MA27646A1 - Derives d'avermectine b1 et d'avermectine b1 monosaccharidique ayant un substituant alcoxymethyle en position 4" ou 4' - Google Patents
Derives d'avermectine b1 et d'avermectine b1 monosaccharidique ayant un substituant alcoxymethyle en position 4" ou 4'Info
- Publication number
- MA27646A1 MA27646A1 MA28349A MA28349A MA27646A1 MA 27646 A1 MA27646 A1 MA 27646A1 MA 28349 A MA28349 A MA 28349A MA 28349 A MA28349 A MA 28349A MA 27646 A1 MA27646 A1 MA 27646A1
- Authority
- MA
- Morocco
- Prior art keywords
- alkyl
- compounds
- tautomer
- alkoxy
- relates
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 5
- 125000004400 (C1-C12) alkyl group Chemical group 0.000 abstract 4
- 125000006710 (C2-C12) alkenyl group Chemical group 0.000 abstract 2
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 125000004642 (C1-C12) alkoxy group Chemical group 0.000 abstract 1
- 125000004643 (C1-C12) haloalkoxy group Chemical group 0.000 abstract 1
- 125000006711 (C2-C12) alkynyl group Chemical group 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 125000005110 aryl thio group Chemical group 0.000 abstract 1
- 125000004104 aryloxy group Chemical group 0.000 abstract 1
- 125000000392 cycloalkenyl group Chemical group 0.000 abstract 1
- 125000000000 cycloalkoxy group Chemical group 0.000 abstract 1
- 125000005149 cycloalkylsulfinyl group Chemical group 0.000 abstract 1
- 125000005144 cycloalkylsulfonyl group Chemical group 0.000 abstract 1
- 125000005366 cycloalkylthio group Chemical group 0.000 abstract 1
- 125000004995 haloalkylthio group Chemical group 0.000 abstract 1
- 125000005347 halocycloalkyl group Chemical group 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 125000005844 heterocyclyloxy group Chemical group 0.000 abstract 1
- 239000000575 pesticide Substances 0.000 abstract 1
- 150000003839 salts Chemical group 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
- A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
- A01N43/22—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom rings with more than six members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Molecular Biology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Tropical Medicine & Parasitology (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0229804.0A GB0229804D0 (en) | 2002-12-20 | 2002-12-20 | Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA27646A1 true MA27646A1 (fr) | 2005-12-01 |
Family
ID=9950151
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA28349A MA27646A1 (fr) | 2002-12-20 | 2005-06-17 | Derives d'avermectine b1 et d'avermectine b1 monosaccharidique ayant un substituant alcoxymethyle en position 4" ou 4' |
Country Status (22)
| Country | Link |
|---|---|
| US (3) | US7737261B2 (enExample) |
| EP (1) | EP1581546B1 (enExample) |
| JP (2) | JP4851094B2 (enExample) |
| KR (1) | KR101109500B1 (enExample) |
| CN (1) | CN1738828B (enExample) |
| AR (1) | AR042533A1 (enExample) |
| AU (1) | AU2003302284B2 (enExample) |
| BR (1) | BR0317601A (enExample) |
| CA (1) | CA2507774C (enExample) |
| CO (1) | CO5690647A1 (enExample) |
| ES (1) | ES2742899T3 (enExample) |
| GB (1) | GB0229804D0 (enExample) |
| IL (1) | IL169092A (enExample) |
| MA (1) | MA27646A1 (enExample) |
| MX (1) | MXPA05006036A (enExample) |
| PE (1) | PE20040713A1 (enExample) |
| PL (1) | PL211483B1 (enExample) |
| RU (1) | RU2330857C2 (enExample) |
| TW (1) | TW200512214A (enExample) |
| UA (1) | UA81281C2 (enExample) |
| WO (1) | WO2004056844A1 (enExample) |
| ZA (1) | ZA200504353B (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0229804D0 (en) * | 2002-12-20 | 2003-01-29 | Syngenta Participations Ag | Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position |
| JP2010006703A (ja) * | 2006-11-07 | 2010-01-14 | Hokko Chem Ind Co Ltd | アベルメクチンモノ配糖体誘導体 |
