JP2008540618A - ソマトスタチン受容体サブタイプ１及び／又は４に選択的なペプチド模倣薬 - Google Patents

ソマトスタチン受容体サブタイプ１及び／又は４に選択的なペプチド模倣薬 Download PDF

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JP2008540618A
JP2008540618A JP2008511739A JP2008511739A JP2008540618A JP 2008540618 A JP2008540618 A JP 2008540618A JP 2008511739 A JP2008511739 A JP 2008511739A JP 2008511739 A JP2008511739 A JP 2008511739A JP 2008540618 A JP2008540618 A JP 2008540618A
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alkyl
amide
mmol
sulfonic acid
methylnaphthalene
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JP2008540618A5 (enExample
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トンペーリ，ユッシ
サロ，ハッリ
カラトサ，オイリ
クヌーティラ，ピア
ラークソ，パイビ
ヘグルンド，イーサ
ホフレン，アンナ−マルヤ
コッコ，クルト
サーレンケト，パウリ
エングストレム，ミア
ブルスター，ジークフリート
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Publication of JP2008540618A5 publication Critical patent/JP2008540618A5/ja
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    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
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    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/10—One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline

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FI20055235A FI20055235A0 (fi) 2005-05-18 2005-05-18 Somatostatiinireseptorialatyyppeihin 1 ja/tai 4 selektiivisesti vaikuttavat peptidienkaltaiset yhdisteet
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CN101472887A (zh) 2006-06-23 2009-07-01 艾博特公司 作为组胺h3受体调节物的环丙胺衍生物
US9186353B2 (en) 2009-04-27 2015-11-17 Abbvie Inc. Treatment of osteoarthritis pain
WO2012037258A1 (en) 2010-09-16 2012-03-22 Abbott Laboratories Processes for preparing 1,2-substituted cyclopropyl derivatives
CA3001882A1 (en) 2015-11-04 2017-05-11 University Of Florida Research Foundation, Inc. Polyamine sulfonamides and uses thereof
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