JP2009541415A5 - - Google Patents

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Publication number
JP2009541415A5
JP2009541415A5 JP2009517107A JP2009517107A JP2009541415A5 JP 2009541415 A5 JP2009541415 A5 JP 2009541415A5 JP 2009517107 A JP2009517107 A JP 2009517107A JP 2009517107 A JP2009517107 A JP 2009517107A JP 2009541415 A5 JP2009541415 A5 JP 2009541415A5
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JP
Japan
Prior art keywords
alkyl
cycloalkyl
tetrazol
hetero
halo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2009517107A
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English (en)
Japanese (ja)
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JP5021734B2 (ja
JP2009541415A (ja
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Priority claimed from PCT/EP2007/055997 external-priority patent/WO2008000645A1/en
Publication of JP2009541415A publication Critical patent/JP2009541415A/ja
Publication of JP2009541415A5 publication Critical patent/JP2009541415A5/ja
Application granted granted Critical
Publication of JP5021734B2 publication Critical patent/JP5021734B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009517107A 2006-06-29 2007-06-18 テトラゾール置換アリールアミド Active JP5021734B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US81729806P 2006-06-29 2006-06-29
US60/817,298 2006-06-29
PCT/EP2007/055997 WO2008000645A1 (en) 2006-06-29 2007-06-18 Tetrazole-substituted arylamides

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2012134357A Division JP5456846B2 (ja) 2006-06-29 2012-06-14 テトラゾール置換アリールアミド

Publications (3)

Publication Number Publication Date
JP2009541415A JP2009541415A (ja) 2009-11-26
JP2009541415A5 true JP2009541415A5 (https=) 2012-06-07
JP5021734B2 JP5021734B2 (ja) 2012-09-12

Family

ID=38462418

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2009517107A Active JP5021734B2 (ja) 2006-06-29 2007-06-18 テトラゾール置換アリールアミド
JP2012134357A Active JP5456846B2 (ja) 2006-06-29 2012-06-14 テトラゾール置換アリールアミド

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2012134357A Active JP5456846B2 (ja) 2006-06-29 2012-06-14 テトラゾール置換アリールアミド

Country Status (15)

Country Link
US (5) US7595405B2 (https=)
EP (2) EP2038264B1 (https=)
JP (2) JP5021734B2 (https=)
KR (1) KR101103143B1 (https=)
CN (2) CN101479250B (https=)
AR (1) AR061667A1 (https=)
AU (1) AU2007263809B2 (https=)
BR (2) BRPI0714315B8 (https=)
CA (1) CA2654915C (https=)
CL (1) CL2007001887A1 (https=)
ES (2) ES2596706T3 (https=)
IL (2) IL195786A (https=)
MX (1) MX2008016423A (https=)
TW (1) TWI334414B (https=)
WO (1) WO2008000645A1 (https=)

