JP2009501233A - バイオアベイラビリティーの高いｏ−デスメチルベンラファキシンスクシネートの経口用遅延放出投薬形態 - Google Patents
バイオアベイラビリティーの高いｏ−デスメチルベンラファキシンスクシネートの経口用遅延放出投薬形態 Download PDFInfo
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- JP2009501233A JP2009501233A JP2008521581A JP2008521581A JP2009501233A JP 2009501233 A JP2009501233 A JP 2009501233A JP 2008521581 A JP2008521581 A JP 2008521581A JP 2008521581 A JP2008521581 A JP 2008521581A JP 2009501233 A JP2009501233 A JP 2009501233A
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Images
Classifications
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- A—HUMAN NECESSITIES
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- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US69962305P | 2005-07-15 | 2005-07-15 | |
| PCT/US2006/027106 WO2007011619A2 (en) | 2005-07-15 | 2006-07-13 | Highly bioavailable oral delayed release dosage forms of o-desmethylvenlafaxine succinate |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009501233A true JP2009501233A (ja) | 2009-01-15 |
| JP2009501233A5 JP2009501233A5 (https=) | 2009-08-27 |
Family
ID=37669348
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008521581A Withdrawn JP2009501233A (ja) | 2005-07-15 | 2006-07-13 | バイオアベイラビリティーの高いｏ−デスメチルベンラファキシンスクシネートの経口用遅延放出投薬形態 |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US20070014859A1 (https=) |
| EP (1) | EP1904040A2 (https=) |
| JP (1) | JP2009501233A (https=) |
| KR (1) | KR20080025405A (https=) |
| CN (1) | CN101247791A (https=) |
| AR (1) | AR054833A1 (https=) |
| AU (1) | AU2006270315A1 (https=) |
| BR (1) | BRPI0613484A2 (https=) |
| CA (1) | CA2612960A1 (https=) |
| CR (1) | CR9626A (https=) |
| EC (1) | ECSP088106A (https=) |
| GT (1) | GT200600307A (https=) |
| IL (1) | IL188313A0 (https=) |
| MX (1) | MX2008000666A (https=) |
| NO (1) | NO20080088L (https=) |
| PE (1) | PE20070192A1 (https=) |
| RU (1) | RU2007148195A (https=) |
| SV (1) | SV2008002612A (https=) |
| TW (1) | TW200740427A (https=) |
| WO (1) | WO2007011619A2 (https=) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR101313702B1 (ko) | 2005-02-03 | 2013-10-04 | 와이어쓰 | 제피티니브 및/또는 에를로티니브 내성암 치료용 약제학적 조성물 |
| DE602006010343D1 (de) * | 2005-03-31 | 2009-12-24 | Wyeth Corp | Kombinationsprodukt aus o-desmethylvenlafaxin und bazedoxifen und verwendungen davon |
| US20080175873A1 (en) * | 2005-06-02 | 2008-07-24 | Biovail Laboratories International S.R.L. | Modified release composition of at least one form of venlafaxine |
| EP1942937A1 (en) | 2005-11-04 | 2008-07-16 | Wyeth | Antineoplastic combinations with mtor inhibitor, herceptin, and/or hki-272 |
| CA2629609A1 (en) * | 2005-12-05 | 2007-06-14 | Wyeth | Process for selective synthesis of enantiomers of substituted 1-(2-amino-1-phenyl-ethyl)-cyclohexanols |
| TW200806282A (en) * | 2006-05-05 | 2008-02-01 | Wyeth Corp | Solid dosage formulations |
| TR200909798T1 (tr) * | 2007-07-12 | 2010-05-21 | Dr. Reddy's Laboratories Ltd. | O-desmetilvenlafaksin. |
| CA2702664A1 (en) * | 2007-10-16 | 2009-04-23 | Alphapharm Pty Ltd | Controlled-release pharmaceutical formulation |
| US8022216B2 (en) | 2007-10-17 | 2011-09-20 | Wyeth Llc | Maleate salts of (E)-N-{4-[3-chloro-4-(2-pyridinylmethoxy)anilino]-3-cyano-7-ethoxy-6-quinolinyl}-4-(dimethylamino)-2-butenamide and crystalline forms thereof |
| BRPI0722303A2 (pt) * | 2007-12-10 | 2014-04-22 | Wyeth Llc | O-desmatil-venlafaxina para tratar transtorno depressivo maior |
| BRPI0914790A2 (pt) | 2008-06-17 | 2015-10-20 | Wyeth Llc | uso de um composto de vinorelbina e um composto de hki-272, composição farmacêutica e produto e kit para o tratamento de neoplasma |
| US8669273B2 (en) | 2008-08-04 | 2014-03-11 | Wyeth Llc | Antineoplastic combinations of 4-anilino-3-cyanoquinolines and capecitabine |
| CN101716168B (zh) * | 2008-10-09 | 2014-09-17 | 北京德众万全医药科技有限公司 | 一种含有去甲文拉法新的盐的药物组合物及其制备方法 |
| EP2191822A1 (en) | 2008-11-26 | 2010-06-02 | LEK Pharmaceuticals d.d. | Controlled release pharmaceutical compositions comprising O-desmethyl-venlafaxine |
| DK3000467T3 (da) | 2009-04-06 | 2023-03-27 | Wyeth Llc | Behandling med neratinib mod brystkræft |
