JP2008503447A5 - - Google Patents

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Publication number
JP2008503447A5
JP2008503447A5 JP2007513845A JP2007513845A JP2008503447A5 JP 2008503447 A5 JP2008503447 A5 JP 2008503447A5 JP 2007513845 A JP2007513845 A JP 2007513845A JP 2007513845 A JP2007513845 A JP 2007513845A JP 2008503447 A5 JP2008503447 A5 JP 2008503447A5
Authority
JP
Japan
Prior art keywords
phenyl
disease
thiazol
acetic acid
fluoro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2007513845A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008503447A (ja
Filing date
Publication date
Priority claimed from GB0412198A external-priority patent/GB0412198D0/en
Priority claimed from GB0414194A external-priority patent/GB0414194D0/en
Priority claimed from GB0424016A external-priority patent/GB0424016D0/en
Application filed filed Critical
Priority claimed from PCT/EP2005/005882 external-priority patent/WO2005116001A1/en
Publication of JP2008503447A publication Critical patent/JP2008503447A/ja
Publication of JP2008503447A5 publication Critical patent/JP2008503447A5/ja
Withdrawn legal-status Critical Current

Links

JP2007513845A 2004-05-29 2005-05-30 Crth2リガンドとしての置換チアゾール酢酸 Withdrawn JP2008503447A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0412198A GB0412198D0 (en) 2004-05-29 2004-05-29 Medicinal use of receptor ligands
GB0414194A GB0414194D0 (en) 2004-06-24 2004-06-24 Medicinal use of receptor ligands
GB0424016A GB0424016D0 (en) 2004-10-29 2004-10-29 Medicinal use of receptor ligands
PCT/EP2005/005882 WO2005116001A1 (en) 2004-05-29 2005-05-30 Substituted thiazoleacetic as crth2 ligands

Publications (2)

Publication Number Publication Date
JP2008503447A JP2008503447A (ja) 2008-02-07
JP2008503447A5 true JP2008503447A5 (enExample) 2008-07-24

Family

ID=34968996

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007513845A Withdrawn JP2008503447A (ja) 2004-05-29 2005-05-30 Crth2リガンドとしての置換チアゾール酢酸

Country Status (13)

Country Link
US (1) US20080119456A1 (enExample)
EP (1) EP1758874A1 (enExample)
JP (1) JP2008503447A (enExample)
KR (1) KR20070044404A (enExample)
AU (1) AU2005247610A1 (enExample)
BR (1) BRPI0511671A (enExample)
CA (1) CA2568742A1 (enExample)
CR (1) CR8837A (enExample)
EA (1) EA200602288A1 (enExample)
IL (1) IL179693A0 (enExample)
MX (1) MXPA06013924A (enExample)
NO (1) NO20066049L (enExample)
WO (1) WO2005116001A1 (enExample)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0427381D0 (en) * 2004-12-14 2005-01-19 Novartis Ag Organic compounds
UY30892A1 (es) * 2007-02-07 2008-09-02 Smithkline Beckman Corp Inhibidores de la actividad akt
US8268872B2 (en) 2008-02-22 2012-09-18 Radius Health, Inc. Selective androgen receptor modulators
BRPI0907844B8 (pt) 2008-02-22 2021-05-25 Radius Health Inc compostos e método para modular um receptor de andrógeno, processos de preparação e composição farmacêutica dos mesmos e seus usos
JP5535931B2 (ja) 2008-10-27 2014-07-02 武田薬品工業株式会社 二環性化合物
WO2010088331A1 (en) * 2009-01-30 2010-08-05 Glaxosmithkline Llc Crystalline n-{(1-s)-2-amino-1-[(3-fluorophenyl)methyl]ethyl}-5-chloro-4-(4-chloro-1-methyl-1h-pyrazol-5-yl)-2-thiophenecarboxamide hydrochloride
EP2516416A1 (en) 2009-12-23 2012-10-31 Ironwood Pharmaceuticals, Inc. Crth2 modulators
AU2011212813B2 (en) 2010-02-04 2014-10-23 Radius Health, Inc. Selective androgen receptor modulators
SI2568806T1 (sl) 2010-05-12 2016-09-30 Radius Health, Inc. Režimi zdravljenja
US8642632B2 (en) 2010-07-02 2014-02-04 Radius Health, Inc. Selective androgen receptor modulators
EP2621901B1 (en) 2010-09-28 2015-07-29 Radius Health, Inc Selective androgen receptor modulators
EP2457900A1 (en) 2010-11-25 2012-05-30 Almirall, S.A. New pyrazole derivatives having CRTh2 antagonistic behaviour
CA2859284A1 (en) 2011-12-16 2013-06-20 Atopix Therapeutics Limited Combination of a crth2 antagonist and a proton pump inhibitor for the treatment of eosinophilic esophagitis
RS63311B1 (sr) 2016-06-22 2022-07-29 Ellipses Pharma Ltd Ar+ metode lečenja raka dojke

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ID24390A (id) * 1997-07-10 2000-07-13 Janssen Pharmaceutica Nv Turunan-turunan 6-azaurasil penghambat il-5
HUP0004238A3 (en) * 1997-11-28 2001-07-30 Lg Chemical Ltd Imidazole derivatives having an inhibitory activity for farnesyl transferase, process for preparation thereof and pharmaceutical compositions containing them
EP0987265A1 (en) * 1998-09-18 2000-03-22 Janssen Pharmaceutica N.V. Interleukin-5 inhibiting 6-azauracil derivatives
EE200200057A (et) * 1999-08-06 2003-04-15 Janssen Pharmaceutica N.V. Kasvutegurit IL-5 pärssiv asauratsiilderivaat, selle saamine ja kasutamine ravimi valmistamiseks ning seda sisaldav farmatseutiline kompositsioon
US7276526B2 (en) * 2001-07-13 2007-10-02 Bristol-Myers Squibb Pharma Company Substituted thiazoles and oxazoles as corticotropin releasing hormone ligands
TW200307542A (en) * 2002-05-30 2003-12-16 Astrazeneca Ab Novel compounds

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