JP2005532289A5 - - Google Patents
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- Publication number
- JP2005532289A5 JP2005532289A5 JP2003583385A JP2003583385A JP2005532289A5 JP 2005532289 A5 JP2005532289 A5 JP 2005532289A5 JP 2003583385 A JP2003583385 A JP 2003583385A JP 2003583385 A JP2003583385 A JP 2003583385A JP 2005532289 A5 JP2005532289 A5 JP 2005532289A5
- Authority
- JP
- Japan
- Prior art keywords
- polymer
- sustained release
- hydrophobic polymer
- hydrophobic
- hydrophilic polymer
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 229920001600 hydrophobic polymer Polymers 0.000 claims description 9
- 229920001477 hydrophilic polymer Polymers 0.000 claims description 7
- 230000002459 sustained Effects 0.000 claims description 6
- 239000011248 coating agent Substances 0.000 claims description 4
- 238000000576 coating method Methods 0.000 claims description 4
- 239000007939 sustained release tablet Substances 0.000 claims 1
- 239000001856 Ethyl cellulose Substances 0.000 description 4
- ZZSNKZQZMQGXPY-UHFFFAOYSA-N Ethyl cellulose Chemical compound CCOCC1OC(OC)C(OCC)C(OCC)C1OC1C(O)C(O)C(OC)C(CO)O1 ZZSNKZQZMQGXPY-UHFFFAOYSA-N 0.000 description 4
- 235000019325 ethyl cellulose Nutrition 0.000 description 4
- 229920001249 ethyl cellulose Polymers 0.000 description 4
- 239000003795 chemical substances by application Substances 0.000 description 2
- QOWAMIUFBNBINS-UHFFFAOYSA-N 2-[6-[4,5-diethoxy-2-(ethoxymethyl)-6-methoxyoxan-3-yl]oxy-4,5-dimethoxy-2-(methoxymethyl)oxan-3-yl]oxy-6-(hydroxymethyl)-5-methoxyoxane-3,4-diol Chemical compound CCOCC1OC(OC)C(OCC)C(OCC)C1OC1C(OC)C(OC)C(OC2C(C(O)C(OC)C(CO)O2)O)C(COC)O1 QOWAMIUFBNBINS-UHFFFAOYSA-N 0.000 description 1
- 239000001761 ethyl methyl cellulose Substances 0.000 description 1
- 235000010944 ethyl methyl cellulose Nutrition 0.000 description 1
- 229920000609 methyl cellulose Polymers 0.000 description 1
- 239000001923 methylcellulose Substances 0.000 description 1
- 235000010981 methylcellulose Nutrition 0.000 description 1
Description
上記徐放剤は疎水性ポリマーを含むことができる。上記疎水性ポリマーはエチルセルロースを含むことができる。
上記徐放性コーティングは疎水性ポリマー及び親水性ポリマーを含むことができる。上記疎水性ポリマーはエチルセルロースを含むことができ、上記親水性ポリマーはメチルセルロースを含むことができる。
上記徐放性コーティングはエチルセルロース及びメチルセルロースを含むことができ、上記徐放剤はエチルセルロースを含むことができる。
上記徐放性コーティングの疎水性ポリマー及び親水性ポリマーは、疎水性ポリマー対親水性ポリマーの重量比55-65:45-35、好ましくは疎水性ポリマー対親水性ポリマーの重量比57:43で存在することができる。
上記徐放性コーティングは疎水性ポリマー及び親水性ポリマーを含むことができる。上記疎水性ポリマーはエチルセルロースを含むことができ、上記親水性ポリマーはメチルセルロースを含むことができる。
上記徐放性コーティングはエチルセルロース及びメチルセルロースを含むことができ、上記徐放剤はエチルセルロースを含むことができる。
上記徐放性コーティングの疎水性ポリマー及び親水性ポリマーは、疎水性ポリマー対親水性ポリマーの重量比55-65:45-35、好ましくは疎水性ポリマー対親水性ポリマーの重量比57:43で存在することができる。
Claims (1)
- 当該徐放性コーティングの疎水性ポリマー及び親水性ポリマーが、当該疎水性ポリマー対当該親水性ポリマーの重量比57:43で存在する、請求項7に記載の徐放性錠剤。
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10/120,501 US7125563B2 (en) | 2002-04-12 | 2002-04-12 | Sustained release pharmaceutical preparations and methods for producing the same |
PCT/US2003/009210 WO2003086364A1 (en) | 2002-04-12 | 2003-04-11 | Sustained release pharmaceutical prepartations and methods for producing the same |
Publications (2)
Publication Number | Publication Date |
---|---|
JP2005532289A JP2005532289A (ja) | 2005-10-27 |
JP2005532289A5 true JP2005532289A5 (ja) | 2006-06-01 |
Family
ID=29214431
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2003583385A Pending JP2005532289A (ja) | 2002-04-12 | 2003-04-11 | 持続放出性医薬製剤及びその製造方法 |
Country Status (10)
Country | Link |
---|---|
US (3) | US7125563B2 (ja) |
