JP2006508107A5 - - Google Patents

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Publication number
JP2006508107A5
JP2006508107A5 JP2004550489A JP2004550489A JP2006508107A5 JP 2006508107 A5 JP2006508107 A5 JP 2006508107A5 JP 2004550489 A JP2004550489 A JP 2004550489A JP 2004550489 A JP2004550489 A JP 2004550489A JP 2006508107 A5 JP2006508107 A5 JP 2006508107A5
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Japan
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compound
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composition
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JP2004550489A
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English (en)
Japanese (ja)
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JP2006508107A (ja
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Priority claimed from PCT/US2003/035188 external-priority patent/WO2004041810A1/en
Publication of JP2006508107A publication Critical patent/JP2006508107A/ja
Publication of JP2006508107A5 publication Critical patent/JP2006508107A5/ja
Pending legal-status Critical Current

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JP2004550489A 2002-11-05 2003-11-05 Ｊａｋおよび他のプロテインキナーゼのインヒビターとして有用な化合物 Pending JP2006508107A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US42404302P 2002-11-05 2002-11-05
PCT/US2003/035188 WO2004041810A1 (en) 2002-11-05 2003-11-05 Compounds useful as inhibitors of jak and other protein kinases

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2010139840A Division JP2010195838A (ja) 2002-11-05 2010-06-18 Ｊａｋおよび他のプロテインキナーゼのインヒビターとして有用な化合物

Publications (2)

Publication Number Publication Date
JP2006508107A JP2006508107A (ja) 2006-03-09
JP2006508107A5 true JP2006508107A5 (https=) 2006-08-31

Family

ID=32312743

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2004550489A Pending JP2006508107A (ja) 2002-11-05 2003-11-05 Ｊａｋおよび他のプロテインキナーゼのインヒビターとして有用な化合物
JP2010139840A Pending JP2010195838A (ja) 2002-11-05 2010-06-18 Ｊａｋおよび他のプロテインキナーゼのインヒビターとして有用な化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2010139840A Pending JP2010195838A (ja) 2002-11-05 2010-06-18 Ｊａｋおよび他のプロテインキナーゼのインヒビターとして有用な化合物

Country Status (6)

Country Link
US (1) US7348335B2 (https=)
EP (1) EP1560824A1 (https=)
JP (2) JP2006508107A (https=)
AU (2) AU2003286895A1 (https=)
CA (1) CA2507406A1 (https=)
WO (1) WO2004041810A1 (https=)

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WO2009107391A1 (ja) * 2008-02-27 2009-09-03 武田薬品工業株式会社 ６員芳香環含有化合物
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TWI729644B (zh) 2014-06-12 2021-06-01 美商西爾拉癌症醫學公司 N-(氰基甲基)-4-(2-(4-𠰌啉基苯基胺基)嘧啶-4-基)苯甲醯胺
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WO2018041989A1 (en) 2016-09-02 2018-03-08 INSERM (Institut National de la Santé et de la Recherche Médicale) Methods for diagnosing and treating refractory celiac disease type 2
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CN114761006A (zh) 2019-11-08 2022-07-15 Inserm(法国国家健康医学研究院) 对激酶抑制剂产生耐药性的癌症的治疗方法
WO2021148581A1 (en) 2020-01-22 2021-07-29 Onxeo Novel dbait molecule and its use
CN113549018B (zh) * 2020-04-24 2024-02-27 中国药科大学 蛋白激酶抑制剂及其衍生物，制备方法、药物组合物和应用
CN115403516B (zh) * 2021-08-03 2024-01-26 河南省儿童医院郑州儿童医院 含3,4,5-三取代基苯环的芳杂环化合物、药物组合物及其制备方法和应用
CN115703760B (zh) * 2021-08-11 2024-05-31 山东大学 2,4-二取代嘧啶类细胞周期蛋白依赖性激酶酶抑制剂及其制备方法和应用
TW202333718A (zh) * 2022-02-03 2023-09-01 美商奈可薩斯醫藥有限公司 芳基烴受體促效劑及其用途
WO2023222565A1 (en) 2022-05-16 2023-11-23 Institut National de la Santé et de la Recherche Médicale Methods for assessing the exhaustion of hematopoietic stems cells induced by chronic inflammation
WO2024051702A1 (zh) * 2022-09-05 2024-03-14 浙江同源康医药股份有限公司 用作cdk4激酶抑制剂的化合物及其应用
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