JP2007524645A5 - - Google Patents
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- Publication number
- JP2007524645A5 JP2007524645A5 JP2006520347A JP2006520347A JP2007524645A5 JP 2007524645 A5 JP2007524645 A5 JP 2007524645A5 JP 2006520347 A JP2006520347 A JP 2006520347A JP 2006520347 A JP2006520347 A JP 2006520347A JP 2007524645 A5 JP2007524645 A5 JP 2007524645A5
- Authority
- JP
- Japan
- Prior art keywords
- bnoh
- meoh
- ratio
- octreotide
- pamoic acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- OKKJLVBELUTLKV-UHFFFAOYSA-N Methanol Chemical compound OC OKKJLVBELUTLKV-UHFFFAOYSA-N 0.000 description 12
- WVDDGKGOMKODPV-UHFFFAOYSA-N Benzyl alcohol Chemical compound OCC1=CC=CC=C1 WVDDGKGOMKODPV-UHFFFAOYSA-N 0.000 description 5
- 239000006184 cosolvent Substances 0.000 description 4
- DEQANNDTNATYII-OULOTJBUSA-N (4r,7s,10s,13r,16s,19r)-10-(4-aminobutyl)-19-[[(2r)-2-amino-3-phenylpropanoyl]amino]-16-benzyl-n-[(2r,3r)-1,3-dihydroxybutan-2-yl]-7-[(1r)-1-hydroxyethyl]-13-(1h-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxa Chemical compound C([C@@H](N)C(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CC=2C3=CC=CC=C3NC=2)NC(=O)[C@H](CC=2C=CC=CC=2)NC1=O)C(=O)N[C@H](CO)[C@H](O)C)C1=CC=CC=C1 DEQANNDTNATYII-OULOTJBUSA-N 0.000 description 3
- 108010016076 Octreotide Proteins 0.000 description 3
- 239000008346 aqueous phase Substances 0.000 description 3
- 238000009472 formulation Methods 0.000 description 3
- 239000000203 mixture Substances 0.000 description 3
- 229960002700 octreotide Drugs 0.000 description 3
- 239000012074 organic phase Substances 0.000 description 3
- WLJNZVDCPSBLRP-UHFFFAOYSA-N pamoic acid Chemical compound C1=CC=C2C(CC=3C4=CC=CC=C4C=C(C=3O)C(=O)O)=C(O)C(C(O)=O)=CC2=C1 WLJNZVDCPSBLRP-UHFFFAOYSA-N 0.000 description 3
- 238000005538 encapsulation Methods 0.000 description 2
- 150000002500 ions Chemical class 0.000 description 1
- 238000000710 polymer precipitation Methods 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US48766303P | 2003-07-15 | 2003-07-15 | |
| US60/487,663 | 2003-07-15 | ||
| PCT/US2004/022816 WO2005009356A2 (en) | 2003-07-15 | 2004-07-15 | Method for the preparation of controlled release formulations |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011100206A Division JP2011144207A (ja) | 2003-07-15 | 2011-04-27 | 制御放出処方物の調製のための方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2007524645A JP2007524645A (ja) | 2007-08-30 |
| JP2007524645A5 true JP2007524645A5 (https=) | 2012-07-19 |
| JP5165239B2 JP5165239B2 (ja) | 2013-03-21 |
Family
ID=34102710
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006520347A Expired - Fee Related JP5165239B2 (ja) | 2003-07-15 | 2004-07-15 | 制御放出処方物の調製のための方法 |
| JP2011100206A Pending JP2011144207A (ja) | 2003-07-15 | 2011-04-27 | 制御放出処方物の調製のための方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011100206A Pending JP2011144207A (ja) | 2003-07-15 | 2011-04-27 | 制御放出処方物の調製のための方法 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US8871269B2 (https=) |
| EP (2) | EP1651136B1 (https=) |
| JP (2) | JP5165239B2 (https=) |
| CN (2) | CN1852687B (https=) |
| AU (1) | AU2004259208B2 (https=) |
| BR (1) | BRPI0412059A (https=) |
| CA (1) | CA2532302C (https=) |
| ES (1) | ES2625343T3 (https=) |
| WO (1) | WO2005009356A2 (https=) |
Families Citing this family (37)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20070207211A1 (en) * | 2003-04-10 | 2007-09-06 | Pr Pharmaceuticals, Inc. | Emulsion-based microparticles and methods for the production thereof |
