JP2006515849A5 - - Google Patents

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Publication number
JP2006515849A5
JP2006515849A5 JP2004561378A JP2004561378A JP2006515849A5 JP 2006515849 A5 JP2006515849 A5 JP 2006515849A5 JP 2004561378 A JP2004561378 A JP 2004561378A JP 2004561378 A JP2004561378 A JP 2004561378A JP 2006515849 A5 JP2006515849 A5 JP 2006515849A5
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JP
Japan
Prior art keywords
alkyl
heterocyclyl
aryl
alkoxy
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2004561378A
Other languages
English (en)
Japanese (ja)
Other versions
JP2006515849A (ja
JP4851094B2 (ja
Filing date
Publication date
Priority claimed from GBGB0229804.0A external-priority patent/GB0229804D0/en
Application filed filed Critical
Publication of JP2006515849A publication Critical patent/JP2006515849A/ja
Publication of JP2006515849A5 publication Critical patent/JP2006515849A5/ja
Application granted granted Critical
Publication of JP4851094B2 publication Critical patent/JP4851094B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2004561378A 2002-12-20 2003-12-19 アベルメクチンｂ１及び４”位又は４’−位にアルコキシメチル置換基を有するアベルメクチンｂ１モノサッカライド誘導体 Expired - Fee Related JP4851094B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0229804.0 2002-12-20
GBGB0229804.0A GB0229804D0 (en) 2002-12-20 2002-12-20 Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position
PCT/EP2003/014613 WO2004056844A1 (en) 2002-12-20 2003-12-19 Avermectin b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4”- or 4’-position

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2010286151A Division JP5302297B2 (ja) 2002-12-20 2010-12-22 ４”位又は４’−位にアルコキシメチル置換基を有するアベルメクチンｂ１及びアベルメクチンｂ１単糖誘導体

Publications (3)

Publication Number Publication Date
JP2006515849A JP2006515849A (ja) 2006-06-08
JP2006515849A5 true JP2006515849A5 (enExample) 2007-02-01
JP4851094B2 JP4851094B2 (ja) 2012-01-11

Family

ID=9950151

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2004561378A Expired - Fee Related JP4851094B2 (ja) 2002-12-20 2003-12-19 アベルメクチンｂ１及び４”位又は４’−位にアルコキシメチル置換基を有するアベルメクチンｂ１モノサッカライド誘導体
JP2010286151A Expired - Fee Related JP5302297B2 (ja) 2002-12-20 2010-12-22 ４”位又は４’−位にアルコキシメチル置換基を有するアベルメクチンｂ１及びアベルメクチンｂ１単糖誘導体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2010286151A Expired - Fee Related JP5302297B2 (ja) 2002-12-20 2010-12-22 ４”位又は４’−位にアルコキシメチル置換基を有するアベルメクチンｂ１及びアベルメクチンｂ１単糖誘導体

Country Status (22)

