|
US8039627B2
(en)
|
2006-11-08 |
2011-10-18 |
Neurocrine Biosciences, Inc. |
Substituted 3-isobutyl-9,10-dimethoxy-1,3,4,6,7,11b-hexahydro-2H-pyrido[2,1-A]isoquinolin-2-ol compounds and methods relating thereto
|
|
HUE038158T2
(hu)
|
2008-09-18 |
2018-09-28 |
Auspex Pharmaceuticals Inc |
Deuterizált benzokinolizin származékok vezikuláris monoamin transzporter-2 inhibitorként
|
|
WO2011153157A2
(en)
*
|
2010-06-01 |
2011-12-08 |
Auspex Pharmaceutical, Inc. |
Benzoquinolone inhibitors of vmat2
|
|
WO2012000308A1
(zh)
*
|
2010-06-29 |
2012-01-05 |
中国药科大学 |
丁苯那嗪的拆分方法
|
|
US8351329B2
(en)
*
|
2010-09-14 |
2013-01-08 |
Cisco Technology, Inc. |
Universal load-balancing tunnel encapsulation
|
|
CN102285984B
(zh)
*
|
2010-11-25 |
2012-10-10 |
江苏威凯尔医药科技有限公司 |
(2R,3R,11bR)-二氢丁苯那嗪及相关化合物的制备方法
|
|
WO2012081031A1
(en)
|
2010-12-15 |
2012-06-21 |
Enaltec Labs Pvt. Ltd. |
Process for preparing tetrabenazine
|
|
CA2883641C
(en)
|
2012-09-18 |
2021-09-14 |
Auspex Pharmaceuticals, Inc. |
Formulations pharmacokinetics of deuterated benzoquinoline inhibitors of vesicular monoamine transporter 2
|
|
US9550780B2
(en)
|
2012-09-18 |
2017-01-24 |
Auspex Pharmaceuticals, Inc. |
Formulations pharmacokinetics of deuterated benzoquinoline inhibitors of vesicular monoamine transporter 2
|
|
MX2015009719A
(es)
*
|
2013-01-31 |
2016-08-08 |
Auspex Pharmaceuticals Inc |
Inhibidores benzoquinolona de vmat2.
|
|
HK1221645A1
(zh)
*
|
2013-09-27 |
2017-06-09 |
Auspex Pharmaceuticals, Inc. |
Vmat2的苯并喹啉抑制剂
|
|
CN105873589B
(zh)
*
|
2013-12-03 |
2019-11-01 |
奥斯拜客斯制药有限公司 |
制造苯并喹啉化合物的方法
|
|
KR20160111999A
(ko)
*
|
2014-01-27 |
2016-09-27 |
오스펙스 파마슈티칼스, 인코포레이티드 |
소포성 모노아민 수송체 2의 벤조퀴놀린 억제제
|
|
CN113413385A
(zh)
|
2014-02-07 |
2021-09-21 |
纽罗克里生物科学有限公司 |
包含抗精神病药物和vmat2抑制剂的药物组合物及其用途
|
|
KR20160117596A
(ko)
|
2014-02-07 |
2016-10-10 |
오스펙스 파마슈티칼스, 인코포레이티드 |
신규 제약 제제
|
|
CN106164066B
(zh)
|
2014-02-13 |
2020-01-17 |
因赛特公司 |
作为lsd1抑制剂的环丙胺
|
|
DK3936130T3
(da)
*
|
2014-05-06 |
2024-03-25 |
Neurocrine Biosciences Inc |
Doseringsskema for Valbenazin til behandling af hyperkinetiske bevægelsesforstyrrelser
|
|
AU2016215033B2
(en)
*
|
2015-02-06 |
2020-06-25 |
Neurocrine Biosciences, Inc. |
(9,10-dimethoxy-3-(2-methylpropyl)-1H,2H,3H,4H,6H,7H,11bH-pyrido-[2,1-a]isoquinolin-2-yl]methanol and compounds, compositions and methods relating thereto
|
|
JP6932641B2
(ja)
|
2015-03-06 |
2021-09-08 |
オースペックス ファーマシューティカルズ インコーポレイテッド |
異常不随意運動障害の処置のための方法
|
|
CN107660205B
(zh)
|
2015-04-03 |
2021-08-27 |
因赛特公司 |
作为lsd1抑制剂的杂环化合物
|
|
JP6919099B2
(ja)
*
|
2015-06-23 |
2021-08-18 |
ニューロクライン バイオサイエンシーズ,インコーポレイテッド |
神経学的疾患または障害を処置するためのvmat2阻害剤
|
|
EA035534B1
(ru)
|
2015-08-12 |
2020-06-30 |
Инсайт Корпорейшн |
Соли ингибитора lsd1
|
|
WO2017060870A1
(en)
|
2015-10-09 |
2017-04-13 |
Hermann Russ |
Combination of deuterated levodopa with carbidopa and opicapone for the treatment of parkinson`s disease
|
|
HRP20240304T1
(hr)
*
|
2015-10-30 |
2024-05-10 |
Neurocrine Biosciences, Inc. |
Soli valbenazin dihidroklorida i njihovi polimorfi
|
|
LT3394057T
(lt)
