JP2007500158A - Lxrアゴニストを用いる炎症性腸疾患の治療方法 - Google Patents
Lxrアゴニストを用いる炎症性腸疾患の治療方法 Download PDFInfo
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- JP2007500158A JP2007500158A JP2006521514A JP2006521514A JP2007500158A JP 2007500158 A JP2007500158 A JP 2007500158A JP 2006521514 A JP2006521514 A JP 2006521514A JP 2006521514 A JP2006521514 A JP 2006521514A JP 2007500158 A JP2007500158 A JP 2007500158A
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- A—HUMAN NECESSITIES
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- A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US49061403P | 2003-07-28 | 2003-07-28 | |
| PCT/EP2004/008426 WO2005013946A2 (en) | 2003-07-28 | 2004-07-27 | Methods of treatment inflammatory bowel with lxr agonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2007500158A true JP2007500158A (ja) | 2007-01-11 |
| JP2007500158A5 JP2007500158A5 (https=) | 2007-08-02 |
Family
ID=34135107
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006521514A Pending JP2007500158A (ja) | 2003-07-28 | 2004-07-27 | Lxrアゴニストを用いる炎症性腸疾患の治療方法 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US20060205819A1 (https=) |
| EP (1) | EP1653938A2 (https=) |
| JP (1) | JP2007500158A (https=) |
| WO (1) | WO2005013946A2 (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7247748B2 (en) | 2002-03-27 | 2007-07-24 | Smithkline Corporation | Amide compounds and methods of using the same |
| AU2003226094A1 (en) | 2002-03-27 | 2003-10-13 | Smithkline Beecham Corporation | Compounds and methods |
| EP1487776A4 (en) | 2002-03-27 | 2005-05-25 | Smithkline Beecham Corp | ACID COMPOUNDS AND ESTERS AND METHODS OF USE THEREOF |
| ATE453389T1 (de) | 2002-03-27 | 2010-01-15 | Smithkline Beecham Corp | Bestimmte pharmazeutisch wertvolle substituierte aminoalkyl-heterocyclen |
| CN109071516B (zh) | 2015-12-15 | 2021-08-31 | 阿斯利康(瑞典)有限公司 | 新颖的化合物 |
| WO2017182981A1 (en) | 2016-04-20 | 2017-10-26 | Washington University | Ppar agonist or lxr agonist for use in the treatment of systemic lupus erythematosus by modulation of lap activity |
| JP2020524660A (ja) | 2017-06-14 | 2020-08-20 | アストラゼネカ・アクチエボラーグAstrazeneca Aktiebolag | Ror−ガンマモジュレーターとして有用な2,3−ジヒドロイソインドール−1−カルボキサミド |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2000054759A2 (en) * | 1999-03-15 | 2000-09-21 | Tularik Inc. | Lxr modulators |
| WO2002024632A2 (en) * | 2000-09-18 | 2002-03-28 | Glaxo Group Limited | Substituted aminopropoxyaryl derivatives useful as agonists for lxr |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2004009091A1 (en) * | 2002-06-17 | 2004-01-29 | Glaxo Group Limited | Purine derivatives as liver x receptor agonists |
-
2004
- 2004-07-27 EP EP04763551A patent/EP1653938A2/en not_active Withdrawn
- 2004-07-27 JP JP2006521514A patent/JP2007500158A/ja active Pending
- 2004-07-27 US US10/566,637 patent/US20060205819A1/en not_active Abandoned
- 2004-07-27 WO PCT/EP2004/008426 patent/WO2005013946A2/en not_active Ceased
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2000054759A2 (en) * | 1999-03-15 | 2000-09-21 | Tularik Inc. | Lxr modulators |
| WO2002024632A2 (en) * | 2000-09-18 | 2002-03-28 | Glaxo Group Limited | Substituted aminopropoxyaryl derivatives useful as agonists for lxr |
Also Published As
| Publication number | Publication date |
|---|---|
| EP1653938A2 (en) | 2006-05-10 |
| WO2005013946A3 (en) | 2005-04-07 |
| US20060205819A1 (en) | 2006-09-14 |
| WO2005013946A2 (en) | 2005-02-17 |
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