JP2010505940A5 - - Google Patents

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Publication number
JP2010505940A5
JP2010505940A5 JP2009531969A JP2009531969A JP2010505940A5 JP 2010505940 A5 JP2010505940 A5 JP 2010505940A5 JP 2009531969 A JP2009531969 A JP 2009531969A JP 2009531969 A JP2009531969 A JP 2009531969A JP 2010505940 A5 JP2010505940 A5 JP 2010505940A5
Authority
JP
Japan
Prior art keywords
phenyl
piperazine
carbonyl
amino
butyryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2009531969A
Other languages
English (en)
Japanese (ja)
Other versions
JP2010505940A (ja
JP5341763B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2007/054155 external-priority patent/WO2008044217A2/en
Publication of JP2010505940A publication Critical patent/JP2010505940A/ja
Publication of JP2010505940A5 publication Critical patent/JP2010505940A5/ja
Application granted granted Critical
Publication of JP5341763B2 publication Critical patent/JP5341763B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2009531969A 2006-10-13 2007-10-12 2−アミノカルボニル−ピリジン誘導体 Expired - Fee Related JP5341763B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IB2006053773 2006-10-13
IBPCT/IB2006/053773 2006-10-13
IBPCT/IB2006/053817 2006-10-17
IB2006053817 2006-10-17
PCT/IB2007/054155 WO2008044217A2 (en) 2006-10-13 2007-10-12 2-aminocarbonyl-pyridine derivatives

Publications (3)

Publication Number Publication Date
JP2010505940A JP2010505940A (ja) 2010-02-25
JP2010505940A5 true JP2010505940A5 (OSRAM) 2013-07-11
JP5341763B2 JP5341763B2 (ja) 2013-11-13

Family

ID=39167796

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009531969A Expired - Fee Related JP5341763B2 (ja) 2006-10-13 2007-10-12 2−アミノカルボニル−ピリジン誘導体

Country Status (17)

Country Link
US (1) US8093250B2 (OSRAM)
EP (1) EP2081903B1 (OSRAM)
JP (1) JP5341763B2 (OSRAM)
KR (1) KR101525260B1 (OSRAM)
AR (1) AR063258A1 (OSRAM)
AU (1) AU2007305925A1 (OSRAM)
BR (1) BRPI0720193A2 (OSRAM)
CA (1) CA2664579C (OSRAM)
CL (1) CL2007002920A1 (OSRAM)
ES (1) ES2473609T3 (OSRAM)
IL (1) IL198059A0 (OSRAM)
MA (1) MA30868B1 (OSRAM)
MX (1) MX2009003724A (OSRAM)
NO (1) NO20091838L (OSRAM)
RU (1) RU2009117705A (OSRAM)
TW (1) TW200823190A (OSRAM)
WO (1) WO2008044217A2 (OSRAM)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200640877A (en) 2005-04-28 2006-12-01 Actelion Pharmaceuticals Ltd Pyrimidine derivatives
AR063258A1 (es) 2006-10-13 2009-01-14 Actelion Pharmaceuticals Ltd Derivados de 2-aminocarbonil-piridina, una composicion farmaceutica que los contiene y su uso en la preparacion de un medicamento para el tratamiento de trastornos vasculares oclusivos.
AR063518A1 (es) 2006-10-25 2009-01-28 Actelion Pharmaceuticals Ltd Derivados 2-fenil-6-aminocarbonil-pirimidina; composicion farmaceutica; y su uso para tratar y/o prevenir enfermedades vasculares perifericas viscerales, hepaticas y renales, enfermedades cardiovasculares y enfermedades cerebrovasculares asociados con la agregacion de plaquetas, incluyendo trombosis
TWI361690B (en) 2007-11-29 2012-04-11 Actelion Pharmaceuticals Ltd Phosphonic acid derivatives
EP2262766B1 (en) 2008-02-29 2015-11-11 Evotec AG Amide compounds, compositions and uses thereof
AR071653A1 (es) 2008-04-11 2010-07-07 Actelion Pharmaceuticals Ltd Derivados 2-fenil-4-ciclopropil-pirimidina
AR071652A1 (es) 2008-04-11 2010-07-07 Actelion Pharmaceuticals Ltd Derivados 2- fenil-piridina substituidos
US20110237578A1 (en) 2008-09-18 2011-09-29 Zhi-Liang Wei Amide compounds, compositions and uses thereof
WO2010116328A2 (en) 2009-04-08 2010-10-14 Actelion Pharmaceuticals Ltd 6-(3-aza-bicyclo[3.1.0]hex-3-yl)-2-phenyl-pyrimidines
EP2421859B1 (en) * 2009-04-22 2014-04-09 Actelion Pharmaceuticals Ltd. Thiazole derivatives and their use as p2y12 receptor antagonists
EP2593434A1 (en) * 2010-07-16 2013-05-22 Purdue Pharma LP Pyridine compounds as sodium channel blockers
WO2013033178A1 (en) 2011-08-30 2013-03-07 University Of Utah Research Foundation Methods and compositions for treating nephrogenic diabetes insipidus
AU2013203824A1 (en) 2012-03-16 2013-10-03 Purdue Pharma L.P. Substituted pyridines and pryimidines as sodium channel blockers
US9714252B2 (en) 2012-12-20 2017-07-25 Purdue Pharma L.P. Cyclic sulfonamides as sodium channel blockers
US10730866B2 (en) 2014-04-07 2020-08-04 Purdue Pharma L.P. Indole derivatives and use thereof
HUE057772T2 (hu) 2016-09-22 2022-06-28 Idorsia Pharmaceuticals Ltd Kristályos formák
KR102510832B1 (ko) 2017-03-15 2023-03-15 이도르시아 파마슈티컬스 리미티드 P2y12 수용체 안타고니스트의 피하 투여

