JP2008524312A5 - - Google Patents
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- JP2008524312A5 JP2008524312A5 JP2007547485A JP2007547485A JP2008524312A5 JP 2008524312 A5 JP2008524312 A5 JP 2008524312A5 JP 2007547485 A JP2007547485 A JP 2007547485A JP 2007547485 A JP2007547485 A JP 2007547485A JP 2008524312 A5 JP2008524312 A5 JP 2008524312A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- results
- various embodiments
- selected number
- vitro studies
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 150000001875 compounds Chemical class 0.000 description 1
- 238000000338 in vitro Methods 0.000 description 1
Description
式（Ｉ）の種々の態様のほとんどを包含する選ばれた数の化合物に関し、試験管内研究の結果を表１０に示す。
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP04106817 | 2004-12-21 | ||
| EP05104873 | 2005-06-03 | ||
| PCT/EP2005/056951 WO2006067139A1 (en) | 2004-12-21 | 2005-12-20 | Triazolone, tetrazolone and imidazolone derivatives for use as alpha-2c adrenoreceptor antagonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008524312A JP2008524312A (ja) | 2008-07-10 |
| JP2008524312A5 true JP2008524312A5 (ja) | 2009-02-12 |
Family
ID=36013649
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007547485A Pending JP2008524312A (ja) | 2004-12-21 | 2005-12-20 | アルファ−２ｃアドレノレセプターアンタゴニストとしての使用のためのトリアゾロン、テトラゾロン及びイミダゾロン誘導体 |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20100029620A1 (ja) |
| EP (1) | EP1831185A1 (ja) |
| JP (1) | JP2008524312A (ja) |
| KR (1) | KR20070090941A (ja) |
| AR (1) | AR052342A1 (ja) |
| AU (1) | AU2005318188A1 (ja) |
| BR (1) | BRPI0516380A (ja) |
| CA (1) | CA2588028A1 (ja) |
| EA (1) | EA011514B1 (ja) |
| IL (1) | IL184048A0 (ja) |
| MX (1) | MX2007007472A (ja) |
| NO (1) | NO20073760L (ja) |
| PA (1) | PA8657301A1 (ja) |
| TW (1) | TW200635906A (ja) |
| WO (1) | WO2006067139A1 (ja) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008083124A1 (en) | 2006-12-28 | 2008-07-10 | Rigel Pharmaceuticals, Inc. | N-substituted-heterocycloalkyloxybenzamide compounds and methods of use |
| EP2566853B1 (en) | 2010-05-05 | 2017-01-25 | Infinity Pharmaceuticals, Inc. | Tetrazolones as inhibitors of fatty acid synthase |
| SG189156A1 (en) * | 2010-10-01 | 2013-05-31 | Taisho Pharmaceutical Co Ltd | 1,2,4-triazolone derivative |
| FR2976287B1 (fr) | 2011-06-09 | 2013-07-05 | Pf Medicament | Derives benzoquinolizidines, leur procede de preparation et leurs applications en therapeutique |
| KR101998442B1 (ko) * | 2011-10-27 | 2019-07-09 | 다이쇼 세이야꾸 가부시끼가이샤 | 아졸 유도체 |
| US9422252B2 (en) | 2012-05-22 | 2016-08-23 | Autifony Therapeutics Limited | Triazoles as Kv3 inhibitors |
| CA2912735A1 (en) * | 2013-06-11 | 2014-12-18 | F. Hoffmann-La Roche Ag | Novel tetrazolone derivatives |
| EP3013342B1 (en) | 2013-06-27 | 2021-04-14 | Cedars-Sinai Medical Center | Adrenoceptors antagonists for the prevention and treatment of neurodegenerative conditions |
| KR20190028763A (ko) | 2016-07-12 | 2019-03-19 | 바이엘 크롭사이언스 악티엔게젤샤프트 | 해충 방제제로서의 바이시클릭 화합물 |
| CA3079819C (en) | 2017-11-06 | 2023-03-14 | Acelot, Inc. | Small molecule drugs and related methods for treatment of diseases related to a.beta.42 oligomer formation |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3355457A (en) * | 1965-05-21 | 1967-11-28 | American Cyanamid Co | Substituted 2-imidazolinones |
| DE2725148A1 (de) * | 1977-06-03 | 1978-12-14 | Hoechst Ag | 1-aryl-4-alkyl-1,2,4-triazol-5-one und verfahren zu ihrer herstellung |
| ATE186540T1 (de) * | 1994-01-24 | 1999-11-15 | Janssen Pharmaceutica Nv | Wasserlösliche azol-antifungus |
| JPH0899975A (ja) * | 1994-08-05 | 1996-04-16 | Nippon Bayeragrochem Kk | ５員複素環置換テトラゾリノン誘導体および除草剤 |
| JPH09183770A (ja) * | 1995-10-31 | 1997-07-15 | Nippon Bayeragrochem Kk | １−アジン−テトラゾリノン類及び除草剤 |
| AU5519098A (en) * | 1996-12-13 | 1998-07-03 | E.I. Du Pont De Nemours And Company | Herbicidal heterocyclic amides |
| WO1998051683A1 (en) * | 1997-05-15 | 1998-11-19 | E.I. Du Pont De Nemours And Company | Herbicidal tetrazolinones |
| EP0957101A1 (en) * | 1998-05-14 | 1999-11-17 | Janssen Pharmaceutica N.V. | Water soluble azoles as broad-spectrum antifungals |
| AU5301799A (en) * | 1998-08-19 | 2000-03-14 | Hokko Chemical Industry Co. Ltd. | Triazolinone derivatives and herbicide compositions |
| JP3837242B2 (ja) * | 1998-08-25 | 2006-10-25 | 北興化学工業株式会社 | トリアゾリノン誘導体および除草剤 |
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2005
- 2005-12-19 AR ARP050105336A patent/AR052342A1/es not_active Application Discontinuation
- 2005-12-20 MX MX2007007472A patent/MX2007007472A/es unknown
- 2005-12-20 WO PCT/EP2005/056951 patent/WO2006067139A1/en active Application Filing
- 2005-12-20 KR KR1020077014061A patent/KR20070090941A/ko not_active Application Discontinuation
- 2005-12-20 EA EA200701345A patent/EA011514B1/ru not_active IP Right Cessation
- 2005-12-20 JP JP2007547485A patent/JP2008524312A/ja active Pending
- 2005-12-20 BR BRPI0516380-3A patent/BRPI0516380A/pt not_active IP Right Cessation
- 2005-12-20 US US11/722,380 patent/US20100029620A1/en not_active Abandoned
- 2005-12-20 PA PA20058657301A patent/PA8657301A1/es unknown
- 2005-12-20 EP EP05823472A patent/EP1831185A1/en not_active Withdrawn
- 2005-12-20 CA CA002588028A patent/CA2588028A1/en not_active Abandoned
- 2005-12-20 AU AU2005318188A patent/AU2005318188A1/en not_active Abandoned
- 2005-12-21 TW TW094145703A patent/TW200635906A/zh unknown
-
2007
- 2007-06-19 IL IL184048A patent/IL184048A0/en unknown
- 2007-07-19 NO NO20073760A patent/NO20073760L/no not_active Application Discontinuation