取り込み阻害剤 |
| JP2001261657A (ja) | 2000-03-17 | 2001-09-26 | Yamanouchi Pharmaceut Co Ltd | シアノフェニル誘導体 |
| BR0114321A (pt) | 2000-09-29 | 2003-07-01 | Glaxo Group Ltd | Composto, composição farmacêutica, uso de um composto, método de tratamento ou profilaxia de doenças inflamatórias, e, processo para preparar um composto |
| ES2197003B1 (es) * | 2002-04-08 | 2005-03-16 | J. URIACH & CIA S.A. | Nuevos compuestos antagonistas de integrinas alfa. |
| EP1644347A1 (en) | 2003-06-20 | 2006-04-12 | Arena Pharmaceuticals, Inc. | N-PHENYL-PIPERAZINE DERIVATIVES AND METHODS OF PROPHYLAXIS OR TREATMENT OF 5HT sb 2C /sb RECEPTOR ASSOCIATED DISEASES |
| CN102633730A (zh) * | 2004-12-03 | 2012-08-15 | 先灵公司 | 作为cb1拮抗剂的取代哌嗪 |
| DE102005000666B3 (de) | 2005-01-04 | 2006-10-05 | Sanofi-Aventis Deutschland Gmbh | Sulfonylpyrrolidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| US20090325975A1 (en) | 2005-07-15 | 2009-12-31 | Helmut H Buschmann | Use of compounds binding to the sigma receptor for the treatment of diabetes-associated pain |
| EP1787679A1 (en) | 2005-07-29 | 2007-05-23 | Laboratorios Del Dr. Esteve, S.A. | Use of compounds binding to the sigma receptor for the treatment of diabetes-associated pain |
| US7790726B2 (en) | 2005-08-16 | 2010-09-07 | Chemocentryx, Inc. | Monocyclic and bicyclic compounds and methods of use |
| EP1991211A1 (en) | 2006-02-28 | 2008-11-19 | Laboratorios Del Dr. Esteve, S.A. | Use of compounds binding to the sigma receptor for the treatment of metabolic syndrome |
| CA2715527A1 (en) | 2007-12-05 | 2009-06-11 | Michael Higginbottom | New compounds iv |
| CA2707822A1 (en) | 2007-12-05 | 2009-06-11 | Astrazeneca Ab | New compounds iii |
| CA2707248A1 (en) | 2007-12-05 | 2009-06-11 | Astrazeneca Ab | New compounds ii |
| US20110275670A1 (en) | 2008-06-04 | 2011-11-10 | Emma Chapman | New Compounds VII |
| WO2009147211A1 (en) | 2008-06-04 | 2009-12-10 | Biovitrum Ab (Publ) | New compounds v |
| CA2726270A1 (en) | 2008-06-04 | 2009-12-10 | Astrazeneca Ab | Small molecule leptin receptor modulators |
| MX2010013359A (es) | 2008-06-04 | 2011-04-07 | Astrazeneca Ab | Nuevos derivados de piridina como mimeticos moduladores del receptor de leptina. |
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2008
- 2008-12-05 US US12/744,359 patent/US20110059969A1/en not_active Abandoned
- 2008-12-05 CA CA2707555A patent/CA2707555A1/en not_active Abandoned
- 2008-12-05 EP EP08856144A patent/EP2229362A1/en not_active Withdrawn
- 2008-12-05 BR BRPI0819989 patent/BRPI0819989A2/pt not_active IP Right Cessation
- 2008-12-05 JP JP2010536469A patent/JP2011506294A/ja active Pending
- 2008-12-05 WO PCT/EP2008/066877 patent/WO2009071658A1/en not_active Ceased
- 2008-12-05 US US12/315,698 patent/US7851471B2/en not_active Expired - Fee Related
- 2008-12-05 MX MX2010006259A patent/MX2010006259A/es not_active Application Discontinuation
- 2008-12-05 EA EA201000926A patent/EA201000926A1/ru unknown
- 2008-12-05 CN CN2008801266306A patent/CN102026975A/zh active Pending
- 2008-12-05 KR KR1020107014723A patent/KR20100093104A/ko not_active Withdrawn
- 2008-12-05 AU AU2008333173A patent/AU2008333173A1/en not_active Abandoned
-
2010
- 2010-05-20 IL IL205874A patent/IL205874A0/en unknown
- 2010-06-03 ZA ZA2010/03976A patent/ZA201003976B/en unknown
- 2010-06-04 DO DO2010000167A patent/DOP2010000167A/es unknown
- 2010-06-04 CO CO10068022A patent/CO6280487A2/es not_active Application Discontinuation
- 2010-06-04 CR CR11479A patent/CR11479A/es not_active Application Discontinuation
- 2010-06-04 EC EC2010010234A patent/ECSP10010234A/es unknown
- 2010-11-01 US US12/917,085 patent/US20110046135A1/en not_active Abandoned