JP2006519831A - テトラゾール及びオキサジアゾロン置換β−アミノ酸誘導体 - Google Patents

テトラゾール及びオキサジアゾロン置換β−アミノ酸誘導体 Download PDF

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JP2006519831A
JP2006519831A JP2006506264A JP2006506264A JP2006519831A JP 2006519831 A JP2006519831 A JP 2006519831A JP 2006506264 A JP2006506264 A JP 2006506264A JP 2006506264 A JP2006506264 A JP 2006506264A JP 2006519831 A JP2006519831 A JP 2006519831A
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tetrazol
pain
disorder
disorders
methyl
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JP2006519831A5 (enExample
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スー バータ ナンシー
ロイド コルブリ ノーマン
アンドリュー フダック Jr. レイモンド
クナップ リン クリスティン
ブラッドリー シュワーズ ジャコブ
ジョン ソーペ アンドリュー
ヨーガン ウストゥロウ デイヴィッド
ズ ジジアン
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ワーナー−ランバート カンパニー リミティド ライアビリティー カンパニー
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Publication of JP2006519831A publication Critical patent/JP2006519831A/ja
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D257/00Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04Five-membered rings
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    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C07D271/071,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical

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  • Health & Medical Sciences (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
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  • Reproductive Health (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Immunology (AREA)
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  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
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JP2006506264A 2003-03-07 2004-02-23 テトラゾール及びオキサジアゾロン置換β−アミノ酸誘導体 Withdrawn JP2006519831A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US45287103P 2003-03-07 2003-03-07
PCT/IB2004/000510 WO2004078734A1 (en) 2003-03-07 2004-02-23 TETRAZOLE AND OXADIAZOLONE SUBSTITUTED β-AMINO ACID DERIVATIVES

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JP2006519831A true JP2006519831A (ja) 2006-08-31
JP2006519831A5 JP2006519831A5 (enExample) 2007-03-01

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JP2006506264A Withdrawn JP2006519831A (ja) 2003-03-07 2004-02-23 テトラゾール及びオキサジアゾロン置換β−アミノ酸誘導体

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US (1) US7250433B2 (enExample)
EP (1) EP1603890A1 (enExample)
JP (1) JP2006519831A (enExample)
BR (1) BRPI0408110A (enExample)
CA (1) CA2518218A1 (enExample)
MX (1) MXPA05009504A (enExample)
WO (1) WO2004078734A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070066591A1 (en) * 2003-05-14 2007-03-22 Xiangping Qian Compounds, compositions, and methods
GB0521743D0 (en) * 2005-10-25 2005-11-30 Novartis Ag Organic compounds
AU2013216828B2 (en) 2012-02-09 2017-01-12 Novus International Inc. Functionalized polymer compositions
MX2015000395A (es) 2012-07-12 2015-04-10 Novus Int Inc Composiciones de matriz y capa para proteccion de bioactivos.

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4087544A (en) * 1974-12-21 1978-05-02 Warner-Lambert Company Treatment of cranial dysfunctions using novel cyclic amino acids
DE2460891C2 (de) * 1974-12-21 1982-09-23 Gödecke AG, 1000 Berlin 1-Aminomethyl-1-cycloalkanessigsäuren und deren Ester, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel
US6197819B1 (en) * 1990-11-27 2001-03-06 Northwestern University Gamma amino butyric acid analogs and optical isomers
WO1999008670A1 (en) 1997-08-20 1999-02-25 Guglietta, Antonio Gaba analogs to prevent and treat gastrointestinal damage
PL341291A1 (en) * 1997-12-16 2001-04-09 Warner Lambert Co 1-substituted derivatives of 1-aminomethyl-ccycloalkanes (gabapentin analogues), their production and application of them in treating neurological disorders
BR9814287A (pt) * 1997-12-16 2000-10-03 Warner Lambert Co "4(3)-aminometil-(tio)piran 4(3) substituìdo ou derivados da piperidina (= análogos da gabapentina), sua preparação e seu uso no tratamento de desordens neurológicas"
CN1210268C (zh) * 1997-12-16 2005-07-13 沃尼尔·朗伯公司 ((环)烷基取代的)-γ-氨基丁酸衍生物(=GABA类似物),其制备和在治疗神经病中的用途
EP1082306A1 (en) * 1998-05-26 2001-03-14 Warner-Lambert Company Conformationally constrained amino acid compounds having affinity for the alpha2delta subunit of a calcium channel
BR9913701A (pt) 1998-09-14 2001-06-05 Warner Lambert Co ácidos alquil pirrolidina-3-carboxìlicos ramificados
KR20040081478A (ko) 2002-01-31 2004-09-21 워너-램버트 캄파니 엘엘씨 이명을 치료하기 위한 알파 2 델타 리간드

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MXPA05009504A (es) 2005-10-18
US20050014804A1 (en) 2005-01-20
WO2004078734A8 (en) 2005-12-15
BRPI0408110A (pt) 2006-03-01
CA2518218A1 (en) 2004-09-16
EP1603890A1 (en) 2005-12-14
US7250433B2 (en) 2007-07-31
WO2004078734A1 (en) 2004-09-16

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