JP2009515893A5 - - Google Patents

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Publication number
JP2009515893A5
JP2009515893A5 JP2008540236A JP2008540236A JP2009515893A5 JP 2009515893 A5 JP2009515893 A5 JP 2009515893A5 JP 2008540236 A JP2008540236 A JP 2008540236A JP 2008540236 A JP2008540236 A JP 2008540236A JP 2009515893 A5 JP2009515893 A5 JP 2009515893A5
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JP
Japan
Prior art keywords
alkyl
halo
cycloalkyl
alkoxy
cycloalkylalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2008540236A
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English (en)
Japanese (ja)
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JP2009515893A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2006/043920 external-priority patent/WO2007070201A1/en
Publication of JP2009515893A publication Critical patent/JP2009515893A/ja
Publication of JP2009515893A5 publication Critical patent/JP2009515893A5/ja
Withdrawn legal-status Critical Current

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JP2008540236A 2005-11-14 2006-11-13 アスパラギン酸プロテアーゼ抑制剤 Withdrawn JP2009515893A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US73656405P 2005-11-14 2005-11-14
US84533106P 2006-09-18 2006-09-18
US84529106P 2006-09-18 2006-09-18
PCT/US2006/043920 WO2007070201A1 (en) 2005-11-14 2006-11-13 Aspartic protease inhibitors

Publications (2)

Publication Number Publication Date
JP2009515893A JP2009515893A (ja) 2009-04-16
JP2009515893A5 true JP2009515893A5 (enExample) 2010-07-15

Family

ID=37812974

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008540236A Withdrawn JP2009515893A (ja) 2005-11-14 2006-11-13 アスパラギン酸プロテアーゼ抑制剤

Country Status (15)

Country Link
US (1) US8487108B2 (enExample)
EP (1) EP1966139B1 (enExample)
JP (1) JP2009515893A (enExample)
KR (1) KR101379663B1 (enExample)
AR (1) AR057890A1 (enExample)
AT (1) ATE538092T1 (enExample)
AU (1) AU2006325322B2 (enExample)
BR (1) BRPI0618585A2 (enExample)
CA (1) CA2628952C (enExample)
NO (1) NO20082108L (enExample)
NZ (1) NZ568042A (enExample)
PE (2) PE20070804A1 (enExample)
SG (1) SG169983A1 (enExample)
TW (1) TWI411607B (enExample)
WO (1) WO2007070201A1 (enExample)

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BR112015003393A2 (pt) 2012-08-16 2017-07-04 Janssen Pharmaceutica Nv pirazóis substituídos como bloqueadores de canal de cálcio de tipo-n
US9453002B2 (en) 2013-08-16 2016-09-27 Janssen Pharmaceutica Nv Substituted imidazoles as N-type calcium channel blockers
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CA3173676A1 (en) * 2020-04-24 2021-10-28 Guangzhou Kangrui Biological Pharmaceutical Technology Co., Ltd. A formulation for treating ophthalmic conditions
US12083099B2 (en) 2020-10-28 2024-09-10 Accencio LLC Methods of treating symptoms of coronavirus infection with viral protease inhibitors
TW202300150A (zh) 2021-03-18 2023-01-01 美商薛定諤公司 環狀化合物及其使用方法
AR129265A1 (es) 2022-05-12 2024-08-07 Syngenta Crop Protection Ag Compuestos de alcoxi-heteroaril-carboxamida o tioamida
WO2024033374A1 (en) 2022-08-11 2024-02-15 Syngenta Crop Protection Ag Novel arylcarboxamide or arylthioamide compounds
EP4634152A1 (en) 2022-12-15 2025-10-22 Syngenta Crop Protection AG Novel bicyclic-carboxamide compounds useful as pesticides
CN116987090B (zh) * 2023-07-25 2025-06-27 乳源东阳光药业有限公司 (4aR,7aS)-6-(2,2-二乙氧基乙基)六氢-5H-[1,4]二恶烷并[2,3-c]吡咯的合成方法

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WO2007117557A2 (en) 2006-04-05 2007-10-18 Vitae Pharmaceuticals, Inc. Diaminopropanol renin inhibitors
US7858624B2 (en) 2006-04-05 2010-12-28 Vitae Pharmaceuticals, Inc. Piperidine and morpholine renin inhibitors
JP2010503682A (ja) 2006-09-18 2010-02-04 ビテ ファーマシューティカルズ， インコーポレイテッド レニン阻害剤としてのピペリジン誘導体
CL2007002689A1 (es) 2006-09-18 2008-04-18 Vitae Pharmaceuticals Inc Compuestos derivados de piperidin-1-carboxamida, inhibidores de la renina; compuestos intermediarios; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como hipertension, insuficiencia cardiaca, fibrosis cardiaca, entre otras.
US20100160424A1 (en) 2007-06-20 2010-06-24 Baldwin John J Renin inhibitors
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AR077692A1 (es) 2009-08-06 2011-09-14 Vitae Pharmaceuticals Inc Sales de 2-((r)-(3-clorofenil) ((r)-1-((s) -2-(metilamino)-3-((r)-tetrahidro-2h-piran-3-il) propilcarbamoil) piperidin -3-il) metoxi) etilcarbamato de metilo

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