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5373586A (en) 1976-12-09 1978-06-30 Mitsubishi Chem Ind Ltd New penicillin derivatives
CA2020437A1 (en) 1989-07-05 1991-01-06 Yoshihide Fuse Cinnamamide derivative
IL123986A (en) * 1997-04-24 2011-10-31 Organon Nv Medicinal compounds
WO1999006402A1 (en) * 1997-07-31 1999-02-11 Ube Industries, Ltd. N-acylamino acid amide compounds and intermediates for preparation thereof
CA2375920A1 (en) * 1999-06-14 2000-12-21 Eli Lilly And Company Compounds
US6861424B2 (en) 2001-06-06 2005-03-01 Schering Aktiengesellschaft Platelet adenosine diphosphate receptor antagonists
KR20050085580A (ko) * 2002-12-11 2005-08-29 쉐링 악티엔게젤샤프트 혈소판 아데노신 디포스페이트 수용체 길항제로서의2-아미노카르보닐-퀴놀린 화합물
TW200640877A (en) 2005-04-28 2006-12-01 Actelion Pharmaceuticals Ltd Pyrimidine derivatives
AU2006305538B2 (en) * 2005-10-21 2012-06-28 Idorsia Pharmaceuticals Ltd Piperazine derivatives as antimalarial agents
AR063258A1 (es) 2006-10-13 2009-01-14 Actelion Pharmaceuticals Ltd Derivados de 2-aminocarbonil-piridina, una composicion farmaceutica que los contiene y su uso en la preparacion de un medicamento para el tratamiento de trastornos vasculares oclusivos.
AR063518A1 (es) 2006-10-25 2009-01-28 Actelion Pharmaceuticals Ltd Derivados 2-fenil-6-aminocarbonil-pirimidina; composicion farmaceutica; y su uso para tratar y/o prevenir enfermedades vasculares perifericas viscerales, hepaticas y renales, enfermedades cardiovasculares y enfermedades cerebrovasculares asociados con la agregacion de plaquetas, incluyendo trombosis
TWI361690B (en) 2007-11-29 2012-04-11 Actelion Pharmaceuticals Ltd Phosphonic acid derivatives
AR071652A1 (es) 2008-04-11 2010-07-07 Actelion Pharmaceuticals Ltd Derivados 2- fenil-piridina substituidos
AR071653A1 (es) 2008-04-11 2010-07-07 Actelion Pharmaceuticals Ltd Derivados 2-fenil-4-ciclopropil-pirimidina
WO2010116328A2 (en) 2009-04-08 2010-10-14 Actelion Pharmaceuticals Ltd 6-(3-aza-bicyclo[3.1.0]hex-3-yl)-2-phenyl-pyrimidines
EP2421859B1 (en) 2009-04-22 2014-04-09 Actelion Pharmaceuticals Ltd. Thiazole derivatives and their use as p2y12 receptor antagonists

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