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AU2013273626B2 (en) * 2007-12-17 2016-04-28 F.Hoffmann-La Roche Ag Triazole-substituted arylamide derivatives and their use as P2X3 and /or P2X2/3 purinergic receptor antagonists
ES2541662T3 (es) 2007-12-17 2015-07-23 F. Hoffmann-La Roche Ag Derivados arilamida sustituidos con triazol y utilización de los mismos como antagonistas de receptores purinérgicos P2X3 y/o P2X2/3
DK2234976T3 (da) 2007-12-17 2013-06-24 Hoffmann La Roche Nye pyrazol-substituerede arylamider
CA2715835C (en) 2008-02-29 2017-03-21 Renovis, Inc. Amide compounds, compositions and uses thereof
JP5608655B2 (ja) * 2008-09-18 2014-10-15 エヴォテック アーゲー Ｐ２ｘ３受容体活性のモジュレーター
MX2011004570A (es) 2008-10-31 2011-06-17 Merck Sharp & Dohme Antagonistas del receptor p2x3 para el tratamiento del dolor.
WO2010069794A1 (en) * 2008-12-16 2010-06-24 F. Hoffmann-La Roche Ag Thiadiazole-substituted arylamides
US8569512B2 (en) 2009-03-23 2013-10-29 Merck Sharp & Dohme Corp. P2X3 receptor antagonists for treatment of pain
WO2010111059A1 (en) 2009-03-23 2010-09-30 Merck Sharp & Dohme Corp. P2x3 receptor antagonists for treatment of pain
AU2010229142A1 (en) 2009-03-23 2011-10-13 Merck Sharp & Dohme Corp. P2X3, receptor antagonists for treatment of pain
EP2246259B1 (en) 2009-04-29 2012-12-12 Eurocopter Deutschland GmbH Rotor wing with integrated tension-torque-transmission element and method for its production
CN105254557A (zh) * 2009-05-29 2016-01-20 拉夸里亚创药株式会社 作为钙或钠通道阻滞剂的芳基取代羧酰胺衍生物
TW201103904A (en) * 2009-06-11 2011-02-01 Hoffmann La Roche Janus kinase inhibitor compounds and methods
SG177308A1 (en) 2009-06-22 2012-02-28 Hoffmann La Roche Novel biphenyl and phenyl-pyridine amides
CN102438989B (zh) 2009-06-22 2015-05-27 霍夫曼-拉罗奇有限公司 噁唑酮和吡咯烷酮取代的芳基酰胺
US8476457B2 (en) 2009-06-22 2013-07-02 Roche Palo Alto Llc Indole, indazole and benzimidazole arylamides as P2X3 and P2X2/3 antagonists
WO2011153359A1 (en) * 2010-06-04 2011-12-08 Albany Molecular Research, Inc. Glycine transporter-1 inhibitors, methods of making them, and uses thereof
DK3381917T3 (da) * 2013-01-31 2021-10-18 Bellus Health Cough Inc Imidazopyridinforbindelser og anvendelser deraf
EP3230281B1 (en) 2014-12-09 2021-05-26 Bayer Aktiengesellschaft 1,3-thiazol-2-yl substituted benzamides
US10183937B2 (en) 2014-12-09 2019-01-22 Bayer Aktiengesellschaft 1,3-thiazol-2-yl substituted benzamides
WO2016169902A1 (en) * 2015-04-23 2016-10-27 F. Hoffmann-La Roche Ag Tetrazole derivatives for use in the treatment of psychiatric disorders
EP3303299B1 (en) * 2015-06-04 2019-04-24 H. Hoffnabb-La Roche Ag Imidazole derivatives
WO2017060202A1 (en) * 2015-10-06 2017-04-13 F. Hoffmann-La Roche Ag Triazole derivatives
CN108473462B (zh) 2016-02-02 2021-06-22 豪夫迈·罗氏有限公司 作为eaat3抑制剂的吡唑-吡啶衍生物
AR108222A1 (es) * 2016-05-05 2018-08-01 Elanco Tiergesundheit Ag Compuestos heteroaril-1,2,4-triazol y heteroaril-tetrazol
WO2017202896A1 (en) 2016-05-27 2017-11-30 F. Hoffmann-La Roche Ag Pyrazol compounds as eaat3 inhibitors
JP7068277B2 (ja) 2016-10-14 2022-05-16 エフ．ホフマン－ラ ロシュ アーゲー Ｅａａｔ３阻害剤としてのイミダゾール化合物
TWI741040B (zh) * 2016-10-20 2021-10-01 德商拜耳作物科學公司 製備3-烷基硫基-2-氯-n-(1-烷基-1h-四唑-5-基)-4-三氟甲基苯甲醯胺之方法
RU2650780C1 (ru) 2016-12-06 2018-04-17 Общество с ограниченной ответственностью "Анальгетики будущего" Пептидный модулятор пуринергических рецепторов
JP7797204B2 (ja) 2019-05-31 2026-01-13 キエシ・フアルマチエウテイチ・ソチエタ・ペル・アチオニ Ｐ２ｘ３阻害剤としてのピリドピリミジン誘導体
CA3139018A1 (en) 2019-05-31 2020-12-03 Chiesi Farmaceutici S.P.A. Amino quinazoline derivatives as p2x3 inhibitors
WO2022112490A1 (en) 2020-11-27 2022-06-02 Chiesi Farmaceutici S.P.A. Amino quinazoline derivatives as p2x3 inhibitors
CA3196335A1 (en) 2020-11-27 2022-06-02 Chiesi Farmaceutici S.P.A. Phthalazine derivatives as p2x3 inhibitors
JP2023550830A (ja) 2020-11-27 2023-12-05 キエシ・フアルマチエウテイチ・ソチエタ・ペル・アチオニ Ｐ２ｘ３阻害剤としての（アザ）キノリン４－アミン誘導体
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