JP2010539244A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2010539244A5 JP2010539244A5 JP2010525985A JP2010525985A JP2010539244A5 JP 2010539244 A5 JP2010539244 A5 JP 2010539244A5 JP 2010525985 A JP2010525985 A JP 2010525985A JP 2010525985 A JP2010525985 A JP 2010525985A JP 2010539244 A5 JP2010539244 A5 JP 2010539244A5
- Authority
- JP
- Japan
- Prior art keywords
- pain
- compound
- compound according
- acute
- composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 0 C*N(C1CC=CCCCC(C)C1)S(C)(=O)=O Chemical compound C*N(C1CC=CCCCC(C)C1)S(C)(=O)=O 0.000 description 17
- JUJWROOIHBZHMG-UHFFFAOYSA-N c1ccncc1 Chemical compound c1ccncc1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 description 3
- LPAGFVYQRIESJQ-UHFFFAOYSA-N C1c2ccccc2NC1 Chemical compound C1c2ccccc2NC1 LPAGFVYQRIESJQ-UHFFFAOYSA-N 0.000 description 2
- XMSNMAGPGAYJHP-UHFFFAOYSA-N CSCC1c2ccccc2NCC1 Chemical compound CSCC1c2ccccc2NCC1 XMSNMAGPGAYJHP-UHFFFAOYSA-N 0.000 description 2
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US99442307P | 2007-09-19 | 2007-09-19 | |
| PCT/US2008/076928 WO2009039328A1 (en) | 2007-09-19 | 2008-09-19 | Pyridyl sulfonamides as modulators of ion channels |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010539244A JP2010539244A (ja) | 2010-12-16 |
| JP2010539244A5 true JP2010539244A5 (enExample) | 2012-11-29 |
Family
ID=40352214
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010525985A Withdrawn JP2010539244A (ja) | 2007-09-19 | 2008-09-19 | イオンチャネルのモジュレーターとしてのピリジルスルホンアミド |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7994174B2 (enExample) |
| EP (1) | EP2201008A1 (enExample) |
| JP (1) | JP2010539244A (enExample) |
| CN (1) | CN101842372A (enExample) |
| AU (1) | AU2008302205A1 (enExample) |
| CA (1) | CA2699892A1 (enExample) |
| MX (1) | MX2010003009A (enExample) |
| NZ (1) | NZ584009A (enExample) |
| WO (1) | WO2009039328A1 (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7615563B2 (en) * | 2003-08-08 | 2009-11-10 | Gonzalez Iii Jesus E | Compositions useful as inhibitors of voltage-gated sodium channels |
| US7786137B2 (en) | 2005-05-10 | 2010-08-31 | Vertex Pharmaceuticals Incorporated | Bicyclic derivatives as modulators of ion channels |
| KR20080021030A (ko) * | 2005-05-16 | 2008-03-06 | 버텍스 파마슈티칼스 인코포레이티드 | 이온 채널 조절인자로서의 바이사이클릭 유도체 |
| WO2007030618A2 (en) * | 2005-09-09 | 2007-03-15 | Vertex Pharmaceuticals Incorporated | Bicyclic derivatives as modulators of voltage gated ion channels |
| EP1948597A1 (en) * | 2005-10-21 | 2008-07-30 | Vertex Pharmaceuticals Incorporated | Derivatives for modulation of ion channels |
| NZ593074A (en) | 2005-12-21 | 2012-04-27 | Vertex Pharma | sulfonamide-pyrrolidone derivatives as Modulators of Ion Channels |
| EP2604599A1 (en) | 2007-04-27 | 2013-06-19 | Purdue Pharma LP | TRPV1 antagonists and uses thereof |
| NZ581309A (en) | 2007-05-25 | 2012-02-24 | Vertex Pharma | Ion channel modulators and methods of use |