| EP2548550A1 (en) | 2003-04-10 | 2013-01-23 | Surmodics Pharmaceuticals, Inc. | Emulsion-based micro particles |
| JP5165239B2 (ja) | 2003-07-15 | 2013-03-21 | ピーアール ファーマシューティカルズ， インコーポレイテッド | 制御放出処方物の調製のための方法 |
| WO2005007122A2 (en) * | 2003-07-18 | 2005-01-27 | Oakwood Laboratories, L.L.C. | Polymer stabilization |
| WO2005009357A2 (en) | 2003-07-23 | 2005-02-03 | Pr Pharmaceuticals, Inc. | Controlled release compositions |
| JP2007517042A (ja) * | 2003-12-30 | 2007-06-28 | デュレクト コーポレーション | 活性物質、好ましくはｇｎｒｈの制御放出のための、好ましくはｐｅｇおよびｐｌｇの混合物を含有するポリマーインプラント |
| EP1679065A1 (en) * | 2005-01-07 | 2006-07-12 | OctoPlus Sciences B.V. | Controlled release compositions for interferon based on PEGT/PBT block copolymers |
| US20100290982A1 (en) * | 2007-04-13 | 2010-11-18 | University Of North Texas Health Science Center At Fort Worth | Solid in oil/water emulsion-diffusion-evaporation formulation for preparing curcumin-loaded plga nanoparticles |
| BRPI0810899A2 (pt) * | 2007-04-13 | 2014-10-29 | Univ North Texas | Formulação de nanopartículas de plga ativadas carregadas com agente ativo para substâncias nano-terapêuticas anticâncer direcionais. |
| NZ580700A (en) * | 2007-04-19 | 2012-01-12 | Dong A Pharm Co Ltd | A biodegradable microsphere composition suitable for the controlled release of glucose controlling peptide and formulation thereof |
| GB0709322D0 (en) * | 2007-05-15 | 2007-06-20 | Nordic Bioscience As | Exposure agent for detection of vitamin d |
| WO2008145183A1 (en) * | 2007-05-30 | 2008-12-04 | Nestec S.A. | Oil-in-water emulsion and its use for the delayed release of active elements |
| ES2667945T3 (es) | 2007-10-08 | 2018-05-16 | Aurinia Pharmaceuticals Inc. | Composiciones oftálmicas que comprenden inhibidores de calcineurina o Inhibidores de mTOR |
| ES2324009B1 (es) * | 2007-11-23 | 2010-05-21 | Gp Pharm S.A. | Composicion farmaceutica de liberacion sostenida de somatostatina o un analogo suyo. |
| US8071914B2 (en) * | 2007-12-26 | 2011-12-06 | Noboru Oshima | Heating apparatus |
| JP5222550B2 (ja) * | 2007-12-27 | 2013-06-26 | 財團法人工業技術研究院 | 徐放性組成物およびその製造方法 |
| US9161943B2 (en) * | 2007-12-31 | 2015-10-20 | Industrial Technology Research Institute | Sustained release composition and manufacturing method thereof |
| WO2009100222A1 (en) * | 2008-02-08 | 2009-08-13 | Qps Llc | Non-polymeric compositions for controlled drug delivery |
| CA2730760A1 (en) | 2008-07-16 | 2010-01-21 | Surmodics Pharmaceuticals, Inc. | Process for preparing microparticles containing bioactive peptides |
| EP2440185B1 (en) | 2009-06-09 | 2015-04-08 | Aurinia Pharmaceuticals Inc. | Topical drug delivery systems for ophthalmic use |
| JP2013501033A (ja) * | 2009-08-05 | 2013-01-10 | ピエリス アーゲー | リポカリン突然変異タンパク質の制御放出製剤 |
| US20110151028A1 (en) * | 2009-12-19 | 2011-06-23 | Filiberto Zadini | Topical vaginal preparation |
| ES2362604B1 (es) * | 2009-12-22 | 2012-06-28 | Bcn Peptides, S.A. | Formulación tópica oftálmica de péptidos. |
| UA123856C2 (uk) * | 2010-03-11 | 2021-06-16 | Уайт Елелсі | Фармацевтичні композиції метилналтрексону та натрію додецилсульфату для перорального введення |
| JP5222917B2 (ja) * | 2010-09-21 | 2013-06-26 | 財團法人工業技術研究院 | 徐放性組成物およびその製造方法 |
| TWI501781B (zh) * | 2010-12-10 | 2015-10-01 | Ind Tech Res Inst | 可控制釋放的組合物及其製造方法 |
| US10046058B2 (en) | 2014-12-02 | 2018-08-14 | Rezolute, Inc. | Use of hydrophobic organic acids to increase hydrophobicity of proteins and protein conjugates |
