JP2010518026A - ナトリウムチャネルが介在する疾患または状態の治療に有用なピリドピリミジノン化合物 - Google Patents
ナトリウムチャネルが介在する疾患または状態の治療に有用なピリドピリミジノン化合物 Download PDFInfo
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- JP2010518026A JP2010518026A JP2009548501A JP2009548501A JP2010518026A JP 2010518026 A JP2010518026 A JP 2010518026A JP 2009548501 A JP2009548501 A JP 2009548501A JP 2009548501 A JP2009548501 A JP 2009548501A JP 2010518026 A JP2010518026 A JP 2010518026A
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- heteroaryl
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- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US88825307P | 2007-02-05 | 2007-02-05 | |
| US91212207P | 2007-04-16 | 2007-04-16 | |
| PCT/US2008/053075 WO2008097991A1 (en) | 2007-02-05 | 2008-02-05 | Pyridopyrimidinone compounds useful in treating sodium channel-mediated diseases or conditions |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010518026A true JP2010518026A (ja) | 2010-05-27 |
| JP2010518026A5 JP2010518026A5 (OSRAM) | 2012-04-12 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP2009548501A Withdrawn JP2010518026A (ja) | 2007-02-05 | 2008-02-05 | ナトリウムチャネルが介在する疾患または状態の治療に有用なピリドピリミジノン化合物 |
Country Status (12)
| Country | Link |
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| US (1) | US20080194616A1 (OSRAM) |
| EP (1) | EP2079737A1 (OSRAM) |
| JP (1) | JP2010518026A (OSRAM) |
| AR (1) | AR065194A1 (OSRAM) |
| AU (1) | AU2008213836A1 (OSRAM) |
| BR (1) | BRPI0807351A2 (OSRAM) |
| CA (1) | CA2677493A1 (OSRAM) |
| CL (1) | CL2008000369A1 (OSRAM) |
| MX (1) | MX2009008338A (OSRAM) |
| RU (1) | RU2009133336A (OSRAM) |
| TW (1) | TW200838539A (OSRAM) |
| WO (1) | WO2008097991A1 (OSRAM) |
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| KR20150032534A (ko) * | 2012-05-22 | 2015-03-26 | 제넨테크, 인크. | Ｎ-치환된 벤즈아미드 및 통증의 치료에서 이들의 용도 |
| KR20150036367A (ko) * | 2012-07-06 | 2015-04-07 | 제넨테크, 인크. | N-치환된 벤즈아미드 및 이의 사용 방법 |
| JP2016532716A (ja) * | 2013-09-10 | 2016-10-20 | クロモセル コーポレイション | とう痛及び糖尿病の治療用ナトリウムチャネル調節物質 |
| JP2018511627A (ja) * | 2015-04-15 | 2018-04-26 | エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ | Ｎｍｄａ受容体のモジュレーターとしてのピリドピリミジノン及びその使用 |
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| JP2023503290A (ja) * | 2019-11-25 | 2023-01-27 | アムジエン・インコーポレーテツド | デルタ－５デサチュラーゼ阻害剤としての複素環式化合物、及び使用法 |
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| JP2017525677A (ja) | 2014-07-07 | 2017-09-07 | ジェネンテック， インコーポレイテッド | 治療用化合物及びその使用方法 |
| CN117736209A (zh) | 2015-02-27 | 2024-03-22 | 因赛特控股公司 | Pi3k抑制剂的盐及其制备方法 |
| US9732097B2 (en) | 2015-05-11 | 2017-08-15 | Incyte Corporation | Process for the synthesis of a phosphoinositide 3-kinase inhibitor |
| WO2016183063A1 (en) | 2015-05-11 | 2016-11-17 | Incyte Corporation | Crystalline forms of a pi3k inhibitor |
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| JPS63112566A (ja) * | 1986-10-28 | 1988-05-17 | Nissan Chem Ind Ltd | ピリミジノン誘導体、その製法および殺虫・殺ダニ・殺菌剤 |
| JP2007509150A (ja) * | 2003-10-21 | 2007-04-12 | メルク エンド カムパニー インコーポレーテッド | 神経障害性疼痛の治療において有用なトリアゾロ−ピリダジン化合物および、この誘導体 |
| AR053713A1 (es) * | 2005-04-20 | 2007-05-16 | Xenon Pharmaceuticals Inc | Compuestos heterociclicos y sus usos como agentes terapeuticos |
