JP2008509143A5

JP2008509143A5 -

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Publication number: JP2008509143A5
Authority: JP; Japan
Prior art keywords: medicament; dispersion; pressure gas; medicament according; disease
Prior art date: 2005-08-03
Legal status : Pending

Application number

JP2007524916A

Other languages

English (en)

Japanese (ja)

Other versions

JP2008509143A (ja

Filing date

2005-08-03

Publication date

2008-09-25

2005-08-03 Application filed filed Critical

2005-08-03 Priority claimed from PCT/US2005/027428 external-priority patent/WO2006017505A2/en

2008-03-27 Publication of JP2008509143A publication Critical patent/JP2008509143A/ja

2008-09-25 Publication of JP2008509143A5 publication Critical patent/JP2008509143A5/ja

Status Pending legal-status Critical Current

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239000003814 drug Substances 0.000 claims description 67
239000000203 mixture Substances 0.000 claims description 65
KQOXLKOJHVFTRN-UHFFFAOYSA-N pleconaril Chemical compound O1N=C(C)C=C1CCCOC1=C(C)C=C(C=2N=C(ON=2)C(F)(F)F)C=C1C KQOXLKOJHVFTRN-UHFFFAOYSA-N 0.000 claims description 56
229960000471 pleconaril Drugs 0.000 claims description 52
208000023504 respiratory system disease Diseases 0.000 claims description 34
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 claims description 30
150000003839 salts Chemical class 0.000 claims description 26
201000010099 disease Diseases 0.000 claims description 25
239000007789 gas Substances 0.000 claims description 19
230000003612 virological effect Effects 0.000 claims description 18
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239000006185 dispersion Substances 0.000 claims description 17
239000002552 dosage form Substances 0.000 claims description 16
208000027866 inflammatory disease Diseases 0.000 claims description 16
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WOFMFGQZHJDGCX-ZULDAHANSA-N mometasone furoate Chemical compound O([C@]1([C@@]2(C)C[C@H](O)[C@]3(Cl)[C@@]4(C)C=CC(=O)C=C4CC[C@H]3[C@@H]2C[C@H]1C)C(=O)CCl)C(=O)C1=CC=CO1 WOFMFGQZHJDGCX-ZULDAHANSA-N 0.000 claims description 9
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VSWPGAIWKHPTKX-UHFFFAOYSA-N 1-methyl-10-[2-(4-methyl-1-piperazinyl)-1-oxoethyl]-5H-thieno[3,4-b][1,5]benzodiazepin-4-one Chemical compound C1CN(C)CCN1CC(=O)N1C2=CC=CC=C2NC(=O)C2=CSC(C)=C21 VSWPGAIWKHPTKX-UHFFFAOYSA-N 0.000 claims description 2
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OEXHQOGQTVQTAT-JRNQLAHRSA-N ipratropium Chemical compound O([C@H]1C[C@H]2CC[C@@H](C1)[N@@+]2(C)C(C)C)C(=O)C(CO)C1=CC=CC=C1 OEXHQOGQTVQTAT-JRNQLAHRSA-N 0.000 claims description 2
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JP2007524916A 2004-08-04 2005-08-03 気道疾患の処置のためのプレコナリルを含む薬学的処方物 Pending JP2008509143A (ja)