JP2009525324A - インドール誘導体の新規なクエン酸塩およびその医薬用途 - Google Patents
インドール誘導体の新規なクエン酸塩およびその医薬用途 Download PDFInfo
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| SA07280004B1 (ar) * | 2006-02-02 | 2011-10-29 | استرازينيكا ايه بي | ملح سترات من مركب 2- هيدروكسي –3- [5- (مورفولين –4- يل ميثيل) بيريدين –2- يل] 1h- إندول –5- كربونيتريل سترات |
| WO2008130312A1 (en) * | 2007-04-18 | 2008-10-30 | Astrazeneca Ab | A new process for the manufacturing of the compound 2-hydroxy-3-[5-(morpholin-4-ylmethyl)pyridin-2-yl]1h-indole-5-carbonitrile 701 |
| US20100267720A1 (en) * | 2007-07-30 | 2010-10-21 | Astrazeneca Ab | Crystalline Forms of 2-Hydroxy-3- [5- (Morpholin- 4- Ylmethyl) Pyridin-2-YL] IH- Indole- 5 -Carbonitrile Citrate |
| US20100189788A1 (en) | 2009-01-23 | 2010-07-29 | Teva Pharmaceutical Industries, Ltd. | Delayed release rasagiline base formulation |
| EP3920885A1 (en) | 2019-02-08 | 2021-12-15 | Frequency Therapeutics, Inc. | Valproic acid compounds and wnt agonists for treating ear disorders |
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| WO2005027823A2 (en) * | 2003-09-24 | 2005-03-31 | Astrazeneca Ab | 3-heterocyclyl-indole derivatives as inhibitors of glycogen synthase kinase-3 (gsk-3) |
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| CA2439593C (en) | 2001-04-05 | 2010-02-09 | Torrent Pharmaceuticals Ltd. | Heterocyclic compounds for aging-related and diabetic vascular complications |
| JP2003009588A (ja) | 2001-06-20 | 2003-01-10 | Toshiba Corp | 車両連続運転装置用インバータ装置 |
| SE0200979D0 (sv) * | 2002-03-28 | 2002-03-28 | Astrazeneca Ab | New compounds |
| US20050054663A1 (en) * | 2003-08-13 | 2005-03-10 | Bennett Christina N. | GSK-3 inhibitors |
| TWI427077B (zh) | 2004-12-30 | 2014-02-21 | Astex Therapeutics Ltd | 吡唑化合物及其用途和含有彼之藥學組成物 |
| SA07280004B1 (ar) * | 2006-02-02 | 2011-10-29 | استرازينيكا ايه بي | ملح سترات من مركب 2- هيدروكسي –3- [5- (مورفولين –4- يل ميثيل) بيريدين –2- يل] 1h- إندول –5- كربونيتريل سترات |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2023523165A (ja) * | 2020-04-07 | 2023-06-02 | シエラ オンコロジー， インコーポレイテッド | Ｃｈｋ１阻害剤の合成方法 |
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| US20070203137A1 (en) | 2007-08-30 |
| MY146102A (en) | 2012-06-29 |
| ECSP088647A (es) | 2008-08-29 |
| IL192888A0 (en) | 2009-02-11 |
| NO20083784L (no) | 2008-10-13 |
| AU2007210336B2 (en) | 2011-03-24 |
| RU2415137C2 (ru) | 2011-03-27 |
| KR20080098022A (ko) | 2008-11-06 |
| CN101379053A (zh) | 2009-03-04 |
| ZA200806725B (en) | 2009-07-29 |
| US20090023732A1 (en) | 2009-01-22 |
| NZ570849A (en) | 2011-01-28 |
| AU2007210336A1 (en) | 2007-08-09 |
| AR059225A1 (es) | 2008-03-19 |
| SG169381A1 (en) | 2011-03-30 |
| SA07280004B1 (ar) | 2011-10-29 |
| UY30126A1 (es) | 2007-09-28 |
| UA94251C2 (ru) | 2011-04-26 |
| RU2008131906A (ru) | 2010-03-10 |
| TW200800977A (en) | 2008-01-01 |
| CA2641900A1 (en) | 2007-08-09 |
| BRPI0706745A2 (pt) | 2011-04-05 |
| EP1981869A1 (en) | 2008-10-22 |
| MX2008009719A (es) | 2008-09-04 |
| US8008294B2 (en) | 2011-08-30 |
| EP1981869A4 (en) | 2010-08-25 |
| PE20090192A1 (es) | 2009-03-20 |
| WO2007089191A1 (en) | 2007-08-09 |
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