| RU2453553C1 (ru) * | 2011-05-11 | 2012-06-20 | Игорь Викторович Заварзин | 5-о-сукциноилавермектин, способ его получения и антипаразитарное средство на его основе |
| RU2472801C1 (ru) * | 2011-05-11 | 2013-01-20 | Игорь Викторович Заварзин | 5-о-производные авермектина, способ их получения и антипаразитарные средства на их основе |
| CN103613625B (zh) * | 2013-12-02 | 2016-03-02 | 兰州大学 | 一种阿维菌素类化合物及其制备方法和在农药中的用途 |
| CN104402954A (zh) * | 2014-11-28 | 2015-03-11 | 大庆志飞生物化工有限公司 | 甲胺基阿维菌素单糖化合物及其制备方法和用途 |
| CN104402953B (zh) * | 2014-11-28 | 2017-07-28 | 大庆志飞生物化工有限公司 | 阿维菌素单糖化合物及其制备方法和用途 |
| JP6577184B2 (ja) | 2014-12-24 | 2019-09-18 | Ntn株式会社 | 転がり軸受 |
| CN107501368B (zh) * | 2017-09-30 | 2020-02-21 | 中国科学院成都生物研究所 | 一种多拉菌素衍生物的合成及其杀虫应用 |
| CN113150053B (zh) * | 2020-01-22 | 2024-10-01 | 华东理工大学 | 偶氮苯类阿维菌素衍生物及其制备方法和应用 |
| CN113817008B (zh) * | 2021-07-15 | 2023-05-23 | 湖州师范学院 | 新型琥珀酰基十六元大环内酯的制备方法及用途 |
Family Cites Families (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US18993A (en) * | 1857-12-29 | Cider-mill | ||
| US87519A (en) * | 1869-03-02 | Improvement in furnace-stoves and registers | ||
| US148520A (en) * | 1874-03-10 | Improvement in faucets | ||
| SE434277B (sv) * | 1976-04-19 | 1984-07-16 | Merck & Co Inc | Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis |
| US4874749A (en) * | 1987-07-31 | 1989-10-17 | Merck & Co., Inc. | 4"-Deoxy-4-N-methylamino avermectin Bla/Blb |
| GB8811037D0 (en) * | 1988-05-10 | 1988-06-15 | Glaxo Group Ltd | Chemical compounds |
| EP0353959A2 (en) | 1988-08-02 | 1990-02-07 | Beecham Group Plc | Antihelmintic macrolide antibiotics |
| SE465605B (sv) * | 1990-02-26 | 1991-10-07 | Harry Nilsson | Skivfilter |
| JP2622197B2 (ja) * | 1990-03-01 | 1997-06-18 | 三共株式会社 | １３−エーテル置換ミルベマイシン誘導体 |
| US5169839A (en) * | 1990-05-11 | 1992-12-08 | Merck & Co., Inc. | Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections |
| US5262400A (en) * | 1991-06-20 | 1993-11-16 | Merck & Co., Inc. | 4α-substituted avermectin derivatives |
| US5411737A (en) * | 1991-10-15 | 1995-05-02 | Merck & Co., Inc. | Slow release syneresing polymeric drug delivery device |
| US5602107A (en) * | 1993-05-10 | 1997-02-11 | Merck & Co., Inc. | Pour-on formulations consisting of gylcols, glycerides and avermectin compounds |
| PL174488B1 (pl) * | 1993-05-10 | 1998-08-31 | Merck & Co Inc | Preparat do zwalczania pasożytów zwierząt oraz sposób wytwarzania preparatu do zwalczania pasożytów zwierząt |
| BR9407300A (pt) * | 1993-08-19 | 1996-10-08 | Merck & Co Inc | Composto cristalino de sal de ácido benzóico de 4'-deóxi-4'-epi-metilamino avermectina B1A/B1B hemiidratado processo para a sua preparação e para o controle de insetos agrícolas e composição útil para o tratamento de infestações de plantas ou de produtos de plantas |
| US5436355A (en) * | 1994-02-03 | 1995-07-25 | Merck & Co., Inc. | Process for making avermectin/zein compositions |
| TW327125B (en) * | 1994-02-07 | 1998-02-21 | Merck & Co Inc | Composition and method for protecting against pine exhausted |
| CA2418968C (en) | 2000-08-09 | 2009-11-24 | The Kitasato Institute | Avermectin derivatives |
| WO2002012248A1 (en) | 2000-08-09 | 2002-02-14 | The Kitasato Institute | Avermectin derivatives |
| WO2003075742A2 (en) * | 2002-03-05 | 2003-09-18 | Merck & Co., Inc. | Biomarker for efficacy of appetite suppressant drugs |
| GB0229804D0 (en) | 2002-12-20 | 2003-01-29 | Syngenta Participations Ag | Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position |
-
2002
- 2002-12-20 GB GBGB0229804.0A patent/GB0229804D0/en not_active Ceased
-
2003
- 2003-12-12 PE PE2003001284A patent/PE20040713A1/es active IP Right Grant
- 2003-12-18 AR ARP030104712A patent/AR042533A1/es active IP Right Grant
- 2003-12-18 TW TW092135927A patent/TW200512214A/zh unknown
- 2003-12-19 WO PCT/EP2003/014613 patent/WO2004056844A1/en not_active Ceased