EP (1) | EP1494653A1 (ja) |
JP (1) | JP2005532289A (ja) |
CN (1) | CN1655765A (ja) |
AU (1) | AU2003218397A1 (ja) |
CA (1) | CA2481667A1 (ja) |
HR (1) | HRP20040945A2 (ja) |
PL (1) | PL373328A1 (ja) |
RU (1) | RU2004133532A (ja) |
WO (1) | WO2003086364A1 (ja) |
Families Citing this family (19)
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ES2272914T3 (es) * | 2003-05-20 | 2007-05-01 | Ethypharm | Composicion farmaceutica oral de liberacion sostenida. |
US8802139B2 (en) | 2003-06-26 | 2014-08-12 | Intellipharmaceutics Corp. | Proton pump-inhibitor-containing capsules which comprise subunits differently structured for a delayed release of the active ingredient |
US8394409B2 (en) | 2004-07-01 | 2013-03-12 | Intellipharmaceutics Corp. | Controlled extended drug release technology |
US10624858B2 (en) | 2004-08-23 | 2020-04-21 | Intellipharmaceutics Corp | Controlled release composition using transition coating, and method of preparing same |
US10064828B1 (en) | 2005-12-23 | 2018-09-04 | Intellipharmaceutics Corp. | Pulsed extended-pulsed and extended-pulsed pulsed drug delivery systems |
CA2645855C (en) | 2006-03-16 | 2015-02-03 | Tris Pharma, Inc. | Modified release formulations containing drug-ion exchange resin complexes |
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US10960077B2 (en) | 2006-05-12 | 2021-03-30 | Intellipharmaceutics Corp. | Abuse and alcohol resistant drug composition |
WO2009147665A1 (en) * | 2008-06-02 | 2009-12-10 | Dexcel Ltd | Process for manufacture of a medicament with granulation and pan coating |
WO2011102506A1 (ja) * | 2010-02-22 | 2011-08-25 | 第一三共株式会社 | 経口用徐放性固形製剤 |
EP2540318B1 (en) | 2010-02-22 | 2018-10-24 | Daiichi Sankyo Company, Limited | Sustained-release solid preparation for oral use |
US8623409B1 (en) | 2010-10-20 | 2014-01-07 | Tris Pharma Inc. | Clonidine formulation |
KR102127625B1 (ko) | 2012-09-03 | 2020-06-29 | 다이이찌 산쿄 가부시키가이샤 | 하이드로모르폰염산염 함유의 경구용 서방성 의약 조성물 |
US11590228B1 (en) | 2015-09-08 | 2023-02-28 | Tris Pharma, Inc | Extended release amphetamine compositions |
US9949964B2 (en) * | 2016-09-07 | 2018-04-24 | Saniona A/S | Tesofensine compositions |
US11590081B1 (en) | 2017-09-24 | 2023-02-28 | Tris Pharma, Inc | Extended release amphetamine tablets |
US11918689B1 (en) | 2020-07-28 | 2024-03-05 | Tris Pharma Inc | Liquid clonidine extended release composition |
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-
2002
- 2002-04-12 US US10/120,501 patent/US7125563B2/en not_active Expired - Fee Related
-
2003
- 2003-04-11 EP EP03714395A patent/EP1494653A1/en not_active Withdrawn
- 2003-04-11 CN CNA038115018A patent/CN1655765A/zh active Pending
- 2003-04-11 PL PL03373328A patent/PL373328A1/xx not_active Application Discontinuation
- 2003-04-11 RU RU2004133532/15A patent/RU2004133532A/ru not_active Application Discontinuation
- 2003-04-11 WO PCT/US2003/009210 patent/WO2003086364A1/en active Application Filing
- 2003-04-11 CA CA002481667A patent/CA2481667A1/en not_active Abandoned
- 2003-04-11 JP JP2003583385A patent/JP2005532289A/ja active Pending
- 2003-04-11 AU AU2003218397A patent/AU2003218397A1/en not_active Abandoned
-
2004
- 2004-10-11 HR HR20040945A patent/HRP20040945A2/hr not_active Application Discontinuation
-
2006
- 2006-01-17 US US11/332,158 patent/US20060105037A1/en not_active Abandoned
-
2008
- 2008-01-09 US US11/971,741 patent/US20080107730A1/en not_active Abandoned
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