JP2008511585A - 食事と共にするａｐｉ投与時に遅延効果を果たす経口投与調剤 - Google Patents
食事と共にするａｐｉ投与時に遅延効果を果たす経口投与調剤 Download PDFInfo
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- JP2008511585A JP2008511585A JP2007528874A JP2007528874A JP2008511585A JP 2008511585 A JP2008511585 A JP 2008511585A JP 2007528874 A JP2007528874 A JP 2007528874A JP 2007528874 A JP2007528874 A JP 2007528874A JP 2008511585 A JP2008511585 A JP 2008511585A
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- api
- forming agent
- gas forming
- delayed
- carbonate
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- DKYWVDODHFEZIM-UHFFFAOYSA-N ketoprofen Chemical compound OC(=O)C(C)C1=CC=CC(C(=O)C=2C=CC=CC=2)=C1 DKYWVDODHFEZIM-UHFFFAOYSA-N 0.000 description 1
- 229960000991 ketoprofen Drugs 0.000 description 1
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- MJIHNNLFOKEZEW-UHFFFAOYSA-N lansoprazole Chemical compound CC1=C(OCC(F)(F)F)C=CN=C1CS(=O)C1=NC2=CC=CC=C2N1 MJIHNNLFOKEZEW-UHFFFAOYSA-N 0.000 description 1
- 229960004502 levodopa Drugs 0.000 description 1
- 229960003376 levofloxacin Drugs 0.000 description 1
- 229950008325 levothyroxine Drugs 0.000 description 1
- 239000007788 liquid Substances 0.000 description 1
- 210000004185 liver Anatomy 0.000 description 1
- 239000000463 material Substances 0.000 description 1
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- 238000002483 medication Methods 0.000 description 1
- XZWYZXLIPXDOLR-UHFFFAOYSA-N metformin Chemical compound CN(C)C(=N)NC(N)=N XZWYZXLIPXDOLR-UHFFFAOYSA-N 0.000 description 1
- 229960003105 metformin Drugs 0.000 description 1
- 229960002237 metoprolol Drugs 0.000 description 1
- IUBSYMUCCVWXPE-UHFFFAOYSA-N metoprolol Chemical compound COCCC1=CC=C(OCC(O)CNC(C)C)C=C1 IUBSYMUCCVWXPE-UHFFFAOYSA-N 0.000 description 1
- 239000011859 microparticle Substances 0.000 description 1
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- 235000001968 nicotinic acid Nutrition 0.000 description 1
- 239000011664 nicotinic acid Substances 0.000 description 1
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- 229960005425 nitrendipine Drugs 0.000 description 1
- 229960001180 norfloxacin Drugs 0.000 description 1
- OGJPXUAPXNRGGI-UHFFFAOYSA-N norfloxacin Chemical compound C1=C2N(CC)C=C(C(O)=O)C(=O)C2=CC(F)=C1N1CCNCC1 OGJPXUAPXNRGGI-UHFFFAOYSA-N 0.000 description 1
- 229960001699 ofloxacin Drugs 0.000 description 1
- 239000008184 oral solid dosage form Substances 0.000 description 1
- 239000007935 oral tablet Substances 0.000 description 1
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- 229960005434 oxybutynin Drugs 0.000 description 1
- 229960002085 oxycodone Drugs 0.000 description 1
- 229960005019 pantoprazole Drugs 0.000 description 1
- 229960004321 pentaerithrityl tetranitrate Drugs 0.000 description 1
- 239000000825 pharmaceutical preparation Substances 0.000 description 1
- 229960002036 phenytoin Drugs 0.000 description 1
- 108090000623 proteins and genes Proteins 0.000 description 1
- 102000004169 proteins and genes Human genes 0.000 description 1
- 150000007660 quinolones Chemical class 0.000 description 1
- 230000000979 retarding effect Effects 0.000 description 1
- 239000000126 substance Substances 0.000 description 1
- 239000005720 sucrose Substances 0.000 description 1
- 239000000725 suspension Substances 0.000 description 1
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- 235000002906 tartaric acid Nutrition 0.000 description 1