| US20190224275A1 (en) | 2017-05-12 | 2019-07-25 | Aurinia Pharmaceuticals Inc. | Protocol for treatment of lupus nephritis |
| US20190117573A1 (en) * | 2017-10-19 | 2019-04-25 | Hyalo Technologies, LLC | Composition and method of preparation of risperidone extended release preparation |
| US20230062487A1 (en) * | 2020-01-24 | 2023-03-02 | W. L. Gore & Associates, Inc. | Sustained-release matrices for adventitial or periadventitial neural ablation and uses thereof |
| CN111643483B (zh) * | 2020-07-06 | 2022-03-29 | 济南大学 | 一种用于制备加兰他敏缓释微球的方法 |
| US11992559B2 (en) | 2021-02-24 | 2024-05-28 | Oakwood Laboratories, Llc | Microsphere formulations comprising lurasidone and methods for making and using the same |
| WO2022226534A2 (en) * | 2021-04-23 | 2022-10-27 | Oakwood Laboratories, Llc | Microsphere formulations comprising multiple non-identical peptides and methods for making the same |
| CA3236685A1 (en) * | 2021-11-18 | 2023-05-25 | Inventage Lab Inc. | Method for preparing microparticles containing poorly soluble drugs |
| US20250009644A1 (en) * | 2021-12-02 | 2025-01-09 | University Of Connecticut | Long-acting injectable in situ forming biodegradable implants comprising non-steroidal anti-inflammatory drugs |
| CN116421578A (zh) * | 2023-03-31 | 2023-07-14 | 辉粒药业(苏州)有限公司 | 生长抑素类似物缓释微球及其制备方法 |
| AU2024253395A1 (en) * | 2023-04-03 | 2025-10-02 | Ferring B.V. | Methods of manufacturing peptide salts |
Family Cites Families (59)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3664963A (en) | 1969-10-22 | 1972-05-23 | Balchem Corp | Encapsulation process |
| US3780195A (en) | 1969-10-22 | 1973-12-18 | Balchem Corp | Encapsulation process |
| DE2059494B2 (de) | 1970-12-03 | 1972-03-16 | Licentia Gmbh | Biegsamer hohlleiter |
| JPS523342B2 (https=) | 1972-01-26 | 1977-01-27 | ||
| US3865352A (en) | 1973-11-16 | 1975-02-11 | Minnesota Mining & Mfg | Static mixing device |
| DE2604832A1 (de) | 1976-02-07 | 1977-08-11 | Basf Ag | Verfahren zur analyse von loesungen |
| US4171981A (en) | 1977-04-29 | 1979-10-23 | The Mead Corporation | Process for the production of hot melt coating compositions containing microcapsules |
| US4183681A (en) | 1978-05-19 | 1980-01-15 | Exxon Research & Engineering Co. | Emulsion preparation method using a packed tube emulsifier |
| US4299501A (en) | 1979-08-10 | 1981-11-10 | Ortho Pharmaceutical Corporation | Continuous process for the preparation of semisolid dispersions |
| US4384975A (en) * | 1980-06-13 | 1983-05-24 | Sandoz, Inc. | Process for preparation of microspheres |
| US4933105A (en) | 1980-06-13 | 1990-06-12 | Sandoz Pharm. Corp. | Process for preparation of microspheres |
| US4389330A (en) | 1980-10-06 | 1983-06-21 | Stolle Research And Development Corporation | Microencapsulation process |
| US4897268A (en) | 1987-08-03 | 1990-01-30 | Southern Research Institute | Drug delivery system and method of making the same |
| GB2209937B (en) | 1987-09-21 | 1991-07-03 | Depiopharm S A | Water insoluble polypeptides |
| DE3732370A1 (de) | 1987-09-25 | 1989-04-06 | Hoechst Ag | Verfahren zur vermischung von lebenden zellen oder mikroorganismen mit einer viskosen fluessigkeit und mischungen, die nach diesem verfahren hergestellt wurden |
| WO1990013361A1 (en) | 1989-05-04 | 1990-11-15 | Southern Research Institute | Improved encapsulation process and products therefrom |
| PH30995A (en) | 1989-07-07 | 1997-12-23 | Novartis Inc | Sustained release formulations of water soluble peptides. |
