JP2008534537A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2008534537A5 JP2008534537A5 JP2008503404A JP2008503404A JP2008534537A5 JP 2008534537 A5 JP2008534537 A5 JP 2008534537A5 JP 2008503404 A JP2008503404 A JP 2008503404A JP 2008503404 A JP2008503404 A JP 2008503404A JP 2008534537 A5 JP2008534537 A5 JP 2008534537A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- represents hydrogen
- hydroxy
- solvate
- salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- KVDBHTAOIKYKMP-UHFFFAOYSA-N CCC(C)(C)CC(C)(C)C(C(O)=O)N Chemical compound CCC(C)(C)CC(C)(C)C(C(O)=O)N KVDBHTAOIKYKMP-UHFFFAOYSA-N 0.000 description 1
- SUYTZMWLZYCZEF-UHFFFAOYSA-N CCC(NCCN)=O Chemical compound CCC(NCCN)=O SUYTZMWLZYCZEF-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102005014247A DE102005014247A1 (de) | 2005-03-30 | 2005-03-30 | Antibakterielle Amid-Makrozyklen VI |
| PCT/EP2006/002564 WO2006103009A1 (de) | 2005-03-30 | 2006-03-21 | Antibakterielle amid-makrozyklen vi |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008534537A JP2008534537A (ja) | 2008-08-28 |
| JP2008534537A5 true JP2008534537A5 (enExample) | 2009-04-30 |
Family
ID=36228560
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008503404A Withdrawn JP2008534537A (ja) | 2005-03-30 | 2006-03-21 | 抗菌性アミドマクロサイクルvi |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20080300231A1 (enExample) |
| EP (1) | EP1866291B1 (enExample) |
| JP (1) | JP2008534537A (enExample) |
| CA (1) | CA2602743A1 (enExample) |
| DE (2) | DE102005014247A1 (enExample) |
| ES (1) | ES2327444T3 (enExample) |
| WO (1) | WO2006103009A1 (enExample) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10358824A1 (de) | 2003-12-16 | 2005-07-21 | Bayer Healthcare Ag | Antibakterielle Makrozyklen mit substituiertem Biphenyl |
| DE102005032781A1 (de) * | 2005-07-14 | 2007-01-18 | Aicuris Gmbh & Co. Kg | Antibakterielle Amid-Markozyklen VII |
| US10501493B2 (en) | 2011-05-27 | 2019-12-10 | Rqx Pharmaceuticals, Inc. | Broad spectrum antibiotics |
| EP2922829B1 (en) * | 2012-11-21 | 2021-08-11 | RQX Pharmaceuticals, Inc. | Macrocyclic broad spectrum antibiotics |
| US10392422B2 (en) | 2014-05-20 | 2019-08-27 | Rqx Pharmaceuticals, Inc. | Macrocyclic broad spectrum antibiotics |
| RU2761476C2 (ru) | 2015-11-20 | 2021-12-08 | АрКьюИкс ФАРМАСЬЮТИКЭЛС, ИНК. | Макроциклические антибиотики широкого спектра действия |
| CN115215923A (zh) | 2019-05-28 | 2022-10-21 | 豪夫迈·罗氏有限公司 | 大环广谱抗生素 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3452136A (en) * | 1968-04-17 | 1969-06-24 | American Cyanamid Co | Antibiotic af283 and production thereof |
| FR2720066B1 (fr) * | 1994-05-20 | 1996-06-28 | Rhone Poulenc Rorer Sa | Peptides antagonistes de la neurotensine. |
| DE10226921A1 (de) * | 2002-06-17 | 2003-12-24 | Bayer Ag | Antibakterielle Amid-Makrozyklen |
| DE10234422A1 (de) * | 2002-07-29 | 2004-02-12 | Bayer Ag | Antibakterielle Ester-Makrozyklen |
| JP2008502583A (ja) * | 2003-10-01 | 2008-01-31 | バイエル・ヘルスケア・アクチェンゲゼルシャフト | 抗細菌性アミド大員環 |
| DE10358824A1 (de) * | 2003-12-16 | 2005-07-21 | Bayer Healthcare Ag | Antibakterielle Makrozyklen mit substituiertem Biphenyl |
| DE102005014240A1 (de) * | 2004-09-24 | 2006-03-30 | Bayer Healthcare Ag | Antibakterielle Amid-Makrozyklen IV |
-
2005
- 2005-03-30 DE DE102005014247A patent/DE102005014247A1/de not_active Withdrawn
-
2006
- 2006-03-21 JP JP2008503404A patent/JP2008534537A/ja not_active Withdrawn
- 2006-03-21 EP EP06723578A patent/EP1866291B1/de not_active Not-in-force
- 2006-03-21 ES ES06723578T patent/ES2327444T3/es active Active
- 2006-03-21 WO PCT/EP2006/002564 patent/WO2006103009A1/de not_active Ceased
- 2006-03-21 DE DE502006004234T patent/DE502006004234D1/de active Active
- 2006-03-21 CA CA002602743A patent/CA2602743A1/en not_active Abandoned
-
2007
- 2007-09-26 US US11/904,550 patent/US20080300231A1/en not_active Abandoned
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2007501809A5 (enExample) | ||
| JP2006182786A5 (enExample) | ||
| EP1857457A3 (en) | Benzimidazole derivative and its use as AII receptor antagonist | |
| JP2006526031A5 (enExample) | ||
| JP2009502743A5 (enExample) | ||
| JP2006518360A (ja) | イマチニブの製造方法、及び該方法により製造されたイマチニブ | |
| JP2008526999A5 (enExample) | ||
| WO2019177975A1 (en) | Antibiotics effective for gram-negative pathogens | |
| CA2637765A1 (en) | Benzamide and heteroarene derivatives | |
| MXPA04005209A (es) | Antagonistas del receptor de adenosina a2a. | |
| JP2011505356A5 (enExample) | ||
| TW200738698A (en) | Organic compounds | |
| RU2004136853A (ru) | (s)-4-амино-5-хлор-2-метокси-n-[1-[1-(2-тетрагидрофурилкарбонил)-4- пиперидини лметил]-4-пиперидинил]бензамид, способ его получения, содержащая его фармацевтическая композиция и промежуточное соединение для его получения | |
| MY145924A (en) | Antibacterial quinoline derivatives | |
| RU2409588C2 (ru) | Бактерицидные содержащие амидные группы макроциклы v | |
| JP2008534537A5 (enExample) | ||
| JP2005502636A5 (enExample) | ||
| JP2005501870A5 (enExample) | ||
| ATE366107T1 (de) | Verwendung von sulfodehydroabietinsäure zur behandlung entzündlicher darmerkrankungen | |
| JP2008534540A5 (enExample) | ||
| JP2005527479A5 (enExample) | ||
| JP2006510659A5 (enExample) | ||
| MY147404A (en) | Process for preparation of n-benzoyl-staurosporine | |
| JP2006512364A5 (enExample) | ||
| JP2008544975A5 (enExample) |