JP2009535344A - 神経炎症性疾患の処置のためのピリダジン化合物を含む処方物 - Google Patents

神経炎症性疾患の処置のためのピリダジン化合物を含む処方物 Download PDF

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JP2009535344A
JP2009535344A JP2009507823A JP2009507823A JP2009535344A JP 2009535344 A JP2009535344 A JP 2009535344A JP 2009507823 A JP2009507823 A JP 2009507823A JP 2009507823 A JP2009507823 A JP 2009507823A JP 2009535344 A JP2009535344 A JP 2009535344A
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compound
alkyl
aryl
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JP2009535344A5 (enExample
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マーティン ワッターソン，
エルディク， リンダ バン
ウェンホイ フー，
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ノースウェスタン ユニバーシティ
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
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JP2009507823A 2006-04-28 2007-04-27 神経炎症性疾患の処置のためのピリダジン化合物を含む処方物 Pending JP2009535344A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79632806P 2006-04-28 2006-04-28
PCT/US2007/010248 WO2007127375A2 (en) 2006-04-28 2007-04-27 Formulations containing pyridazine compounds for treating neuroinflammatory diseases

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JP2009535344A true JP2009535344A (ja) 2009-10-01
JP2009535344A5 JP2009535344A5 (enExample) 2011-06-16

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US (2) US20090325973A1 (enExample)
EP (1) EP2063894B1 (enExample)
JP (1) JP2009535344A (enExample)
CN (1) CN101754762A (enExample)
AU (1) AU2007243280A1 (enExample)
BR (1) BRPI0710938A2 (enExample)
CA (1) CA2650625A1 (enExample)
IL (1) IL194968A0 (enExample)
MX (1) MX2008013843A (enExample)
WO (1) WO2007127375A2 (enExample)

Cited By (1)

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WO2006050359A2 (en) 2004-11-02 2006-05-11 Northwestern University Pyridazine compounds and methods
CA2650711A1 (en) 2006-04-28 2007-11-08 Northwestern University Compositions and treatments using pyridazine compounds and cholinesterase inhibitors
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JP5894540B2 (ja) 2010-02-18 2016-03-30 ブイティーブイ・セラピューティクス・エルエルシー フェニル−ヘテロアリール誘導体とその使用の方法
WO2011156901A2 (en) * 2010-06-17 2011-12-22 Waratah Pharmaceuticals Inc. Compounds, compositions and methods for treatment of multiple sclerosis
WO2012031383A1 (zh) 2010-09-06 2012-03-15 中国科学院广州生物医药与健康研究院 酰胺类化合物
TW202413340A (zh) 2016-07-12 2024-04-01 美商銳新醫藥公司 作為異位shp2抑制劑之2,5-雙取代型3-甲基吡嗪及2,5,6-三取代型3-甲基吡嗪
RU2019126455A (ru) 2017-01-23 2021-02-24 Революшн Медсинз, Инк. Пиридиновые соединения в качестве аллостерических ингибиторов shp2
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JP2020536881A (ja) * 2017-10-12 2020-12-17 レヴォリューション・メディスンズ，インコーポレイテッド アロステリックｓｈｐ２阻害剤としてのピリジン、ピラジンおよびトリアジン化合物
RU2020123241A (ru) 2017-12-15 2022-01-17 Революшн Медсинз, Инк. Полициклические соединения в качестве аллостерических ингибиторов shp2
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