- XUIIKFGFIJCVMT-UHFFFAOYSA-N thyroxine-binding globulin Natural products IC1=CC(CC([NH3+])C([O-])=O)=CC(I)=C1OC1=CC(I)=C(O)C(I)=C1 XUIIKFGFIJCVMT-UHFFFAOYSA-N 0.000 description 1
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- TVYLLZQTGLZFBW-GOEBONIOSA-N tramadol Natural products COC1=CC=CC([C@@]2(O)[C@@H](CCCC2)CN(C)C)=C1 TVYLLZQTGLZFBW-GOEBONIOSA-N 0.000 description 1
- 229960000604 valproic acid Drugs 0.000 description 1
Images
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/485—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004042139A DE102004042139B4 (de) | 2004-08-31 | 2004-08-31 | Perorale Darreichungsformen zur Erzielung eines Retardierungseffektes nach der Arzneimitteleinnahme mit einer Mahlzeit |
| PCT/EP2005/054260 WO2006024638A2 (de) | 2004-08-31 | 2005-08-30 | Perorale darreichungsformen zur erzielung eines retardierungseffektes nach der arzneimitteleinnahme mit einer mahlzeit |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008511585A true JP2008511585A (ja) | 2008-04-17 |
| JP2008511585A5 JP2008511585A5 (enExample) | 2008-10-09 |
Family
ID=35745691
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007528874A Pending JP2008511585A (ja) | 2004-08-31 | 2005-08-30 | 食事と共にするａｐｉ投与時に遅延効果を果たす経口投与調剤 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20090010906A1 (enExample) |
| EP (1) | EP1814512A2 (enExample) |
| JP (1) | JP2008511585A (enExample) |
| DE (1) | DE102004042139B4 (enExample) |
| EA (1) | EA013429B1 (enExample) |
| UA (1) | UA94031C2 (enExample) |
| WO (1) | WO2006024638A2 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102007041588A1 (de) | 2007-09-01 | 2009-03-05 | Lts Lohmann Therapie-Systeme Ag | Arzneimittel mit Hefe |
| CN103142552A (zh) * | 2013-02-22 | 2013-06-12 | 广州科的信医药技术有限公司 | 一种洛伐他汀肠溶缓释微丸胶囊及其制备方法 |
Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS61286322A (ja) * | 1985-06-12 | 1986-12-16 | Teijin Ltd | 経口徐放性製剤 |
| JPS62207209A (ja) * | 1986-03-07 | 1987-09-11 | Teijin Ltd | 経口徐放性製剤 |
| WO2003011255A1 (en) * | 2001-07-04 | 2003-02-13 | Sun Pharmaceutical Industries Limited | Gastric retention controlled drug delivery system |
| JP2003531161A (ja) * | 2000-04-20 | 2003-10-21 | エティファーム | 発泡性顆粒剤およびその調製法 |
| JP2004521955A (ja) * | 2001-07-09 | 2004-07-22 | キュレーターズ・オブ・ザ・ユニバーシティ・オブ・ミズーリ | 新規置換ベンズイミダゾール製剤およびその使用方法 |
Family Cites Families (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1139991A (en) * | 1965-07-19 | 1969-01-15 | Armour Pharma | Stabilized enzyme composition |
| GB1573487A (en) * | 1977-05-23 | 1980-08-28 | Bristol Myers Co | Bile acid binding composition |
| CA1182049A (en) * | 1981-07-13 | 1985-02-05 | Francis J. Sterbenz | Apap antacid composition |
| DE3681348D1 (de) * | 1985-06-11 | 1991-10-17 | Teijin Ltd | Oral-arzneizubereitung mit retardwirkung. |
| DE3543999A1 (de) * | 1985-12-13 | 1987-06-19 | Bayer Ag | Hochreine acarbose |
| JPS62195323A (ja) * | 1986-02-24 | 1987-08-28 | Eisai Co Ltd | 胃内滞留型粒子 |
| US4929605A (en) * | 1987-10-07 | 1990-05-29 | Merrell Dow Pharmaceuticals Inc. | Pharmaceutical composition for piperidinoalkanol derivatives |
| US5096714A (en) * | 1988-06-28 | 1992-03-17 | Hauser-Kuhrts, Inc. | Prolonged release drug tablet formulations |
| US5004651A (en) * | 1989-01-24 | 1991-04-02 | Abbott Laboratories | Stabilizing system for solid dosage forms |
| US4975281A (en) * | 1989-01-30 | 1990-12-04 | E. R. Squibb & Sons, Inc. | Anti-ulcer composition |
| CA2030449A1 (en) * | 1989-11-22 | 1991-05-23 | Eric H. Kuhrts | Prolonged release drug tablet formulations |
