JP2010504913A - 炎症及び免疫関連使用のための縮合環化合物 - Google Patents

炎症及び免疫関連使用のための縮合環化合物 Download PDF

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JP2010504913A
JP2010504913A JP2009529277A JP2009529277A JP2010504913A JP 2010504913 A JP2010504913 A JP 2010504913A JP 2009529277 A JP2009529277 A JP 2009529277A JP 2009529277 A JP2009529277 A JP 2009529277A JP 2010504913 A JP2010504913 A JP 2010504913A
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JP2010504913A5 (OSRAM
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フウ ボ,ニャ
チェ,クィンリン
チェン,ショウジュン
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シンタ ファーマシューティカルズ コーポレーション
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    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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  • Obesity (AREA)
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  • Pain & Pain Management (AREA)
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  • Ophthalmology & Optometry (AREA)
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JP2009529277A 2006-09-26 2007-09-26 炎症及び免疫関連使用のための縮合環化合物 Ceased JP2010504913A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US84732506P 2006-09-26 2006-09-26
US11/861,278 US8779154B2 (en) 2006-09-26 2007-09-25 Fused ring compounds for inflammation and immune-related uses
PCT/US2007/020864 WO2008039520A2 (en) 2006-09-26 2007-09-26 Fused ring compounds for inflammation and immune-related uses

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JP2010504913A true JP2010504913A (ja) 2010-02-18
JP2010504913A5 JP2010504913A5 (OSRAM) 2011-08-18

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US (1) US8779154B2 (OSRAM)
EP (1) EP2086983A4 (OSRAM)
JP (1) JP2010504913A (OSRAM)
AU (1) AU2007300450B2 (OSRAM)
CA (1) CA2664301A1 (OSRAM)
WO (1) WO2008039520A2 (OSRAM)

Cited By (3)

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JP2011509261A (ja) * 2008-01-07 2011-03-24 シンタ ファーマシューティカルズ コーポレーション 炎症および免疫関連用途向けの化合物
JP2011517457A (ja) * 2008-03-31 2011-06-09 ジェネンテック, インコーポレイテッド ベンゾピランおよびベンゾキセピンpi3k阻害剤化合物および使用方法
JP2016510752A (ja) * 2013-03-06 2016-04-11 ヤンセン ファーマシューティカ エヌ.ベー. ヒスタミンh4受容体のベンゾイミダゾール−2−イルピリミジンモジュレータ

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US8119643B2 (en) * 2006-03-20 2012-02-21 Synta Pharmaceuticals Corp. Benzoimidazolyl-pyrazine compounds for inflammation and immune-related uses
RS51423B (sr) 2006-03-31 2011-02-28 Janssen Pharmaceutica N.V. Benzoimidazol-2-il pirimidini i pirazini kao modulatori histaminskog h4 receptora
US9371311B2 (en) 2008-06-30 2016-06-21 Janssen Pharmaceutica Nv Benzoimidazol-2-yl pyrimidine derivatives
US8288379B2 (en) * 2009-04-22 2012-10-16 Boehringer Ingelheim International Gmbh Thia-triaza-cyclopentazulenes
RU2600927C2 (ru) 2009-09-28 2016-10-27 Ф.Хоффманн-Ля Рош Аг Бензоксазепиновые ингибиторы pi3k и способы применения
PE20140918A1 (es) * 2009-09-28 2014-08-06 Hoffmann La Roche Compuestos de benzoxepina inhibidores de la pi3k
US8993612B2 (en) 2009-10-08 2015-03-31 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel and methods for treatment of non-small cell lung cancer
US8377970B2 (en) 2009-10-08 2013-02-19 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel
EP2493866A1 (en) * 2009-10-29 2012-09-05 Bristol-Myers Squibb Company Tricyclic heterocyclic compounds
JP2013511279A (ja) 2009-11-20 2013-04-04 アムジエン・インコーポレーテツド 抗Orai1抗原結合蛋白及びその使用
RU2013143747A (ru) 2011-03-21 2015-04-27 Ф. Хоффманн-Ля Рош Аг Соединения бензоксазепина, селективные в отношении pi3k p110 дельта и способы их применения
WO2013113863A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
WO2013113716A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
WO2013113773A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
WO2013113791A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
CN104220428A (zh) 2012-02-03 2014-12-17 巴斯夫欧洲公司 杀真菌嘧啶化合物
WO2013113776A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
WO2013135672A1 (en) 2012-03-13 2013-09-19 Basf Se Fungicidal pyrimidine compounds
EA201491667A1 (ru) 2012-03-13 2015-03-31 Басф Се Фунгицидные соединения пиримидина
EP2738172A1 (en) 2012-11-28 2014-06-04 Almirall, S.A. New bicyclic compounds as crac channel modulators
WO2014118099A1 (en) 2013-01-30 2014-08-07 Basf Se Fungicidal naphthoquinones and derivatives
EP2848615A1 (en) 2013-07-03 2015-03-18 Almirall, S.A. New pyrazole derivatives as CRAC channel modulators
JP7029445B2 (ja) 2016-09-02 2022-03-03 ブリストル-マイヤーズ スクイブ カンパニー 置換された三環式ヘテロ環化合物
CA3063288A1 (en) 2017-05-12 2018-11-15 Mavalon Therapeutics Limited Substituted heterocyclic compounds as allosteric modulators of group ii metabotropic glutamate receptors
WO2019032632A1 (en) 2017-08-09 2019-02-14 Bristol-Myers Squibb Company ALKYLPHENYL COMPOUNDS
US11059784B2 (en) 2017-08-09 2021-07-13 Bristol-Myers Squibb Company Oxime ether compounds
BR112021004893A2 (pt) 2018-09-14 2021-06-01 Rhizen Pharmaceuticals A G composições compreendendo um inibidor de crac e um corticosteroide e métodos de uso dos mesmos
AU2021207804A1 (en) 2020-01-13 2022-09-01 Verge Analytics, Inc. Substituted pyrazolo-pyrimidines and uses thereof
CN114621070B (zh) * 2022-04-02 2024-03-19 上海陶术生物科技有限公司 3,4-二氢萘-1(2h)-酮衍生物的合成方法
WO2025082467A1 (zh) * 2023-10-19 2025-04-24 成都先导药物开发股份有限公司 一种免疫调节剂

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