JP2008531690A - イオンチャネルリガンドとしてのアミド誘導体並びにそれを使用する医薬組成物及び方法 - Google Patents

イオンチャネルリガンドとしてのアミド誘導体並びにそれを使用する医薬組成物及び方法 Download PDF

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JP2008531690A
JP2008531690A JP2007558085A JP2007558085A JP2008531690A JP 2008531690 A JP2008531690 A JP 2008531690A JP 2007558085 A JP2007558085 A JP 2007558085A JP 2007558085 A JP2007558085 A JP 2007558085A JP 2008531690 A JP2008531690 A JP 2008531690A
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benzamide
methyl
trien
enyl
alkyl
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JP2008531690A5 (enExample
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ケルリ ミチャエル
キンカイド ジョフン
ドゥンクトン マットヘウ
サハスラブドヘ キラン
ジャナガニ サチナラハナ
ビー． ウパサニ ラビンドラ
ウ グオキアン
ファング ユンフェング
ウェイ ズヒ−リアング
カウブ カルル
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レノビス， インコーポレイテッド
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US8853392B2 (en) 2007-06-03 2014-10-07 Vanderbilt University Benzamide mGluR5 positive allosteric modulators and methods of making and using same
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FR2933977B1 (fr) * 2008-07-18 2013-04-26 Centre Nat Rech Scient Derives heterocycliques utiles dans le traitement des maladies neurodegeneratives
US20140113824A1 (en) 2011-05-10 2014-04-24 Bayer Intellectual Property Gmbh Bicyclic (thio)carbonylamidines
KR101961973B1 (ko) * 2011-09-29 2019-03-25 미쓰이가가쿠 아그로 가부시키가이샤 3,4-디히드로이소퀴놀린 유도체의 제조방법 및 그 제조중간체
KR101961972B1 (ko) * 2011-09-29 2019-03-25 미쓰이가가쿠 아그로 가부시키가이샤 4,4-디플루오로-3,4-디히드로이소퀴놀린 유도체의 제조방법
WO2013080156A1 (en) 2011-11-30 2013-06-06 Actelion Pharmaceuticals Ltd 3,7-disubstituted octahydro-2h-pyrido[4,3-e][1,3]oxazin-2-one antibiotics
WO2014113467A1 (en) * 2013-01-15 2014-07-24 Board Of Regents, The University Of Texas System Stat3 inhibitor
CN115353479A (zh) * 2022-07-27 2022-11-18 常州琦诺生物科技有限公司 一种5-溴-2-碘嘧啶的制备方法

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