JP2008540618A5 - - Google Patents
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- Publication number
- JP2008540618A5 JP2008540618A5 JP2008511739A JP2008511739A JP2008540618A5 JP 2008540618 A5 JP2008540618 A5 JP 2008540618A5 JP 2008511739 A JP2008511739 A JP 2008511739A JP 2008511739 A JP2008511739 A JP 2008511739A JP 2008540618 A5 JP2008540618 A5 JP 2008540618A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- substituted
- amide
- sulfonic acid
- methylnaphthalene
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US68202005P | 2005-05-18 | 2005-05-18 | |
| FI20055235A FI20055235A0 (fi) | 2005-05-18 | 2005-05-18 | Somatostatiinireseptorialatyyppeihin 1 ja/tai 4 selektiivisesti vaikuttavat peptidienkaltaiset yhdisteet |
| PCT/FI2006/050197 WO2006123020A1 (en) | 2005-05-18 | 2006-05-16 | Peptidomimetics selective for the somatostatin receptor subtypes 1 and/or 4 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008540618A JP2008540618A (ja) | 2008-11-20 |
| JP2008540618A5 true JP2008540618A5 (https=) | 2009-07-02 |
Family
ID=37430963
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008511739A Pending JP2008540618A (ja) | 2005-05-18 | 2006-05-16 | ソマトスタチン受容体サブタイプ１及び／又は４に選択的なペプチド模倣薬 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20100048549A1 (https=) |
| EP (1) | EP1885693A4 (https=) |
| JP (1) | JP2008540618A (https=) |
| CA (1) | CA2609161A1 (https=) |
| WO (1) | WO2006123020A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103382174A (zh) | 2006-06-23 | 2013-11-06 | 雅培制药有限公司 | 作为组胺h3受体调节物的环丙胺衍生物 |
| US9108948B2 (en) | 2006-06-23 | 2015-08-18 | Abbvie Inc. | Cyclopropyl amine derivatives |
| US9186353B2 (en) | 2009-04-27 | 2015-11-17 | Abbvie Inc. | Treatment of osteoarthritis pain |
| US8853390B2 (en) | 2010-09-16 | 2014-10-07 | Abbvie Inc. | Processes for preparing 1,2-substituted cyclopropyl derivatives |
| EP3371149A4 (en) * | 2015-11-04 | 2019-03-20 | University of Florida Research Foundation, Inc. | POLYAMINE SULFONAMIDES AND USES THEREOF |
| CN114949174B (zh) * | 2022-07-19 | 2025-09-30 | 山东大学齐鲁医院 | Cst-14在制备糖尿病皮肤溃疡、破损治疗药物中的应用 |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4485101A (en) * | 1983-10-11 | 1984-11-27 | Administrators Of The Tulane Educational Fund | Peptides |
| US5409894A (en) * | 1991-03-14 | 1995-04-25 | Sandoz Ltd. | Method of preventing balloon catheterization blood vessel damage |
| JPH069402A (ja) * | 1991-05-15 | 1994-01-18 | Hiroyoshi Hidaka | 抗潰瘍剤 |
| FR2689130B1 (fr) * | 1992-03-30 | 1994-05-27 | Synthelabo | Derives de 1-[2 (arylsulfonylamino)ethyl-1-oxo] piperidine, leur preparation et leur application en therapeutique. |
| US5248673A (en) * | 1992-12-23 | 1993-09-28 | Bristol-Myers Squibb Co. | Bisamidine derivatives as thrombin inhibitors |
| KR0173034B1 (ko) * | 1995-04-28 | 1999-03-30 | 성재갑 | 선택적 트롬빈 억제제 |
| WO1997029097A1 (en) * | 1996-02-09 | 1997-08-14 | Smithkline Beecham Plc | Sulfonamide derivatives as 5ht7 receptor antagonists |
| DE69832376T2 (de) * | 1997-04-21 | 2006-08-03 | Takeda Pharmaceutical Co. Ltd. | 4,1-benzoxazepine, ihre analoga, und ihre verwendung als somatostatin-agonisten |
| GB9711043D0 (en) * | 1997-05-29 | 1997-07-23 | Ciba Geigy Ag | Organic compounds |
| US6124256A (en) * | 1998-03-27 | 2000-09-26 | Haeyry; Pekka | Method for the prevention of a patient's fibroproliferative vasculopathy |
| EP1070054A1 (en) * | 1998-04-08 | 2001-01-24 | Takeda Chemical Industries, Ltd. | Amine compounds, their production and their use as somatostatin receptor antagonists or agonists |
| FR2800735B1 (fr) * | 1999-11-09 | 2002-02-01 | Centre Nat Rech Scient | Nouvelles aralkyle-1,2-diamines possedant une activite calcimimetique et leur mode de preparation |
| GB0013060D0 (en) * | 2000-05-31 | 2000-07-19 | Astrazeneca Ab | Chemical compounds |
| JP2005535710A (ja) * | 2002-08-09 | 2005-11-24 | トランス テック ファーマ，インコーポレイテッド | アリールおよびヘテロアリール化合物ならびに凝固を調節する方法 |
| GB0314476D0 (en) * | 2003-06-20 | 2003-07-23 | Glaxo Group Ltd | Compounds |
| FI20031454A0 (fi) * | 2003-10-06 | 2003-10-06 | Juvantia Pharma Ltd Oy | Selektiivisiä somatostatiinireseptori 1 ja/tai 4 -agonisteja ja -antagonisteja |
| WO2005033068A1 (en) * | 2003-10-06 | 2005-04-14 | Oy Juvantia Pharma Ltd | Somatostatin receptor 1 and/or 4 selective agonists and antagonists |
| FI20031455A0 (fi) * | 2003-10-06 | 2003-10-06 | Juvantia Pharma Ltd Oy | Sulfonyyliamino-peptidomimeettejä, jotka ovat aktiivisia somatostatiinireseptorialatyyppien 4 (SSTR4) ja 1 (SSTR1) suhteen |
| JP4521531B2 (ja) * | 2004-07-01 | 2010-08-11 | 財団法人名古屋産業科学研究所 | 不斉アシル化触媒及び光学分割方法 |
-
2006
- 2006-05-16 US US11/919,968 patent/US20100048549A1/en not_active Abandoned
- 2006-05-16 JP JP2008511739A patent/JP2008540618A/ja active Pending
- 2006-05-16 CA CA002609161A patent/CA2609161A1/en not_active Abandoned
- 2006-05-16 WO PCT/FI2006/050197 patent/WO2006123020A1/en not_active Ceased
- 2006-05-16 EP EP06725954A patent/EP1885693A4/en not_active Withdrawn
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