|
2015-12-23 |
2022-06-27 |
Neurocrine Biosciences, Inc. |
Sintezės būdas, skirtas pagaminti (s)-(2r,3r,11br)-3-izobutil-9,10-dimetoksi-2,3,4,6,7,11b-heksahidro-1h-pirido[2,1-a]izochinolin-2-ilo 2-amino-3-metilbutanoato di(4-metilbenzensulfonatą)
|
|
WO2017182916A1
(en)
*
|
2016-04-22 |
2017-10-26 |
Lupin Limited |
Novel process for preparation of tetrabenazine and deutetrabenazine
|
|
ES2811048T3
(es)
|
2016-06-29 |
2021-03-10 |
Crystal Pharmaceutical Suzhou Co Ltd |
Formas cristalinas de NBI-98854, método de preparación para las mismas y uso de las mismas
|
|
EP3523300A1
(en)
*
|
2016-10-06 |
2019-08-14 |
Assia Chemical Industries Ltd. |
Solid state forms of valbenazine
|
|
EP4400171A3
(en)
|
2016-12-02 |
2024-09-11 |
Neurocrine Biosciences, Inc. |
Use of valbenazine for treating schizophrenia or schizoaffective disorder
|
|
US10703750B2
(en)
|
2017-01-10 |
2020-07-07 |
Sandoz Ag |
Crystalline valbenazine free base
|
|
KR20190108146A
(ko)
|
2017-01-27 |
2019-09-23 |
뉴로크린 바이오사이언시즈 인코퍼레이티드 |
특정 vmat2 억제제의 투여 방법
|
|
CA3054238A1
(en)
|
2017-02-27 |
2018-08-30 |
Sandoz Ag |
Crystalline forms of valbenazine salts
|
|
WO2018164996A1
(en)
|
2017-03-06 |
2018-09-13 |
Neurocrine Biosciences, Inc. |
Dosing regimen for valbenazine
|
|
KR20230003308A
(ko)
|
2017-03-15 |
2023-01-05 |
오스펙스 파마슈티칼스, 인코포레이티드 |
듀테트라베나진의 유사체, 이의 제조 및 용도
|
|
GB201705306D0
(en)
|
2017-04-01 |
2017-05-17 |
Adeptio Pharmaceuticals Ltd |
Pharmaceutical compositions
|
|
GB201705302D0
(en)
|
2017-04-01 |
2017-05-17 |
Adeptio Pharmaceuticals Ltd |
Pharmaceutical compositions
|
|
JP7250692B2
(ja)
*
|
2017-04-01 |
2023-04-03 |
アデプティオ ファーマシューティカルズ リミテッド |
運動障害の治療における使用のためのジヒドロテトラベナジン
|
|
GB201705304D0
(en)
|
2017-04-01 |
2017-05-17 |
Adeptio Pharmaceuticals Ltd |
Pharmaceutical compositions
|
|
GB201705303D0
(en)
|
2017-04-01 |
2017-05-17 |
Adeptio Pharmaceuticals Ltd |
Pharmaceutical compositions
|
|
JOP20190239A1
(ar)
*
|
2017-04-19 |
2019-10-09 |
Neurocrine Biosciences Inc |
مركبات مثبطة لـ vmat2 وتركيبات منها
|
|
US20200179352A1
(en)
|
2017-04-26 |
2020-06-11 |
Neurocrine Biosciences, Inc. |
Use of valbenazine for treating levodopa-induced dyskinesia
|
|
IL309802A
(en)
|
2017-09-21 |
2024-02-01 |
Neurocrine Biosciences Inc |
High dose valbenazine formulation and related preparations, methods and kits
|
|
JP2021502959A
(ja)
|
2017-10-10 |
2021-02-04 |
ニューロクライン バイオサイエンシーズ,インコーポレイテッド |
特定のvmat2インヒビターを投与するための方法
|
|
KR20250070134A
(ko)
|
2017-10-10 |
2025-05-20 |
뉴로크린 바이오사이언시즈 인코퍼레이티드 |
특정 vmat2 억제제의 투여 방법
|
|
CA3081709A1
(en)
*
|
2017-11-08 |
2019-05-16 |
Yuhua Li |
Esters of dihydrotetrabenazine
|
|
WO2019104141A1
(en)
|
2017-11-22 |
2019-05-31 |
Teva Pharmaceuticals Usa, Inc. |
Solid state form of valbenazine
|
|
EP3733666B1
(en)
|
2017-12-26 |
2022-09-21 |
Crystal Pharmaceutical (Suzhou) Co., Ltd. |
Crystal form of valbenazine di-p-toluenesulfonate, preparation method thereof and use thereof
|
|
CN110092785A
(zh)
*
|
2018-01-31 |
2019-08-06 |
广东东阳光药业有限公司 |
一种丁苯那嗪的动态拆分方法
|
|
GB201808464D0
(en)
|
2018-05-23 |
2018-07-11 |