Country Link
US (3) US7737261B2 (enExample)
EP (1) EP1581546B1 (enExample)
JP (2) JP4851094B2 (enExample)
KR (1) KR101109500B1 (enExample)
CN (1) CN1738828B (enExample)
AR (1) AR042533A1 (enExample)
AU (1) AU2003302284B2 (enExample)
BR (1) BR0317601A (enExample)
CA (1) CA2507774C (enExample)
CO (1) CO5690647A1 (enExample)
ES (1) ES2742899T3 (enExample)
GB (1) GB0229804D0 (enExample)
IL (1) IL169092A (enExample)
MA (1) MA27646A1 (enExample)
MX (1) MXPA05006036A (enExample)
PE (1) PE20040713A1 (enExample)
PL (1) PL211483B1 (enExample)
RU (1) RU2330857C2 (enExample)
TW (1) TW200512214A (enExample)
UA (1) UA81281C2 (enExample)
WO (1) WO2004056844A1 (enExample)
ZA (1) ZA200504353B (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0229804D0 (en) * 2002-12-20 2003-01-29 Syngenta Participations Ag Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position
JP2010006703A (ja) * 2006-11-07 2010-01-14 Hokko Chem Ind Co Ltd アベルメクチンモノ配糖体誘導体
RU2453553C1 (ru) * 2011-05-11 2012-06-20 Игорь Викторович Заварзин 5-о-сукциноилавермектин, способ его получения и антипаразитарное средство на его основе
RU2472801C1 (ru) * 2011-05-11 2013-01-20 Игорь Викторович Заварзин 5-о-производные авермектина, способ их получения и антипаразитарные средства на их основе
CN103613625B (zh) * 2013-12-02 2016-03-02 兰州大学 一种阿维菌素类化合物及其制备方法和在农药中的用途
CN104402954A (zh) * 2014-11-28 2015-03-11 大庆志飞生物化工有限公司 甲胺基阿维菌素单糖化合物及其制备方法和用途
CN104402953B (zh) * 2014-11-28 2017-07-28 大庆志飞生物化工有限公司 阿维菌素单糖化合物及其制备方法和用途
JP6577184B2 (ja) 2014-12-24 2019-09-18 Ntn株式会社 転がり軸受
CN107501368B (zh) * 2017-09-30 2020-02-21 中国科学院成都生物研究所 一种多拉菌素衍生物的合成及其杀虫应用
CN113150053B (zh) * 2020-01-22 2024-10-01 华东理工大学 偶氮苯类阿维菌素衍生物及其制备方法和应用
CN113817008B (zh) * 2021-07-15 2023-05-23 湖州师范学院 新型琥珀酰基十六元大环内酯的制备方法及用途

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US87519A (en) * 1869-03-02 Improvement in furnace-stoves and registers
US18993A (en) * 1857-12-29 Cider-mill
US148520A (en) * 1874-03-10 Improvement in faucets
SE434277B (sv) * 1976-04-19 1984-07-16 Merck & Co Inc Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis
US4874749A (en) * 1987-07-31 1989-10-17 Merck & Co., Inc. 4"-Deoxy-4-N-methylamino avermectin Bla/Blb
GB8811037D0 (en) * 1988-05-10 1988-06-15 Glaxo Group Ltd Chemical compounds
EP0353959A2 (en) 1988-08-02 1990-02-07 Beecham Group Plc Antihelmintic macrolide antibiotics
SE465605B (sv) * 1990-02-26 1991-10-07 Harry Nilsson Skivfilter
JP2622197B2 (ja) * 1990-03-01 1997-06-18 三共株式会社 １３−エーテル置換ミルベマイシン誘導体
US5169839A (en) * 1990-05-11 1992-12-08 Merck & Co., Inc. Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections
US5262400A (en) * 1991-06-20 1993-11-16 Merck & Co., Inc. 4α-substituted avermectin derivatives
US5411737A (en) * 1991-10-15 1995-05-02 Merck & Co., Inc. Slow release syneresing polymeric drug delivery device
PL174488B1 (pl) * 1993-05-10 1998-08-31 Merck & Co Inc Preparat do zwalczania pasożytów zwierząt oraz sposób wytwarzania preparatu do zwalczania pasożytów zwierząt
US5602107A (en) * 1993-05-10 1997-02-11 Merck & Co., Inc. Pour-on formulations consisting of gylcols, glycerides and avermectin compounds
NZ273129A (en) * 1993-08-19 1996-08-27 Merck & Co Inc 4"-deoxy-4"-epi-methylamino avermectin b1a/b1b benzoic acid salt hemihydrate; pesticidal compositions
US5436355A (en) * 1994-02-03 1995-07-25 Merck & Co., Inc. Process for making avermectin/zein compositions
TW327125B (en) * 1994-02-07 1998-02-21 Merck & Co Inc Composition and method for protecting against pine exhausted
AU2001277712A1 (en) 2000-08-09 2002-02-18 The Kitasato Institute Avermectin derivatives
US20040087519A1 (en) 2000-08-09 2004-05-06 Satoshi Omura Avermectin derivatives
WO2003075742A2 (en) * 2002-03-05 2003-09-18 Merck & Co., Inc. Biomarker for efficacy of appetite suppressant drugs
GB0229804D0 (en) 2002-12-20 2003-01-29 Syngenta Participations Ag Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position

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