JP2008524329A5 - - Google Patents

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Publication number
JP2008524329A5
JP2008524329A5 JP2007548319A JP2007548319A JP2008524329A5 JP 2008524329 A5 JP2008524329 A5 JP 2008524329A5 JP 2007548319 A JP2007548319 A JP 2007548319A JP 2007548319 A JP2007548319 A JP 2007548319A JP 2008524329 A5 JP2008524329 A5 JP 2008524329A5
Authority
JP
Japan
Prior art keywords
cancer
pharmaceutical composition
mammal
pharmaceutically acceptable
treatment
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2007548319A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008524329A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2005/045563 external-priority patent/WO2006068933A2/en
Publication of JP2008524329A publication Critical patent/JP2008524329A/ja
Publication of JP2008524329A5 publication Critical patent/JP2008524329A5/ja
Withdrawn legal-status Critical Current

Links

JP2007548319A 2004-12-21 2005-12-15 有糸分裂キネシン阻害剤 Withdrawn JP2008524329A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US63772204P 2004-12-21 2004-12-21
PCT/US2005/045563 WO2006068933A2 (en) 2004-12-21 2005-12-15 Mitotic kinesin inhibitors

Publications (2)

Publication Number Publication Date
JP2008524329A JP2008524329A (ja) 2008-07-10
JP2008524329A5 true JP2008524329A5 (enExample) 2008-12-11

Family

ID=36602225

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007548319A Withdrawn JP2008524329A (ja) 2004-12-21 2005-12-15 有糸分裂キネシン阻害剤

Country Status (7)

Country Link
US (1) US20080045492A1 (enExample)
EP (1) EP1831176A2 (enExample)
JP (1) JP2008524329A (enExample)
CN (1) CN101084194A (enExample)
AU (1) AU2005319455A1 (enExample)
CA (1) CA2589827A1 (enExample)
WO (1) WO2006068933A2 (enExample)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007011647A2 (en) * 2005-07-15 2007-01-25 Kalypsys, Inc. Inhibitors of mitotic kinesin ksp
EP1950202A1 (en) * 2007-01-24 2008-07-30 Laboratorios del Dr. Esteve S.A. Substituted pyrazoline compounds, their preparation and use as medicaments with ACAT inhibition activity
EP2114891A1 (en) * 2007-01-17 2009-11-11 Laboratorios Del. Dr. Esteve, S.A. Substituted pyrazoline compounds with acat inhibition activity
JP5455915B2 (ja) 2007-10-19 2014-03-26 メルク・シャープ・アンド・ドーム・コーポレーション Kspキネシン活性を阻害するためのスピロ縮合した1,3,4−チアジアゾール誘導体
BRPI0817897A2 (pt) * 2007-11-02 2019-09-24 Methylgene Inc composto, composição, e, métodos de inibição da atividade hdac, e de tratamento de uma doença responsiva a um inibidor de atividade hdac
US9029411B2 (en) 2008-01-25 2015-05-12 Millennium Pharmaceuticals, Inc. Thiophenes and uses thereof
US8796314B2 (en) 2009-01-30 2014-08-05 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
US9139589B2 (en) 2009-01-30 2015-09-22 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
US9090601B2 (en) 2009-01-30 2015-07-28 Millennium Pharmaceuticals, Inc. Thiazole derivatives
EP2603216A4 (en) 2010-08-11 2013-12-18 Millennium Pharm Inc HETEROARYLE AND USES THEREOF
WO2012021611A1 (en) 2010-08-11 2012-02-16 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
MA34797B1 (fr) 2010-08-11 2014-01-02 Millennium Pharm Inc Hétéroaryles et leurs utilisations
WO2012051410A2 (en) 2010-10-13 2012-04-19 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
US9226505B2 (en) 2011-09-23 2016-01-05 Bayer Intellectual Property Gmbh 4-substituted 1-phenylpyrazole-3-carboxylic acid derivatives as agents against abiotic plant stress
UY34539A (es) * 2011-12-23 2013-06-28 Millennium Pharm Inc Heteroarilos y usos de los mismos
WO2014134391A1 (en) 2013-02-28 2014-09-04 Bristol-Myers Squibb Company Phenylpyrazole derivatives as potent rock1 and rock2 inhibitors
AR094929A1 (es) 2013-02-28 2015-09-09 Bristol Myers Squibb Co Derivados de fenilpirazol como inhibidores potentes de rock1 y rock2
CN103992274A (zh) * 2014-04-18 2014-08-20 南京安美科技有限公司 合成选择性非甾体抗炎镇痛药Celebrex(塞来昔布)的方法
WO2026070814A1 (ja) * 2024-09-30 2026-04-02 大日本印刷株式会社 重合性液晶化合物及びその製造方法、重合性組成物、重合体、位相差フィルム及びその製造方法、転写用積層体、光学部材及びその製造方法、並びに表示装置

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1539727B1 (en) * 2002-07-17 2009-02-18 Cytokinetics, Inc. Compounds, compositions, and methods for treating cellular proliferative diseases
JP2008505089A (ja) * 2004-07-01 2008-02-21 メルク エンド カムパニー インコーポレーテッド 有糸分裂キネシン阻害剤
CN101155583B (zh) * 2005-04-07 2011-01-19 默沙东公司 有丝分裂驱动蛋白的抑制剂

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