| US5683719A (en) * | 1990-11-22 | 1997-11-04 | British Technology Group Limited | Controlled release compositions |
| GB9025372D0 (en) * | 1990-11-22 | 1991-01-09 | Nat Res Dev | Pharmaceutical dosage forms |
| UA37214C2 (uk) * | 1991-01-30 | 2001-05-15 | Дзе Веллкам Фаундейшн Лімітед | Таблетки, що диспергуються у воді, та спосіб їх виготовлення |
| YU48263B (sh) * | 1991-06-17 | 1997-09-30 | Byk Gulden Lomberg Chemische Fabrik Gmbh. | Postupak za dobijanje farmaceutskog preparata na bazi pantoprazola |
| HU9203780D0 (en) * | 1991-12-12 | 1993-03-29 | Sandoz Ag | Stabilized pharmaceutical products of hmg-coa reductase inhibitor and method for producing them |
| GB9224021D0 (en) * | 1992-11-16 | 1993-01-06 | Boots Co Plc | Effervescent compositions |
| US6071539A (en) * | 1996-09-20 | 2000-06-06 | Ethypharm, Sa | Effervescent granules and methods for their preparation |
| GB9704524D0 (en) * | 1997-03-05 | 1997-04-23 | Smithkline Beecham Plc | Composition |
| US20010046473A1 (en) * | 1997-04-18 | 2001-11-29 | Jerome Besse | Gastric-retained pharmaceutical composition and method for its use |
| US6235311B1 (en) * | 1998-03-18 | 2001-05-22 | Bristol-Myers Squibb Company | Pharmaceutical composition containing a combination of a statin and aspirin and method |
| DK0976395T3 (da) * | 1998-07-30 | 2005-11-14 | Merck Sante Sas | Tablet til langvarig afgivelse af et lægemiddel i maven |
| AP1659A (en) * | 1998-09-14 | 2006-09-06 | Ranbaxy Laboratories Ltd | Orally administered controlled drug delivery system providing temporal and spatial control. |
| AP2002002410A0 (en) * | 1999-08-04 | 2002-03-31 | Ranbaxy Laboratories Ltd | Hydrodynamically Balancing Oral Drug Delivery System |
| WO2003097018A1 (en) * | 2002-02-04 | 2003-11-27 | Ranbaxy Laboratories Limited | Hydrodynamically balancing oral drug delivery system with biphasic release |
| GB0114069D0 (en) * | 2001-06-08 | 2001-08-01 | Smithkline Beecham Plc | Composition |
-
2004
- 2004-08-31 DE DE102004042139A patent/DE102004042139B4/de not_active Expired - Fee Related
-
2005
- 2005-08-30 EP EP05775898A patent/EP1814512A2/de not_active Withdrawn
- 2005-08-30 EA EA200700524A patent/EA013429B1/ru not_active IP Right Cessation
- 2005-08-30 JP JP2007528874A patent/JP2008511585A/ja active Pending
- 2005-08-30 UA UAA200703512A patent/UA94031C2/ru unknown
- 2005-08-30 WO PCT/EP2005/054260 patent/WO2006024638A2/de not_active Ceased
- 2005-08-30 US US11/574,317 patent/US20090010906A1/en not_active Abandoned
Patent Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS61286322A (ja) * | 1985-06-12 | 1986-12-16 | Teijin Ltd | 経口徐放性製剤 |
| JPS62207209A (ja) * | 1986-03-07 | 1987-09-11 | Teijin Ltd | 経口徐放性製剤 |
| JP2003531161A (ja) * | 2000-04-20 | 2003-10-21 | エティファーム | 発泡性顆粒剤およびその調製法 |
| WO2003011255A1 (en) * | 2001-07-04 | 2003-02-13 | Sun Pharmaceutical Industries Limited | Gastric retention controlled drug delivery system |
| JP2004521955A (ja) * | 2001-07-09 | 2004-07-22 | キュレーターズ・オブ・ザ・ユニバーシティ・オブ・ミズーリ | 新規置換ベンズイミダゾール製剤およびその使用方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| EA013429B1 (ru) | 2010-04-30 |
| UA94031C2 (ru) | 2011-04-11 |
| DE102004042139B4 (de) | 2009-06-10 |
| US20090010906A1 (en) | 2009-01-08 |
| EA200700524A1 (ru) | 2007-08-31 |
| WO2006024638A3 (de) | 2007-04-05 |
| WO2006024638A2 (de) | 2006-03-09 |
| DE102004042139A1 (de) | 2006-03-02 |
| EP1814512A2 (de) | 2007-08-08 |
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