Adeptio Pharmaceuticals Ltd |
Pharmaceutical compounds for use in treating huntington's disease
|
|
WO2019241555A1
(en)
*
|
2018-06-14 |
2019-12-19 |
Neurocrine Biosciences, Inc. |
Vmat2 inhibitor compounds, compositions, and methods relating thereto
|
|
JOP20200336A1
(ar)
|
2018-08-15 |
2020-12-22 |
Neurocrine Biosciences Inc |
طرق إعطاء مثبطات vmat2 معينة
|
|
US10968200B2
(en)
|
2018-08-31 |
2021-04-06 |
Incyte Corporation |
Salts of an LSD1 inhibitor and processes for preparing the same
|
|
WO2020070236A1
(en)
|
2018-10-04 |
2020-04-09 |
Adeptio Pharmaceuticals Limited |
(+)-alpha-dihydrotetrabenazine dosage regimen for treating movement disorders
|
|
CA3065236A1
(en)
|
2018-12-27 |
2020-06-27 |
Apotex Inc. |
Novel crystalline form of valbenazine dibesylate
|
|
WO2020213014A1
(en)
|
2019-04-19 |
2020-10-22 |
Mylan Laboratories Limited |
An improved process for the preparation of valbenazine and its salts
|
|
US10689380B1
(en)
|
2019-07-30 |
2020-06-23 |
Farmhispania S.A. |
Crystalline forms of valbenazine ditosylate
|
|
WO2021027792A1
(zh)
*
|
2019-08-12 |
2021-02-18 |
山东绿叶制药有限公司 |
Vmat2抑制剂及其制备方法和应用
|
|
US10940141B1
(en)
|
2019-08-23 |
2021-03-09 |
Neurocrine Biosciences, Inc. |
Methods for the administration of certain VMAT2 inhibitors
|
|
CA3150961A1
(en)
|
2019-09-13 |
2021-03-18 |
John Tucker |
Processes for the synthesis of valbenazine
|
|
CN110698397A
(zh)
*
|
2019-10-28 |
2020-01-17 |
南京红杉生物科技有限公司 |
丁苯那嗪中间体及其合成方法、应用和合成用中间产物
|
|
JP2024511053A
(ja)
|
2021-03-22 |
2024-03-12 |
ニューロクライン バイオサイエンシーズ,インコーポレイテッド |
Vmat2阻害剤および使用方法
|
|
US20240239791A1
(en)
|
2021-04-26 |
2024-07-18 |
Neurocrine Biosciences, Inc. |
Processes for the synthesis of valbenazine
|
|
AU2022302155A1
(en)
|
2021-06-30 |
2024-02-08 |
Neurocrine Biosciences, Inc. |
Valbenazine for use in the treatment of dyskinesia due to cerebral palsy
|
|
JP2024524324A
(ja)
|
2021-06-30 |
2024-07-05 |
ニューロクライン バイオサイエンシーズ,インコーポレイテッド |
統合失調症のアドオン処置において使用するためのバルベナジン
|
|
WO2023172849A1
(en)
|
2022-03-07 |
2023-09-14 |
Neurocrine Biosciences, Inc. |
Valbenazine, a vmat2 inhibitor, as a free base a tosylate or ditosylate salt, for use in the treatment of chorea associated with huntington's disease
|
|
CN119907800A
(zh)
|
2022-09-21 |
2025-04-29 |
纽罗克里生物科学有限公司 |
六氢-2H-吡啶并[2,1-a]异喹啉VMAT2抑制剂及其使用方法
|
|
WO2025038938A1
(en)
|
2023-08-17 |
2025-02-20 |
Neurocrine Biosciences, Inc. |
Valbenazine for use in the treatment of huntington's chorea
|
|
WO2025038959A1
(en)
|
2023-08-17 |
2025-02-20 |
Neurocrine Biosciences, Inc. |
Methods for the administration of certain vmat2 inhibitors
|
|
WO2025096823A1
(en)
|
2023-11-01 |
2025-05-08 |
Neurocrine Biosciences, Inc. |
Improvement, maintenance or reduction of decline of motor function associated with huntington disease using valbenazine
|
|
WO2025188830A1
(en)
|
2024-03-06 |
2025-09-12 |
Neurocrine Biosciences, Inc. |
Methods for the administration of certain vmat2 inhibitors
|
|
WO2025199234A1
(en)
|
2024-03-20 |
2025-09-25 |
Neurocrine Biosciences, Inc. |
Vmat2 inhibitors and methods of use
|