| AU2008321142A1 (en) * | 2007-11-13 | 2009-05-22 | Vertex Pharmaceuticals Incorporated | Heterocyclic derivatives as modulators of ion channels |
| AU2008321137A1 (en) | 2007-11-13 | 2009-05-22 | Vertex Pharmaceuticals Incorporated | 4(-3-(-2-(phenyl)morpholino)-2-oxopyrrolidin-1-yl)-n-(thiazol-2-yl)benzenesulfonamide derivati ves and related compounds as modulators of ion channels for the treatment of pain |
| CN102099356A (zh) * | 2008-07-01 | 2011-06-15 | 沃泰克斯药物股份有限公司 | 用作离子通道调节剂的杂环衍生物 |
| WO2011035332A1 (en) | 2009-09-21 | 2011-03-24 | Chemocentryx, Inc. | Pyrrolidinone carboxamide derivatives as chemerin-r ( chemr23 ) modulators |
| US9273043B2 (en) | 2011-06-22 | 2016-03-01 | Purdue Pharma L.P. | TRPV1 antagonists including dihydroxy substituent and uses thereof |
| EA022973B1 (ru) | 2011-06-27 | 2016-03-31 | Ньюрон Фармасьютикалс С.П.А. | Фторированные арилалкиламинокарбоксамидные производные |
| US10510973B2 (en) * | 2014-12-17 | 2019-12-17 | Universal Display Corporation | Color-stable organic light emitting diode stack |
| EP3886854A4 (en) | 2018-11-30 | 2022-07-06 | Nuvation Bio Inc. | Pyrrole and pyrazole compounds and methods of use thereof |
| US12588382B2 (en) | 2019-07-29 | 2026-03-24 | Universal Display Corporation | Color stable multicolor OLED device structures |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7615356B2 (en) | 2000-07-10 | 2009-11-10 | Vertex Pharmaceuticals (San Diego) Llc | Ion channel assay methods |
| EP1631558A1 (en) | 2003-05-21 | 2006-03-08 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type i |
| TW200524888A (en) * | 2003-08-08 | 2005-08-01 | Vertex Pharma | Compositions useful as inhibitors of voltage-gated ion channels |
| US7615563B2 (en) * | 2003-08-08 | 2009-11-10 | Gonzalez Iii Jesus E | Compositions useful as inhibitors of voltage-gated sodium channels |
| JP2007261945A (ja) | 2004-04-07 | 2007-10-11 | Taisho Pharmaceut Co Ltd | チアゾール誘導体 |
| US7786137B2 (en) * | 2005-05-10 | 2010-08-31 | Vertex Pharmaceuticals Incorporated | Bicyclic derivatives as modulators of ion channels |
| KR20080021030A (ko) * | 2005-05-16 | 2008-03-06 | 버텍스 파마슈티칼스 인코포레이티드 | 이온 채널 조절인자로서의 바이사이클릭 유도체 |
| GT200600196A (es) * | 2005-05-23 | 2007-01-15 | Compuestos n-formil de hidroxilamina | |
| WO2006133459A1 (en) * | 2005-06-09 | 2006-12-14 | Vertex Pharmaceuticals Incorporated | Indane derivatives as modulators of ion channels |
| WO2007030618A2 (en) * | 2005-09-09 | 2007-03-15 | Vertex Pharmaceuticals Incorporated | Bicyclic derivatives as modulators of voltage gated ion channels |
| ES2383090T3 (es) * | 2005-10-12 | 2012-06-18 | Vertex Pharmaceuticals, Inc. | Derivados de bifenilo como moduladores de los canales iónicos dependientes de voltaje |
| EP1948597A1 (en) * | 2005-10-21 | 2008-07-30 | Vertex Pharmaceuticals Incorporated | Derivatives for modulation of ion channels |
| NZ593074A (en) * | 2005-12-21 | 2012-04-27 | Vertex Pharma | sulfonamide-pyrrolidone derivatives as Modulators of Ion Channels |
| AU2008321142A1 (en) * | 2007-11-13 | 2009-05-22 | Vertex Pharmaceuticals Incorporated | Heterocyclic derivatives as modulators of ion channels |
