JP2009541415A5 - - Google Patents

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Publication number
JP2009541415A5
JP2009541415A5 JP2009517107A JP2009517107A JP2009541415A5 JP 2009541415 A5 JP2009541415 A5 JP 2009541415A5 JP 2009517107 A JP2009517107 A JP 2009517107A JP 2009517107 A JP2009517107 A JP 2009517107A JP 2009541415 A5 JP2009541415 A5 JP 2009541415A5
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JP
Japan
Prior art keywords
alkyl
cycloalkyl
tetrazol
hetero
halo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2009517107A
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English (en)
Japanese (ja)
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JP5021734B2 (ja
JP2009541415A (ja
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Priority claimed from PCT/EP2007/055997 external-priority patent/WO2008000645A1/en
Publication of JP2009541415A publication Critical patent/JP2009541415A/ja
Publication of JP2009541415A5 publication Critical patent/JP2009541415A5/ja
Application granted granted Critical
Publication of JP5021734B2 publication Critical patent/JP5021734B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009517107A 2006-06-29 2007-06-18 テトラゾール置換アリールアミド Active JP5021734B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US81729806P 2006-06-29 2006-06-29
US60/817,298 2006-06-29
PCT/EP2007/055997 WO2008000645A1 (en) 2006-06-29 2007-06-18 Tetrazole-substituted arylamides

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2012134357A Division JP5456846B2 (ja) 2006-06-29 2012-06-14 テトラゾール置換アリールアミド

Publications (3)

Publication Number Publication Date
JP2009541415A JP2009541415A (ja) 2009-11-26
JP2009541415A5 true JP2009541415A5 (https=) 2012-06-07
JP5021734B2 JP5021734B2 (ja) 2012-09-12

Family

ID=38462418

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2009517107A Active JP5021734B2 (ja) 2006-06-29 2007-06-18 テトラゾール置換アリールアミド
JP2012134357A Active JP5456846B2 (ja) 2006-06-29 2012-06-14 テトラゾール置換アリールアミド

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2012134357A Active JP5456846B2 (ja) 2006-06-29 2012-06-14 テトラゾール置換アリールアミド

Country Status (15)

Country Link
US (5) US7595405B2 (https=)
EP (2) EP2592070B1 (https=)
JP (2) JP5021734B2 (https=)
KR (1) KR101103143B1 (https=)
CN (2) CN103159692B (https=)
AR (1) AR061667A1 (https=)
AU (1) AU2007263809B2 (https=)
BR (2) BRPI0714315B8 (https=)
CA (1) CA2654915C (https=)
CL (1) CL2007001887A1 (https=)
ES (2) ES2604542T3 (https=)
IL (2) IL195786A (https=)
MX (1) MX2008016423A (https=)
TW (1) TWI334414B (https=)
WO (1) WO2008000645A1 (https=)

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ES2417182T3 (es) 2007-12-17 2013-08-06 F. Hoffmann-La Roche Ag Nuevas arilamidas sustituidas con pirazol
ES2542245T3 (es) * 2007-12-17 2015-08-03 F. Hoffmann-La Roche Ag Derivados de arilamida sustituido con triazol y su utilización como antagonistas del receptor purinérgico P2x3 y/o P2x2/3
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CA2737038A1 (en) * 2008-09-18 2010-03-25 Evotec Ag Amide compounds, compositions and uses thereof
ES2534199T3 (es) * 2008-10-31 2015-04-20 Merck Sharp & Dohme Corp. Antagonistas del receptor P2X3 para el tratamiento del dolor
EP2379518B1 (en) 2008-12-16 2014-05-07 F. Hoffmann-La Roche AG Thiadiazole-substituted arylamides
AU2010229144B2 (en) 2009-03-23 2012-07-12 Merck Sharp & Dohme Corp. P2X3, receptor antagonists for treatment of pain
US8946231B2 (en) 2009-03-23 2015-02-03 Merck Sharp & Dohme Corp. P2X3, receptor antagonists for treatment of pain
WO2010111058A1 (en) 2009-03-23 2010-09-30 Merck Sharp & Dohme Corp. P2x3, receptor antagonists for treatment of pain
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EP2435407B1 (en) * 2009-05-29 2019-12-25 RaQualia Pharma Inc. Aryl substituted carboxamide derivatives as calcium or sodium channel blockers
AR077033A1 (es) * 2009-06-11 2011-07-27 Hoffmann La Roche Compuestos inhibidores de las quinasas de janus y su uso en el tratamiento de enfermedades inmunologicas
US8476457B2 (en) 2009-06-22 2013-07-02 Roche Palo Alto Llc Indole, indazole and benzimidazole arylamides as P2X3 and P2X2/3 antagonists
EP2445889B1 (en) * 2009-06-22 2016-08-10 F.Hoffmann-La Roche Ag Novel benzoxazolone -substituted arylamides
CN102574778B (zh) * 2009-06-22 2015-01-07 弗·哈夫曼-拉罗切有限公司 新的联苯基和苯基-吡啶酰胺类化合物
AU2011261375B2 (en) * 2010-06-04 2016-09-22 Albany Molecular Research, Inc. Glycine transporter-1 inhibitors, methods of making them, and uses thereof
US9598409B2 (en) * 2013-01-31 2017-03-21 Neomed Institute Imidazopyridine compounds and uses thereof
HUE058009T2 (hu) 2014-12-09 2022-06-28 Bayer Ag 1,3-Tiazol-2-il szubsztituált benzamid-származékok
US10183937B2 (en) 2014-12-09 2019-01-22 Bayer Aktiengesellschaft 1,3-thiazol-2-yl substituted benzamides
CN107207449B (zh) * 2015-04-23 2020-11-10 豪夫迈·罗氏有限公司 用于治疗精神障碍的四唑衍生物
JP6877359B2 (ja) * 2015-06-04 2021-05-26 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ イミダゾール誘導体
CN108137566B (zh) * 2015-10-06 2021-05-25 豪夫迈·罗氏有限公司 三唑衍生物
EP3411365B1 (en) 2016-02-02 2019-11-20 H. Hoffnabb-La Roche Ag Pyrazol-pyridine derivatives as eaat3 inhibitors
TWI696615B (zh) * 2016-05-05 2020-06-21 瑞士商伊蘭科動物健康公司 雜芳基-1,2,4-三唑及雜芳基-三唑化合物
EP3464246B1 (en) 2016-05-27 2020-07-08 H. Hoffnabb-La Roche Ag Pyrazol compounds as eaat3 inhibitors
CN109563049B (zh) 2016-10-14 2022-11-29 豪夫迈·罗氏有限公司 作为eaat3抑制剂的咪唑化合物
TWI741040B (zh) * 2016-10-20 2021-10-01 德商拜耳作物科學公司 製備3-烷基硫基-2-氯-n-(1-烷基-1h-四唑-5-基)-4-三氟甲基苯甲醯胺之方法
RU2650780C1 (ru) 2016-12-06 2018-04-17 Общество с ограниченной ответственностью "Анальгетики будущего" Пептидный модулятор пуринергических рецепторов
CN114222741B (zh) 2019-05-31 2025-12-30 奇斯药制品公司 作为p2x3抑制剂的吡啶并嘧啶类衍生物
BR112021022099A2 (pt) 2019-05-31 2021-12-28 Chiesi Farm Spa Derivados de amino quinazolina como inibidores de p2x3
JP2023550830A (ja) 2020-11-27 2023-12-05 キエシ・フアルマチエウテイチ・ソチエタ・ペル・アチオニ Ｐ２ｘ３阻害剤としての（アザ）キノリン４－アミン誘導体
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