JP2007506703A5 - - Google Patents

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Publication number
JP2007506703A5
JP2007506703A5 JP2006527374A JP2006527374A JP2007506703A5 JP 2007506703 A5 JP2007506703 A5 JP 2007506703A5 JP 2006527374 A JP2006527374 A JP 2006527374A JP 2006527374 A JP2006527374 A JP 2006527374A JP 2007506703 A5 JP2007506703 A5 JP 2007506703A5
Authority
JP
Japan
Prior art keywords
alkyl
optionally substituted
quinolinecarboxamide
hydrogen
alkoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2006527374A
Other languages
English (en)
Japanese (ja)
Other versions
JP2007506703A (ja
Filing date
Publication date
Priority claimed from GBGB0322722.0A external-priority patent/GB0322722D0/en
Application filed filed Critical
Publication of JP2007506703A publication Critical patent/JP2007506703A/ja
Publication of JP2007506703A5 publication Critical patent/JP2007506703A5/ja
Pending legal-status Critical Current

Links

JP2006527374A 2003-09-27 2004-09-23 Pde4阻害剤としての4−アミノキノリン−3−カルボキサミド誘導体 Pending JP2007506703A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0322722.0A GB0322722D0 (en) 2003-09-27 2003-09-27 Compounds
PCT/EP2004/010844 WO2005030212A1 (en) 2003-09-27 2004-09-23 4-aminoquinoline-3-carboxamide derivatives as pde4 inhibitors

Publications (2)

Publication Number Publication Date
JP2007506703A JP2007506703A (ja) 2007-03-22
JP2007506703A5 true JP2007506703A5 (enExample) 2007-09-20

Family

ID=29287002

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006527374A Pending JP2007506703A (ja) 2003-09-27 2004-09-23 Pde4阻害剤としての4−アミノキノリン−3−カルボキサミド誘導体

Country Status (10)

Country Link
US (1) US20080096884A1 (enExample)
EP (1) EP1673086B1 (enExample)
JP (1) JP2007506703A (enExample)
AR (1) AR045824A1 (enExample)
AT (1) ATE384530T1 (enExample)
DE (1) DE602004011548T2 (enExample)
ES (1) ES2298806T3 (enExample)
GB (1) GB0322722D0 (enExample)
TW (1) TW200526584A (enExample)
WO (1) WO2005030212A1 (enExample)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI328009B (en) * 2003-05-21 2010-08-01 Glaxo Group Ltd Quinoline derivatives as phosphodiesterase inhibitors
GB0601951D0 (en) 2006-01-31 2006-03-15 Novartis Ag Organic compounds
GB0605462D0 (en) * 2006-03-17 2006-04-26 Glaxo Group Ltd Novel compounds
US20100041662A1 (en) 2006-10-30 2010-02-18 Sandrine Ferrand Heterocyclic compounds as antiinflammatory agents
WO2009087224A1 (en) 2008-01-11 2009-07-16 Novartis Ag Pyrimidines as kinase inhibitors
JP2012513464A (ja) * 2008-12-23 2012-06-14 ザ トラスティーズ オブ コロンビア ユニヴァーシティ イン ザ シティ オブ ニューヨーク ホスホジエステラーゼ阻害剤及びその使用
CA2749403A1 (en) 2009-01-13 2010-09-02 Glaxo Group Limited Pyrimidinecarboxamide derivatives as inhibitors of syk kinase
AR081377A1 (es) 2010-05-10 2012-08-29 Gilead Sciences Inc Compuestos de pirazolopiridina bifuncionales
NZ603136A (en) 2010-05-10 2014-11-28 Gilead Sciences Inc Bifunctional quinoline derivatives
UY33597A (es) 2010-09-09 2012-04-30 Irm Llc Compuestos y composiciones como inhibidores de la trk
WO2012034095A1 (en) 2010-09-09 2012-03-15 Irm Llc Compounds and compositions as trk inhibitors
JP5959541B2 (ja) 2011-02-25 2016-08-02 ノバルティス アーゲー Trk阻害剤としてのピラゾロ[1,5−a]ピリジン
KR20150119370A (ko) 2013-02-19 2015-10-23 화이자 인코포레이티드 Cns 장애 및 다른 장애의 치료를 위한 pde4 동종효소의 억제제로서의 아자벤즈이미다졸 화합물
EP3172210B1 (en) 2014-07-24 2020-01-15 Pfizer Inc Pyrazolopyrimidine compounds
WO2016020786A1 (en) 2014-08-06 2016-02-11 Pfizer Inc. Imidazopyridazine compounds
MA41140A (fr) 2014-12-12 2017-10-17 Cancer Research Tech Ltd Dérivés de 2,4-dioxo-quinazoline-6-sulfonamide en tant qu'inhibiteurs de la parg
MA41179A (fr) 2014-12-19 2017-10-24 Cancer Research Tech Ltd Composés inhibiteurs de parg
KR20180086187A (ko) 2015-10-05 2018-07-30 더 트러스티이스 오브 콜롬비아 유니버시티 인 더 시티 오브 뉴욕 자가포식 유동의 활성체 및 포스포리파제 d 및 타우를 포함하는 단백질 응집물의 클리어런스 및 단백질질환의 치료
WO2023183850A1 (en) 2022-03-23 2023-09-28 Ideaya Biosciences, Inc. Piperazine substituted indazole compounds as inhibitors of parg
TW202430172A (zh) * 2023-01-17 2024-08-01 大陸商瑞石生物醫藥有限公司 Pde4抑制劑、其製備方法及其在醫藥上的應用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK0480052T3 (da) * 1990-03-28 1998-05-11 Otsuka Pharma Co Ltd Quinolinderivat, antiulcus-lægemiddel indeholdende derivatet og fremstilling af derivatet
US5834485A (en) * 1996-05-20 1998-11-10 Chiroscience Limited Quinoline sulfonamides and their therapeutic use
US6093732A (en) * 1997-12-22 2000-07-25 Pharmacia & Upjohn Company 4-hydroxyquinoline-3-carboxamides and hydrazides as antiviral agents
US6576644B2 (en) * 2000-09-06 2003-06-10 Bristol-Myers Squibb Co. Quinoline inhibitors of cGMP phosphodiesterase
SE0101675D0 (sv) * 2001-05-11 2001-05-11 Astrazeneca Ab Novel composition
JO2311B1 (en) * 2001-08-29 2005-09-12 ميرك فروست كندا ليمتد Alkyl inhibitors Ariel phosphodiesterase-4

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