- 2003-12-19 AU AU2003302284A patent/AU2003302284B2/en not_active Ceased
- 2003-12-19 KR KR1020057011622A patent/KR101109500B1/ko not_active Expired - Fee Related
- 2003-12-19 US US10/539,274 patent/US7737261B2/en active Active
- 2003-12-19 UA UAA200507209A patent/UA81281C2/uk unknown
- 2003-12-19 MX MXPA05006036A patent/MXPA05006036A/es active IP Right Grant
- 2003-12-19 RU RU2005122943/04A patent/RU2330857C2/ru active
- 2003-12-19 ES ES03810843T patent/ES2742899T3/es not_active Expired - Lifetime
- 2003-12-19 CN CN2003801088575A patent/CN1738828B/zh not_active Expired - Lifetime
- 2003-12-19 CA CA2507774A patent/CA2507774C/en not_active Expired - Fee Related
- 2003-12-19 EP EP03810843.7A patent/EP1581546B1/en not_active Expired - Lifetime
- 2003-12-19 JP JP2004561378A patent/JP4851094B2/ja not_active Expired - Fee Related
- 2003-12-19 PL PL377497A patent/PL211483B1/pl unknown
- 2003-12-19 BR BR0317601-0A patent/BR0317601A/pt not_active Application Discontinuation
-
2005
- 2005-06-09 IL IL169092A patent/IL169092A/en active IP Right Grant
- 2005-06-17 CO CO05059203A patent/CO5690647A1/es not_active Application Discontinuation
- 2005-06-17 MA MA28349A patent/MA27646A1/fr unknown
-
2006
- 2006-01-06 ZA ZA200504353A patent/ZA200504353B/en unknown
-
2010
- 2010-04-27 US US12/768,280 patent/US8017589B2/en not_active Expired - Fee Related
- 2010-12-22 JP JP2010286151A patent/JP5302297B2/ja not_active Expired - Fee Related
-
2011
- 2011-05-27 US US13/117,292 patent/US8263566B2/en not_active Expired - Fee Related
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| MA27646A1 (fr) | Derives d'avermectine b1 et d'avermectine b1 monosaccharidique ayant un substituant alcoxymethyle en position 4" ou 4' | |
| CA2545644A1 (en) | Melanocortin receptor agonists | |
| BR0212893A (pt) | Derivados de 4-pirimidona-3-substituìdo | |
| DE50202573D1 (en) | Pyrazolylsubstituierte thienyloxy-pyridine | |
| MA30024B1 (fr) | 5-arylisoxazolines pour lutter contre des parasites invertebres | |
| MA30428B1 (fr) | Derives de dihydropyrazolopyrimidinones | |
| MXPA05012033A (es) | Compuesto de pirimidina y composicion para el control de plagas que contiene el mismo. | |
| MD3864B2 (en) | Cyanoanthranilamide compounds, compositions on base thereof and method for invertebrate pest control | |
| CA2453609A1 (en) | Bridged piperidine derivatives as melanocortin receptor agonists | |
| MD4157B1 (en) | Isoxazolines for controlling invertebrate pests | |
| DK1427720T3 (da) | 3-substitueret-4-pyrimidonderivater | |
| ID25649A (id) | Turunan-turunan sikloalkena, produksi serta penggunaannya | |
| MA31785B1 (fr) | Nouveaux dérivés d'imidazole | |
| ES2367820T3 (es) | Derivados de la pirimidina y sus usos como pesticidas. | |
| NO308734B1 (no) | Oksimetere, mellomprodukter til bruk ved fremstilling derav, mikrobicid blanding inneholdende eterene og anvendelse av eterene | |
| MA31784B1 (fr) | Nouveaux dérivés d'imidazole | |
| TW200510444A (en) | Avermectins substituted in the 4" and 4'-positions having pesticidal properties | |
| RU2004109165A (ru) | Производные 4"-дезокси-4-(s)-аминоавермектина | |
| TNSN07043A1 (fr) | Oxazolidinones contenant des oxindoles, servant d'agents antibacteriens | |
| TW200420574A (en) | Avermectin-and avermectin monosaccharide derivatives substituted in the 4"-or 4'-position having pesticidal properties | |
| MA27275A1 (fr) | Derives de 4"-desoxy-4"-(s)-amidoavermectine | |
| KR910014357A (ko) | 신규 치환 β-피리미디닐옥시(티오)-및 β-트리아지닐옥시(티오) 시클로알칸카르복실산 유도체, 그의 제조 방법, 및 제초제, 살균제 및 식물 성장 조절제로서의 용도 | |
| HU202056B (en) | Acaricidal composition comprising 2,3-diamino-maleic acid-nitryl-azomethine derivatives and process for producing such compounds | |
| BR9403269A (pt) | Composto processo para a preparação do mesmo composição fungicida e processo para combater fungos | |
| JPH0827120A (ja) | テトラヒドロピリミジノン誘導体 |