| US5112604A (en) * | 1989-09-01 | 1992-05-12 | Riker Laboratories, Inc. | Oral suspension formulation |
| MY107937A (en) * | 1990-02-13 | 1996-06-29 | Takeda Chemical Industries Ltd | Prolonged release microcapsules. |
| US6120805A (en) * | 1990-04-06 | 2000-09-19 | Rhone-Poulenc Rorer Sa | Microspheres, process for their preparation and their use |
| FR2660556B1 (fr) | 1990-04-06 | 1994-09-16 | Rhone Poulenc Sante | Microspheres, leur procede de preparation et leur utilisation. |
| US5733566A (en) | 1990-05-15 | 1998-03-31 | Alkermes Controlled Therapeutics Inc. Ii | Controlled release of antiparasitic agents in animals |
| NZ260909A (en) | 1993-07-05 | 1995-04-27 | Takeda Chemical Industries Ltd | Production of sustained release preparation by allowing a water-soluble polypeptide to permeate into a biodegradable matrix in an aqueous solution |
| CA2474701C (en) | 1993-11-19 | 2009-01-27 | Alkermes Controlled Therapeutics Inc. Ii | Preparation of biodegradeable microparticles containing a biologically active agent |
| JP2832143B2 (ja) | 1993-12-28 | 1998-12-02 | 信越化学工業株式会社 | シリコーン微粒子およびその製造方法 |
| WO1997004747A1 (en) | 1995-07-27 | 1997-02-13 | Dunn James M | Drug delivery systems for macromolecular drugs |
| US5629277A (en) * | 1995-10-04 | 1997-05-13 | William L. Brown | Paint removing composition |
| US6140040A (en) | 1995-10-06 | 2000-10-31 | Advanced Minerals Corporation | Method of mechanically separating microparticles suspended in fluids using particulate media |
| EP0799616A1 (en) | 1996-04-01 | 1997-10-08 | Takeda Chemical Industries, Ltd. | Oral composition comprising a fumagillol derivative |
| AU5678398A (en) * | 1997-01-29 | 1998-08-18 | Takeda Chemical Industries Ltd. | Sustained-release microspheres, their production and use |
| JPH10273447A (ja) | 1997-01-29 | 1998-10-13 | Takeda Chem Ind Ltd | 徐放性マイクロスフィア、その製造法および用途 |
| SE9701161D0 (sv) * | 1997-03-27 | 1997-03-27 | Karolinska Innovations Ab | New use I |
| AR012448A1 (es) | 1997-04-18 | 2000-10-18 | Ipsen Pharma Biotech | Composicion en forma de microcapsulas o de implantes que comprende un excipiente biodegradable, polimero o co-polimero, o una mezcla de talesexcipientes, y una sustancia activa o una mezcla de sustancias activas, procedimiento para la preparacion de una sustancia soluble en agua de elevada |
| ES2175668T3 (es) | 1997-12-16 | 2002-11-16 | Chiron Corp | Uso de microparticulas combinadas con emulsiones de aceite en agua submicronicas. |
| CA2316273A1 (en) | 1998-01-16 | 1999-07-22 | Takeda Chemical Industries, Ltd. | Sustained-release composition, method of its production and use thereof |
| US6270700B1 (en) * | 1998-07-23 | 2001-08-07 | Societe De Conseils De Recherches Et D'applications Scientifiques, Sas | Encapsulation of water soluble peptides |
| JP3012608B1 (ja) | 1998-09-17 | 2000-02-28 | 農林水産省食品総合研究所長 | マイクロチャネル装置及び同装置を用いたエマルションの製造方法 |
| US6194006B1 (en) * | 1998-12-30 | 2001-02-27 | Alkermes Controlled Therapeutics Inc. Ii | Preparation of microparticles having a selected release profile |
| EP1044683A1 (en) * | 1999-04-15 | 2000-10-18 | Debio Recherche Pharmaceutique S.A. | One-step dispersion method for the microencapsulation of water soluble substances |
| US6291013B1 (en) | 1999-05-03 | 2001-09-18 | Southern Biosystems, Inc. | Emulsion-based processes for making microparticles |
| US7919119B2 (en) | 1999-05-27 | 2011-04-05 | Acusphere, Inc. | Porous drug matrices and methods of manufacture thereof |