| CA2780332C (en) | 2009-11-09 | 2018-01-30 | Wyeth Llc | Coated drug spheroids and uses thereof for eliminating or reducing conditions such as emesis and diarrhea |
| MX2012010659A (es) | 2010-03-31 | 2013-03-05 | Wockhardt Ltd | Composicion farmaceutica de liberacion modificada que comprende desvenlafaxina o sus sales. |
| CN102085197B (zh) * | 2010-12-14 | 2013-08-14 | 北京万生药业有限责任公司 | 一种文拉法辛缓释制剂及其制备方法 |
| KR20140030156A (ko) | 2011-04-12 | 2014-03-11 | 루핀 리미티드 | 방출-조절되는 데스벤라팍신 약학 조성물 |
| CN111008356B (zh) * | 2019-11-13 | 2023-06-16 | 成都理工大学 | 一种基于WTSVD算法扣除背景的γ能谱集分析方法 |
| CN114288273B (zh) * | 2022-02-11 | 2022-10-18 | 桂林华信制药有限公司 | 一种盐酸文拉法辛缓释胶囊及其生产工艺 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6274171B1 (en) * | 1996-03-25 | 2001-08-14 | American Home Products Corporation | Extended release formulation of venlafaxine hydrochloride |
| WO2000076955A1 (en) * | 1999-06-15 | 2000-12-21 | American Home Products Corporation | Enantiomers of o-desmethyl venlafaxine |
| AR021347A1 (es) * | 1999-10-20 | 2002-07-17 | Cipla Ltd | Una composicion farmaceutica que contiene acido(s) bisfosfoncio o sal(es) del mismo y un proceso de preparacion de la misma |
| US20030190352A1 (en) * | 2002-03-28 | 2003-10-09 | Synthon Bv | Compositions of venlafaxine base |
| US6703044B1 (en) * | 2002-10-25 | 2004-03-09 | Dexcel Pharma Tech, Ltd | Venlafaxine formulations |
| ES2277030T3 (es) * | 2003-05-02 | 2007-07-01 | Dexcel Ltd. | Formulacion en comprimidos de venlafaxina de liberacion prolongada. |
| AU2005212166A1 (en) * | 2004-02-06 | 2005-08-25 | Wyeth | Multiparticulate O-desmethylvenlafaxine salts and uses thereof |
| US8394409B2 (en) * | 2004-07-01 | 2013-03-12 | Intellipharmaceutics Corp. | Controlled extended drug release technology |
-
2006
- 2006-07-13 US US11/486,324 patent/US20070014859A1/en not_active Abandoned
- 2006-07-13 SV SV2006002612A patent/SV2008002612A/es unknown
- 2006-07-13 MX MX2008000666A patent/MX2008000666A/es not_active Application Discontinuation
- 2006-07-13 PE PE2006000833A patent/PE20070192A1/es not_active Application Discontinuation
- 2006-07-13 CA CA002612960A patent/CA2612960A1/en not_active Abandoned
- 2006-07-13 WO PCT/US2006/027106 patent/WO2007011619A2/en not_active Ceased
- 2006-07-13 EP EP06787061A patent/EP1904040A2/en not_active Withdrawn
- 2006-07-13 AU AU2006270315A patent/AU2006270315A1/en not_active Abandoned
- 2006-07-13 TW TW095125660A patent/TW200740427A/zh unknown
- 2006-07-13 JP JP2008521581A patent/JP2009501233A/ja not_active Withdrawn
- 2006-07-13 AR ARP060103012A patent/AR054833A1/es unknown
- 2006-07-13 CN CNA2006800258002A patent/CN101247791A/zh active Pending
- 2006-07-13 BR BRPI0613484A patent/BRPI0613484A2/pt not_active IP Right Cessation
- 2006-07-13 RU RU2007148195/15A patent/RU2007148195A/ru unknown
- 2006-07-13 KR KR1020087001067A patent/KR20080025405A/ko not_active Withdrawn
- 2006-07-13 GT GT200600307A patent/GT200600307A/es unknown
-
2007
- 2007-12-20 IL IL188313A patent/IL188313A0/en unknown
- 2007-12-20 CR CR9626A patent/CR9626A/es not_active Application Discontinuation
-
2008
- 2008-01-07 NO NO20080088A patent/NO20080088L/no not_active Application Discontinuation
- 2008-01-14 EC EC2008008106A patent/ECSP088106A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2007011619A2 (en) | 2007-01-25 |
| MX2008000666A (es) | 2008-03-13 |
| US20070014859A1 (en) | 2007-01-18 |
| SV2008002612A (es) | 2008-08-29 |
| EP1904040A2 (en) | 2008-04-02 |
| BRPI0613484A2 (pt) | 2016-11-16 |
| CR9626A (es) | 2008-04-10 |
| KR20080025405A (ko) | 2008-03-20 |
| NO20080088L (no) | 2008-04-02 |
| CA2612960A1 (en) | 2007-01-25 |
| GT200600307A (es) | 2008-04-24 |
| WO2007011619A3 (en) | 2007-06-21 |
| RU2007148195A (ru) | 2009-08-20 |
| PE20070192A1 (es) | 2007-03-16 |
| CN101247791A (zh) | 2008-08-20 |
| ECSP088106A (es) | 2008-02-20 |
| IL188313A0 (en) | 2008-04-13 |
| TW200740427A (en) | 2007-11-01 |
| AU2006270315A1 (en) | 2007-01-25 |
| AR054833A1 (es) | 2007-07-18 |
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