JP2008524312A5 - - Google Patents

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Publication number
JP2008524312A5
JP2008524312A5 JP2007547485A JP2007547485A JP2008524312A5 JP 2008524312 A5 JP2008524312 A5 JP 2008524312A5 JP 2007547485 A JP2007547485 A JP 2007547485A JP 2007547485 A JP2007547485 A JP 2007547485A JP 2008524312 A5 JP2008524312 A5 JP 2008524312A5
Authority
JP
Japan
Prior art keywords
formula
results
various embodiments
selected number
vitro studies
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2007547485A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008524312A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2005/056951 external-priority patent/WO2006067139A1/en
Publication of JP2008524312A publication Critical patent/JP2008524312A/ja
Publication of JP2008524312A5 publication Critical patent/JP2008524312A5/ja
Pending legal-status Critical Current

Links

JP2007547485A 2004-12-21 2005-12-20 アルファ−2cアドレノレセプターアンタゴニストとしての使用のためのトリアゾロン、テトラゾロン及びイミダゾロン誘導体 Pending JP2008524312A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP04106817 2004-12-21
EP05104873 2005-06-03
PCT/EP2005/056951 WO2006067139A1 (en) 2004-12-21 2005-12-20 Triazolone, tetrazolone and imidazolone derivatives for use as alpha-2c adrenoreceptor antagonists

Publications (2)

Publication Number Publication Date
JP2008524312A JP2008524312A (ja) 2008-07-10
JP2008524312A5 true JP2008524312A5 (https=) 2009-02-12

Family

ID=36013649

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007547485A Pending JP2008524312A (ja) 2004-12-21 2005-12-20 アルファ−2cアドレノレセプターアンタゴニストとしての使用のためのトリアゾロン、テトラゾロン及びイミダゾロン誘導体

Country Status (15)

Country Link
US (1) US20100029620A1 (https=)
EP (1) EP1831185A1 (https=)
JP (1) JP2008524312A (https=)
KR (1) KR20070090941A (https=)
AR (1) AR052342A1 (https=)
AU (1) AU2005318188A1 (https=)
BR (1) BRPI0516380A (https=)
CA (1) CA2588028A1 (https=)
EA (1) EA011514B1 (https=)
IL (1) IL184048A0 (https=)
MX (1) MX2007007472A (https=)
NO (1) NO20073760L (https=)
PA (1) PA8657301A1 (https=)
TW (1) TW200635906A (https=)
WO (1) WO2006067139A1 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2674237C (en) 2006-12-28 2015-11-24 Rigel Pharmaceuticals, Inc. N-substituted-heterocycloalkyloxybenzamide compounds and methods of use
EP3159331A1 (en) 2010-05-05 2017-04-26 Infinity Pharmaceuticals, Inc. Tetrazolones as inhibitors of fatty acid synthase
MX2013003633A (es) * 2010-10-01 2013-04-24 Taisho Pharmaceutical Co Ltd Derivado de 1, 2, 4-triazolona.
FR2976287B1 (fr) 2011-06-09 2013-07-05 Pf Medicament Derives benzoquinolizidines, leur procede de preparation et leurs applications en therapeutique
PL2772482T3 (pl) * 2011-10-27 2016-08-31 Taisho Pharmaceutical Co Ltd Pochodna azolu
US9422252B2 (en) 2012-05-22 2016-08-23 Autifony Therapeutics Limited Triazoles as Kv3 inhibitors
BR112015030824A2 (pt) * 2013-06-11 2017-07-25 Hoffmann La Roche novos derivados de tetrazolona
KR20160026897A (ko) 2013-06-27 2016-03-09 세다르스-신나이 메디칼 센터 신경퇴행성 질환의 예방 및 치료를 위한 아드레날린 수용체 길항제
CN109476646A (zh) 2016-07-12 2019-03-15 拜耳作物科学股份公司 作为害虫防治剂的双环化合物
CA3185336A1 (en) * 2017-11-06 2019-05-09 Acelot, Inc. Small molecule drugs and related methods for treatment of diseases related to a.beta.42 oligomer formation
JP2021183586A (ja) * 2020-05-22 2021-12-02 武田薬品工業株式会社 複素環化合物

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3355457A (en) * 1965-05-21 1967-11-28 American Cyanamid Co Substituted 2-imidazolinones
DE2725148A1 (de) * 1977-06-03 1978-12-14 Hoechst Ag 1-aryl-4-alkyl-1,2,4-triazol-5-one und verfahren zu ihrer herstellung
SG48386A1 (en) * 1994-01-24 1998-04-17 Janssen Pharmaceutica Nv Watersoluble azole antifungals
JPH0899975A (ja) * 1994-08-05 1996-04-16 Nippon Bayeragrochem Kk 5員複素環置換テトラゾリノン誘導体および除草剤
JPH09183770A (ja) * 1995-10-31 1997-07-15 Nippon Bayeragrochem Kk 1−アジン−テトラゾリノン類及び除草剤
WO1998025912A1 (en) * 1996-12-13 1998-06-18 E.I. Du Pont De Nemours And Company Herbicidal heterocyclic amides
WO1998051683A1 (en) * 1997-05-15 1998-11-19 E.I. Du Pont De Nemours And Company Herbicidal tetrazolinones
EP0957101A1 (en) * 1998-05-14 1999-11-17 Janssen Pharmaceutica N.V. Water soluble azoles as broad-spectrum antifungals
JP3837242B2 (ja) * 1998-08-25 2006-10-25 北興化学工業株式会社 トリアゾリノン誘導体および除草剤
WO2000010984A1 (en) * 1998-08-19 2000-03-02 Hokko Chemical Industry Co., Ltd. Triazolinone derivatives and herbicide compositions

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