| AU7853500A (en) | 1999-10-08 | 2001-04-23 | Procter & Gamble Company, The | Apparatus and process for in-line preparation of hipes |
| AUPQ529000A0 (en) * | 2000-01-28 | 2000-02-17 | Research Laboratories Of Australia Pty Ltd | Toner characterization cell |
| US6953593B2 (en) | 2000-02-01 | 2005-10-11 | Lipoprotein Technologies, Inc. | Sustained-release microencapsulated delivery system |
| US6264987B1 (en) | 2000-05-19 | 2001-07-24 | Alkermes Controlled Therapeutics Inc. Ii | Method for preparing microparticles having a selected polymer molecular weight |
| US6306423B1 (en) | 2000-06-02 | 2001-10-23 | Allergan Sales, Inc. | Neurotoxin implant |
| JP2002126043A (ja) * | 2000-07-17 | 2002-05-08 | Takeda Chem Ind Ltd | 凍結乾燥物の製造法 |
| US6565873B1 (en) | 2000-10-25 | 2003-05-20 | Salvona Llc | Biodegradable bioadhesive controlled release system of nano-particles for oral care products |
| ES2382636T3 (es) * | 2000-10-31 | 2012-06-12 | Surmodics Pharmaceuticals, Inc. | Método para producir composiciones para la administración mejorada de moléculas bioactivas |
| EP1352269A2 (en) | 2001-01-15 | 2003-10-15 | 3M Innovative Properties Company | Multilayer infrared reflecting film with high and smooth transmission in visible wavelength region and laminate articles made therefrom |
| WO2002058672A2 (en) | 2001-01-26 | 2002-08-01 | Debio Recherche Pharmaceutique S.A. | Microparticles of biodegradable polymer encapsulating a biologically active substance |
| AR034641A1 (es) | 2001-06-29 | 2004-03-03 | Takeda Pharmaceutical | Composicion de liberacion controlada y metodo para producirla |
| US20060083778A1 (en) | 2002-05-03 | 2006-04-20 | Dean Allison | Controlled release compositions of estradiol metabolites |
| US20100143485A1 (en) * | 2003-03-05 | 2010-06-10 | Hudnut Paul S | Oxycontin controlled release formulations and methods of using same |
| EP2548550A1 (en) | 2003-04-10 | 2013-01-23 | Surmodics Pharmaceuticals, Inc. | Emulsion-based micro particles |
| US20070207211A1 (en) | 2003-04-10 | 2007-09-06 | Pr Pharmaceuticals, Inc. | Emulsion-based microparticles and methods for the production thereof |
| CA2521381C (en) | 2003-04-11 | 2020-05-26 | Rezolute, Inc. | Method for preparation of site-specific protein conjugates |
| JP5165239B2 (ja) | 2003-07-15 | 2013-03-21 | ピーアール ファーマシューティカルズ， インコーポレイテッド | 制御放出処方物の調製のための方法 |
| WO2005009357A2 (en) | 2003-07-23 | 2005-02-03 | Pr Pharmaceuticals, Inc. | Controlled release compositions |
-
2004
- 2004-07-15 JP JP2006520347A patent/JP5165239B2/ja not_active Expired - Fee Related
- 2004-07-15 WO PCT/US2004/022816 patent/WO2005009356A2/en not_active Ceased
- 2004-07-15 EP EP04778360.0A patent/EP1651136B1/en not_active Expired - Lifetime
- 2004-07-15 EP EP11187402A patent/EP2462896A1/en not_active Withdrawn
- 2004-07-15 ES ES04778360.0T patent/ES2625343T3/es not_active Expired - Lifetime
- 2004-07-15 US US10/564,494 patent/US8871269B2/en active Active
- 2004-07-15 CN CN200480026606.7A patent/CN1852687B/zh not_active Expired - Fee Related
- 2004-07-15 CN CN2012104691508A patent/CN102935069A/zh active Pending
- 2004-07-15 AU AU2004259208A patent/AU2004259208B2/en not_active Ceased
- 2004-07-15 CA CA2532302A patent/CA2532302C/en not_active Expired - Fee Related
- 2004-07-15 BR BRPI0412059-0A patent/BRPI0412059A/pt not_active IP Right Cessation
-
2011
- 2011-04-27 JP JP2011100206A patent/JP2011144207A/ja active Pending
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