| WO2007002701A2 (en) * | 2005-06-27 | 2007-01-04 | Amgen Inc. | Anti-inflammatory aryl nitrile compounds |
| EP1937678B1 (en) * | 2005-10-04 | 2011-07-27 | Istituto Di Ricerche Di Biologia Molecolare P. Angeletti S.P.A. | Hiv integrase inhibitors |
| EP1818058A3 (en) * | 2006-02-13 | 2007-11-07 | Astion Pharma A/S | Treatment of mmp-mediated dermatological diseases with pemirolast |
-
2008
- 2008-02-05 WO PCT/US2008/053075 patent/WO2008097991A1/en not_active Ceased
- 2008-02-05 CA CA002677493A patent/CA2677493A1/en not_active Abandoned
- 2008-02-05 BR BRPI0807351-1A patent/BRPI0807351A2/pt not_active IP Right Cessation
- 2008-02-05 US US12/026,435 patent/US20080194616A1/en not_active Abandoned
- 2008-02-05 AR ARP080100493A patent/AR065194A1/es unknown
- 2008-02-05 MX MX2009008338A patent/MX2009008338A/es unknown
- 2008-02-05 AU AU2008213836A patent/AU2008213836A1/en not_active Abandoned
- 2008-02-05 EP EP08729067A patent/EP2079737A1/en not_active Withdrawn
- 2008-02-05 TW TW097104675A patent/TW200838539A/zh unknown
- 2008-02-05 JP JP2009548501A patent/JP2010518026A/ja not_active Withdrawn
- 2008-02-05 CL CL200800369A patent/CL2008000369A1/es unknown
- 2008-02-05 RU RU2009133336/04A patent/RU2009133336A/ru unknown
Cited By (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20150032534A (ko) * | 2012-05-22 | 2015-03-26 | 제넨테크, 인크. | Ｎ-치환된 벤즈아미드 및 통증의 치료에서 이들의 용도 |
| KR101719893B1 (ko) * | 2012-05-22 | 2017-03-24 | 제넨테크, 인크. | Ｎ-치환된 벤즈아미드 및 통증의 치료에서 이들의 용도 |
| KR20150036367A (ko) * | 2012-07-06 | 2015-04-07 | 제넨테크, 인크. | N-치환된 벤즈아미드 및 이의 사용 방법 |
| KR101663436B1 (ko) * | 2012-07-06 | 2016-10-06 | 제넨테크, 인크. | N-치환된 벤즈아미드 및 이의 사용 방법 |
| JP2016532716A (ja) * | 2013-09-10 | 2016-10-20 | クロモセル コーポレイション | とう痛及び糖尿病の治療用ナトリウムチャネル調節物質 |
| JP2018511627A (ja) * | 2015-04-15 | 2018-04-26 | エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ | Ｎｍｄａ受容体のモジュレーターとしてのピリドピリミジノン及びその使用 |
| JP2018517754A (ja) * | 2015-06-18 | 2018-07-05 | セファロン、インク． | １，４−置換ピペリジン誘導体 |
| JP6999424B2 (ja) | 2015-06-18 | 2022-01-18 | エイティナイン バイオ リミテッド | １，４－置換ピペリジン誘導体 |
| US11702388B2 (en) | 2015-06-18 | 2023-07-18 | 89Bio Ltd | 1,4-substituted piperidine derivatives |
| US11878966B2 (en) | 2015-06-18 | 2024-01-23 | 89Bio Ltd | Substituted 4-benzyl and 4-benzoyl piperidine derivates |
| US12098130B2 (en) | 2015-06-18 | 2024-09-24 | 89Bio Ltd | 1,4-substituted piperidine derivatives |
| US12441702B2 (en) | 2015-06-18 | 2025-10-14 | Cephalon Llc | Substituted 4-benzyl and 4-benzoyl piperidine derivates |
| JP2023503290A (ja) * | 2019-11-25 | 2023-01-27 | アムジエン・インコーポレーテツド | デルタ－５デサチュラーゼ阻害剤としての複素環式化合物、及び使用法 |
| JP7638987B2 (ja) | 2019-11-25 | 2025-03-04 | アムジエン・インコーポレーテツド | デルタ－５デサチュラーゼ阻害剤としての複素環式化合物、及び使用法 |
Also Published As
| Publication number | Publication date |
|---|---|
| AU2008213836A1 (en) | 2008-08-14 |
| US20080194616A1 (en) | 2008-08-14 |
| RU2009133336A (ru) | 2011-03-20 |
| BRPI0807351A2 (pt) | 2014-05-20 |
| CA2677493A1 (en) | 2008-08-14 |
| MX2009008338A (es) | 2009-08-12 |
| EP2079737A1 (en) | 2009-07-22 |
| WO2008097991A1 (en) | 2008-08-14 |
| AR065194A1 (es) | 2009-05-20 |
| TW200838539A (en) | 2008-10-01 |
| CL2008000369A1 (es) | 2008-04-18 |
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