| AU2008321137A1 (en) * | 2007-11-13 | 2009-05-22 | Vertex Pharmaceuticals Incorporated | 4(-3-(-2-(phenyl)morpholino)-2-oxopyrrolidin-1-yl)-n-(thiazol-2-yl)benzenesulfonamide derivati ves and related compounds as modulators of ion channels for the treatment of pain |
| CN102099356A (zh) * | 2008-07-01 | 2011-06-15 | 沃泰克斯药物股份有限公司 | 用作离子通道调节剂的杂环衍生物 |
-
2008
- 2008-09-17 US US12/212,063 patent/US7994174B2/en not_active Expired - Fee Related
- 2008-09-19 NZ NZ584009A patent/NZ584009A/en not_active IP Right Cessation
- 2008-09-19 CA CA2699892A patent/CA2699892A1/en not_active Abandoned
- 2008-09-19 WO PCT/US2008/076928 patent/WO2009039328A1/en not_active Ceased
- 2008-09-19 EP EP08831349A patent/EP2201008A1/en not_active Withdrawn
- 2008-09-19 AU AU2008302205A patent/AU2008302205A1/en not_active Abandoned
- 2008-09-19 CN CN200880113677A patent/CN101842372A/zh active Pending
- 2008-09-19 MX MX2010003009A patent/MX2010003009A/es active IP Right Grant
- 2008-09-19 JP JP2010525985A patent/JP2010539244A/ja not_active Withdrawn
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2011526919A5 (enExample) | ||
| JP2011503112A5 (enExample) | ||
| JP7607732B2 (ja) | 置換ピロロピリミジンｊａｋ阻害剤ならびにこれを作製および使用する方法 | |
| JP2014508756A5 (enExample) | ||
| RU2011103451A (ru) | Гетероциклические производные в качестве модуляторов ионных каналов | |
| JP2010528035A5 (enExample) | ||
| RU2010123781A (ru) | Производные 4-(2-фенил)-морфолино)-2-оксопирролидин-1-ил)-n-(тиазол-2-ил)бензолсульфонамида и родственные соединения в качестве модуляторов ионных каналов для лечения боли | |
| JP2011500598A5 (enExample) | ||
| RU2009100159A (ru) | Тиенопирамидины, полезные в качестве модуляторов ионных каналов | |
| JP2011503191A5 (enExample) | ||
| JP2014504642A5 (enExample) | ||
| RU2010123876A (ru) | Гетероциклические производные в качестве модуляторов ионных каналов | |
| JP2014508169A5 (enExample) | ||
| US9309224B2 (en) | N-acyl-N′-(pyridin-2-yl) ureas and analogs exhibiting anti-cancer and anti-proliferative activities | |
| RU2016104080A (ru) | Амиды конденсированного пиперидина в качестве модуляторов ионных каналов | |
| JP2009544618A5 (enExample) | ||
| MXPA04009784A (es) | Tiazolidin-4-carbonitrilos y analogos y su uso como inhibidores de dipeptidil-peptidas. | |
| JP7331843B2 (ja) | Ｂｔｋ阻害活性を有する化合物を有効成分として含む自己免疫疾患の予防および／または治療剤 | |
| EP4125891A1 (en) | Process, compositions, and crystalline forms of substituted pyridinone-pyridinyl compounds | |
| EA034759B1 (ru) | Пролекарства рилузола и их применение | |
| RU2006101452A (ru) | Пиридазинил-пиперазины и их применение в качестве лигандов h3 гистаминового рецептора | |
| JP2011500599A5 (enExample) | ||
| JP2008511670A5 (enExample) | ||
| EA025086B9 (ru) | Производные индоламида и родственные соединения для использования при лечении нейродегенеративных заболеваний | |
| AU2018251118A1 (en) | Pharmaceutical composition containing MOR agonist and KOR agonist, and uses thereof |