JP2009519988A - アデノシンａ３受容体モジュレーターとしてのピロロ［１，２−ａ］キノキサリン誘導体およびその使用 - Google Patents
アデノシンａ３受容体モジュレーターとしてのピロロ［１，２−ａ］キノキサリン誘導体およびその使用 Download PDFInfo
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- JP2009519988A JP2009519988A JP2008546234A JP2008546234A JP2009519988A JP 2009519988 A JP2009519988 A JP 2009519988A JP 2008546234 A JP2008546234 A JP 2008546234A JP 2008546234 A JP2008546234 A JP 2008546234A JP 2009519988 A JP2009519988 A JP 2009519988A
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Landscapes
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| EP05292739A EP1798233A1 (en) | 2005-12-19 | 2005-12-19 | Pyrrolo[1,2-a]quinoxaline derivatives as Adenosine A3 receptor modulators and uses thereof |
| PCT/EP2006/012258 WO2007071379A1 (en) | 2005-12-19 | 2006-12-19 | PYRROLO [l,2-A]QUINOXALINE DERIVATIVES AS ADENOSINE A3 RECEPTOR MODULATORS AND USES THEREOF |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009519988A true JP2009519988A (ja) | 2009-05-21 |
| JP2009519988A5 JP2009519988A5 (enExample) | 2010-01-21 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP2008546234A Withdrawn JP2009519988A (ja) | 2005-12-19 | 2006-12-19 | アデノシンａ３受容体モジュレーターとしてのピロロ［１，２−ａ］キノキサリン誘導体およびその使用 |
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| Country | Link |
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| US (1) | US20090093476A1 (enExample) |
| EP (2) | EP1798233A1 (enExample) |
| JP (1) | JP2009519988A (enExample) |
| AU (1) | AU2006328934A1 (enExample) |
| CA (1) | CA2634165A1 (enExample) |
| WO (1) | WO2007071379A1 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2014144969A (ja) * | 2014-04-10 | 2014-08-14 | Can-Fite Biopharma Ltd | 肝細胞の増殖を誘導する方法及びその使用 |
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| GB0615809D0 (en) * | 2006-08-09 | 2006-09-20 | Istituto Di Ricerche D Biolog | Therapeutic compounds |
| CA2672860C (en) | 2006-12-28 | 2013-01-29 | Abbott Laboratories | Inhibitors of poly(adp-ribose)polymerase |
| ES2490606T3 (es) | 2007-10-15 | 2014-09-04 | Can-Fite Biopharma Ltd. | Procedimiento para inducir proliferación de hepatocitos y usos del mismo |
| WO2010014921A2 (en) | 2008-08-01 | 2010-02-04 | The United States Of America, As Represented By The Secretary, Department Of Health And Human Services | A3 adenosine receptor antagonists and partial agonists |
| EP2260038B1 (en) | 2008-03-31 | 2014-12-03 | The United States Of America, As Represented By The Secretary, Department Of Health And Human Services | Purine derivatives as a3 adenosine receptor-selective agonists |
| US8916570B2 (en) | 2008-03-31 | 2014-12-23 | The United States Of America, As Represented By The Secretary, Department Of Health And Human Services | A3 adenosine receptor agonists and antagonists |
| US9181253B2 (en) | 2008-08-01 | 2015-11-10 | The United States Of America, As Represented By The Secretary, Department Of Health And Human Services | Adenosine receptor agonists, partial agonists, and antagonists |
| WO2018005863A1 (en) | 2016-07-01 | 2018-01-04 | G1 Therapeutics, Inc. | Pyrimidine-based compounds for the treatment of cancer |
| BR112022025238A2 (pt) | 2020-06-11 | 2023-02-14 | Chdi Foundation Inc | Compostos heterocíclicos e agentes de imageamento para formar imagem da proteína huntingtina |
| CN114560862A (zh) * | 2022-03-08 | 2022-05-31 | 山东龙辰药业有限公司 | 一种吡咯并[1,2-a]喹喔啉-4(5h)-酮及其衍生物的合成方法 |
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| CA2289731A1 (en) | 1997-05-09 | 1998-11-12 | The United States Of America, Represented By The Secretary, Department O F Health And Human Services | Methods and compositions for reducing ischemic injury of the heart by administering adenosine receptor agonists and antagonists |
| JP2003517423A (ja) * | 1997-07-29 | 2003-05-27 | メドコ リサーチ、インコーポレイテッド | アデノシンレセプターモジュレーターとしてのｎ６−置換アデノシン−５′−ウロナミド |
| US6376521B1 (en) | 1998-07-10 | 2002-04-23 | The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services | A3 adenosine receptor antagonists |
| US6921825B2 (en) * | 1998-09-16 | 2005-07-26 | King Pharmaceuticuals Research & Development, Inc. | Adenosine A3 receptor modulators |
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2006
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| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2014144969A (ja) * | 2014-04-10 | 2014-08-14 | Can-Fite Biopharma Ltd | 肝細胞の増殖を誘導する方法及びその使用 |
Also Published As
| Publication number | Publication date |
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| CA2634165A1 (en) | 2007-06-28 |
| EP1973916A1 (en) | 2008-10-01 |
| US20090093476A1 (en) | 2009-04-09 |
| EP1798233A1 (en) | 2007-06-20 |
| WO2007071379A1 (en) | 2007-06-28 |
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