JP2007516278A5 - - Google Patents

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Publication number
JP2007516278A5
JP2007516278A5 JP2006546881A JP2006546881A JP2007516278A5 JP 2007516278 A5 JP2007516278 A5 JP 2007516278A5 JP 2006546881 A JP2006546881 A JP 2006546881A JP 2006546881 A JP2006546881 A JP 2006546881A JP 2007516278 A5 JP2007516278 A5 JP 2007516278A5
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JP
Japan
Prior art keywords
cisapride
pat
cns
moiety
unrestricted
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JP2006546881A
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English (en)
Japanese (ja)
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JP4740152B2 (ja
JP2007516278A (ja
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Publication date
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Priority claimed from PCT/NO2004/000399 external-priority patent/WO2005061483A2/en
Publication of JP2007516278A publication Critical patent/JP2007516278A/ja
Publication of JP2007516278A5 publication Critical patent/JP2007516278A5/ja
Application granted granted Critical
Publication of JP4740152B2 publication Critical patent/JP4740152B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2006546881A 2003-12-23 2004-12-23 末梢性５−ｈｔ受容体の修飾因子 Expired - Fee Related JP4740152B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DKPA200301924 2003-12-23
DKPA200301924 2003-12-23
PCT/NO2004/000399 WO2005061483A2 (en) 2003-12-23 2004-12-23 Modulators of peripheral 5-ht receptors

Publications (3)

Publication Number Publication Date
JP2007516278A JP2007516278A (ja) 2007-06-21
JP2007516278A5 true JP2007516278A5 (enExample) 2008-08-14
JP4740152B2 JP4740152B2 (ja) 2011-08-03

Family

ID=34707211

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006546881A Expired - Fee Related JP4740152B2 (ja) 2003-12-23 2004-12-23 末梢性５−ｈｔ受容体の修飾因子

Country Status (10)

Country Link
US (1) US7834010B2 (enExample)
EP (1) EP1701951B1 (enExample)
JP (1) JP4740152B2 (enExample)
AT (1) ATE457309T1 (enExample)
AU (1) AU2004303722B2 (enExample)
CA (1) CA2551171C (enExample)
DE (1) DE602004025508D1 (enExample)
DK (1) DK1701951T3 (enExample)
ES (1) ES2340855T3 (enExample)
WO (1) WO2005061483A2 (enExample)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0211230D0 (en) 2002-05-16 2002-06-26 Medinnova Sf Treatment of heart failure
EP1902044A1 (en) * 2005-07-07 2008-03-26 Bio Medisinsk Innovasjon AS 5-htx modulators
WO2007010390A1 (en) 2005-07-22 2007-01-25 Pfizer Japan Inc. Indazolecarboxamide derivatives as 5ht4 receptor agonists
ITMI20062230A1 (it) * 2006-11-22 2008-05-23 Acraf Composto 2-alchil-indazolico procedimento per preparalo e composizione farmaceutica che lo comprende
SI2610258T1 (sl) 2007-10-19 2014-12-31 Boehringer Ingelheim International Gmbh Substituirani piperidino-dihidrotienopirimidini
UA99927C2 (uk) * 2007-11-12 2012-10-25 Ацьенде Кимике Риуните Анджелини Франческо А.Чи.Р.А.Ф. С.П.А. Медикамент, який є активним при невропатичному болі
US8642772B2 (en) 2008-10-14 2014-02-04 Sk Biopharmaceuticals Co., Ltd. Piperidine compounds, pharmaceutical composition comprising the same and its use
JP2012519160A (ja) 2009-02-27 2012-08-23 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｐｄｅ４阻害剤及びｎｓａｉｄを含有する組み合わせ薬
GB0905641D0 (en) 2009-04-01 2009-05-13 Serodus As Compounds
AU2010340142B2 (en) * 2009-12-17 2014-05-08 Merck Sharp & Dohme Corp. Quinoline amide M1 receptor positive allosteric modulators
WO2011124525A1 (de) 2010-04-08 2011-10-13 Boehringer Ingelheim International Gmbh Arnzeimittelkombinationen enthaltend pde4-inhibitoren und ep4-rezeptor-antagonisten
DK2976337T3 (en) * 2013-03-20 2018-07-16 Suven Life Sciences Ltd 5-amino-quinoline-8-carboxamide derivatives as 5-HT4 receptor agonists
EA029951B1 (ru) * 2013-12-16 2018-06-29 Сувен Лайф Сайенсиз Лимитед Соединения индазола в качестве агонистов 5-ht-рецептора
WO2016029218A1 (en) * 2014-08-22 2016-02-25 The Arizona Board Of Regents On Behalf Of The University Of Arizona Substituted 1-arylethyl-4-acylaminopiperidine derivatives as opioid/alpha-adrenoreceptor modulators and method of their preparation
CN111606837A (zh) * 2020-06-15 2020-09-01 千辉药业（安徽）有限责任公司 一种维格列汀的合成方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4494547A (en) 1981-03-30 1985-01-22 North Carolina Central University 2H-isoindolediones, their synthesis and use as radiosensitizers
RU2104279C1 (ru) 1992-03-12 1998-02-10 Смитклайн Бичам Плс Конденсированное индольное производное или его фармацевтически приемлемая соль, фармацевтическая композиция, проявляющая активность антагониста 5-нт*004-рецептора
HU218698B (hu) * 1994-09-27 2000-11-28 Janssen Pharmaceutica N.V. Gyógyászati hatású N-szubsztituált piperidinil-(biciklusos benzoát)-származékok, intermedierjeik, előállításuk és alkalmazásuk
US6147093A (en) 1996-07-19 2000-11-14 Sepracor Inc. Methods for treating gastroesophageal reflux disease
US20010031751A1 (en) 1997-12-05 2001-10-18 Smithkline Beecham P.L.C. Pharmaceuticals
JPH11292846A (ja) 1998-02-10 1999-10-26 Hokuriku Seiyaku Co Ltd ベンズアミド誘導体及びそれを含有する医薬
AR022338A1 (es) 1999-02-04 2002-09-04 Hokuriku Pharmaceutical Un compuesto de benzamida, medicamento que lo contiene, y uso para la manufactura de un medicamento para el tratamiento o prevencion de una enfermedad digestiva o para mejorar la movilidad del tracto gastrointestinal.
JP3398111B2 (ja) * 1999-02-04 2003-04-21 北陸製薬株式会社 ベンズアミド誘導体及びそれを含有する医薬
US6552046B2 (en) 2000-06-07 2003-04-22 Aryx Therapeutics Materials and methods for the treatment of gastroesophageal reflux disease
US6552004B1 (en) 2000-10-30 2003-04-22 Universite De Montreal Delivery system for entrapping charged macromolecules and a method for preparing same
US6598534B2 (en) 2001-06-04 2003-07-29 Raytheon Company Warhead with aligned projectiles
US6624163B2 (en) 2001-11-29 2003-09-23 Hoffman-La Roche Inc. Benzothiazole derivatives

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