JP2007509058A5 - - Google Patents

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Publication number
JP2007509058A5
JP2007509058A5 JP2006535367A JP2006535367A JP2007509058A5 JP 2007509058 A5 JP2007509058 A5 JP 2007509058A5 JP 2006535367 A JP2006535367 A JP 2006535367A JP 2006535367 A JP2006535367 A JP 2006535367A JP 2007509058 A5 JP2007509058 A5 JP 2007509058A5
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JP
Japan
Prior art keywords
lower alkyl
cancer
compound
halo
hydrogen
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JP2006535367A
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English (en)
Japanese (ja)
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JP4755991B2 (ja
JP2007509058A (ja
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Priority claimed from PCT/US2004/034179 external-priority patent/WO2005037273A1/en
Publication of JP2007509058A publication Critical patent/JP2007509058A/ja
Publication of JP2007509058A5 publication Critical patent/JP2007509058A5/ja
Application granted granted Critical
Publication of JP4755991B2 publication Critical patent/JP4755991B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2006535367A 2003-10-16 2004-10-15 Ｒａｆキナーゼインヒビターとしての置換ベンゾアゾールおよびその使用 Expired - Fee Related JP4755991B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US51196603P 2003-10-16 2003-10-16
US60/511,966 2003-10-16
PCT/US2004/034179 WO2005037273A1 (en) 2003-10-16 2004-10-15 Substituted benzazoles and use thereof as inhibitors of raf kinase

Publications (3)

Publication Number Publication Date
JP2007509058A JP2007509058A (ja) 2007-04-12
JP2007509058A5 true JP2007509058A5 (cg-RX-API-DMAC7.html) 2007-11-15
JP4755991B2 JP4755991B2 (ja) 2011-08-24

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ID=34465300

Family Applications (1)

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JP2006535367A Expired - Fee Related JP4755991B2 (ja) 2003-10-16 2004-10-15 Ｒａｆキナーゼインヒビターとしての置換ベンゾアゾールおよびその使用

Country Status (16)

Country Link
US (3) US7423150B2 (cg-RX-API-DMAC7.html)
EP (1) EP1682126B1 (cg-RX-API-DMAC7.html)
JP (1) JP4755991B2 (cg-RX-API-DMAC7.html)
KR (1) KR20060118472A (cg-RX-API-DMAC7.html)
CN (1) CN1889951A (cg-RX-API-DMAC7.html)
AT (1) ATE435015T1 (cg-RX-API-DMAC7.html)
AU (1) AU2004281151A1 (cg-RX-API-DMAC7.html)
CA (1) CA2542653A1 (cg-RX-API-DMAC7.html)
DE (1) DE602004021838D1 (cg-RX-API-DMAC7.html)
ES (1) ES2327418T3 (cg-RX-API-DMAC7.html)
IL (1) IL174965A0 (cg-RX-API-DMAC7.html)
MX (1) MXPA06004236A (cg-RX-API-DMAC7.html)
PL (1) PL1682126T3 (cg-RX-API-DMAC7.html)
PT (1) PT1682126E (cg-RX-API-DMAC7.html)
TW (1) TW200526208A (cg-RX-API-DMAC7.html)
WO (1) WO2005037273A1 (cg-RX-API-DMAC7.html)

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JP5985401B2 (ja) 2010-03-09 2016-09-06 デイナ ファーバー キャンサー インスティチュート，インコーポレイテッド 第一の癌療法に対する耐性を現に有するか、または、そのような耐性を生じる患者において癌を診断および治療する方法
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US9408885B2 (en) 2011-12-01 2016-08-09 Vib Vzw Combinations of therapeutic agents for treating melanoma
US8969388B1 (en) * 2012-07-28 2015-03-03 Sunshine Lake Pharma Co., Ltd. Substituted pyrazolone compounds and methods of use
US9242969B2 (en) 2013-03-14 2016-01-26 Novartis Ag Biaryl amide compounds as kinase inhibitors
UY36294A (es) 2014-09-12 2016-04-29 Novartis Ag Compuestos y composiciones como inhibidores de quinasa
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KR102881316B1 (ko) 2019-05-13 2025-11-05 노파르티스 아게 암 치료를 위한 raf 억제제로서의 n-(3-(2-(2-하이드록시에톡시)-6-모르폴리노피리딘-4-일)-4-메틸페닐)-2 (트리플루오로메틸)이소니코틴아미드의 새로운 결정질 형태
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